CN1917882A - 非典型抗精神病药物与促肾上腺皮质激素释放因子拮抗剂的治疗剂组合 - Google Patents
非典型抗精神病药物与促肾上腺皮质激素释放因子拮抗剂的治疗剂组合 Download PDFInfo
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- CN1917882A CN1917882A CNA2005800049430A CN200580004943A CN1917882A CN 1917882 A CN1917882 A CN 1917882A CN A2005800049430 A CNA2005800049430 A CN A2005800049430A CN 200580004943 A CN200580004943 A CN 200580004943A CN 1917882 A CN1917882 A CN 1917882A
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- alkyl
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- Health & Medical Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54473104P | 2004-02-13 | 2004-02-13 | |
| US60/544,731 | 2004-02-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1917882A true CN1917882A (zh) | 2007-02-21 |
Family
ID=34886075
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA2005800049430A Pending CN1917882A (zh) | 2004-02-13 | 2005-02-01 | 非典型抗精神病药物与促肾上腺皮质激素释放因子拮抗剂的治疗剂组合 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20050209250A1 (https=) |
| EP (1) | EP1718311A1 (https=) |
| JP (1) | JP2007522200A (https=) |
| KR (1) | KR20060110006A (https=) |
| CN (1) | CN1917882A (https=) |
| AU (1) | AU2005215257A1 (https=) |
| BR (1) | BRPI0507609A (https=) |
| CA (1) | CA2556160A1 (https=) |
| IL (1) | IL177433A0 (https=) |
| NO (1) | NO20064054L (https=) |
| RU (1) | RU2006129307A (https=) |
| TW (1) | TW200538128A (https=) |
| WO (1) | WO2005079807A1 (https=) |
| ZA (1) | ZA200606636B (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI568448B (zh) * | 2010-01-07 | 2017-02-01 | 阿艾克麥斯製藥愛爾蘭有限公司 | 四級銨鹽前藥 |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050171088A1 (en) * | 2004-01-30 | 2005-08-04 | Astrazeneca Ab | Treatment of psychoses with dibenzothiazepine antipsychotic |
| EP2170399A1 (en) * | 2007-06-05 | 2010-04-07 | Synthon B.V. | Intranasal administration of asenapine and pharmaceutical compositions therefor |
| AU2008337286B2 (en) * | 2007-12-19 | 2014-08-07 | Cancer Research Technology Limited | Pyrido[2,3-b]pyrazine-8-substituted compounds and their use |
| US20100298397A1 (en) * | 2009-05-19 | 2010-11-25 | Singh Nikhilesh N | Method of treatment of obsessive compulsive disorder with ondansetron |
| CA2937222C (en) | 2009-06-25 | 2019-06-04 | Alkermes Pharma Ireland Limited | Prodrugs of nh-acidic compounds |
| LT2445502T (lt) | 2009-06-25 | 2017-09-25 | Alkermes Pharma Ireland Limited | Heterocikliniai junginiai, skirti neurologinių ir fiziologinių susirgimų gydymui |
| WO2011084849A1 (en) * | 2010-01-07 | 2011-07-14 | Alkermes, Inc. | Diaryldiazepine prodrugs for the treatment of neurological and psychological disorders |
| WO2011084848A2 (en) | 2010-01-07 | 2011-07-14 | Alkermes, Inc. | Prodrugs of heteraromatic compounds |
| AU2011270701B2 (en) | 2010-06-24 | 2015-05-14 | Alkermes Pharma Ireland Limited | Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives |
| US20120302616A1 (en) * | 2010-12-03 | 2012-11-29 | Nikhilesh Singh | Method of treatment of obsessive compulsive disorder with ondansetron |
| BR112013023847B1 (pt) | 2011-03-18 | 2021-02-23 | Alkermes Pharma Ireland Limited | composições farmacêuticas compreendendo ésteres de sorbitano e uso das mesmas |
| NZ722096A (en) | 2011-12-15 | 2016-11-25 | Alkermes Pharma Ireland Ltd | Prodrugs of secondary amine compounds |
| AU2013235526B2 (en) | 2012-03-19 | 2017-11-30 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising benzyl alcohol |
| AU2013235523B9 (en) | 2012-03-19 | 2018-01-04 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising glycerol esters |
| CA2867121C (en) | 2012-03-19 | 2021-05-25 | Alkermes Pharma Ireland Limited | Pharmaceutical compositions comprising fatty acid esters |
| JP6654042B2 (ja) | 2012-09-19 | 2020-02-26 | アルカームス ファーマ アイルランド リミテッド | 貯蔵安定性が改善された医薬組成物 |
| US20140206667A1 (en) | 2012-11-14 | 2014-07-24 | Michela Gallagher | Methods and compositions for treating schizophrenia |
| WO2015112642A1 (en) | 2014-01-21 | 2015-07-30 | Neurocrine Biosciences, Inc. | Crf1 receptor antagonists for the treatment of congenital adrenal hyperplasia |
| CN106132415A (zh) | 2014-03-20 | 2016-11-16 | 奥克梅斯制药爱尔兰有限公司 | 具有增加的注射速度的阿立哌唑制剂 |
| EP3510029B1 (en) * | 2016-09-07 | 2025-11-05 | The Regents of The University of California | Allosteric corticotropin-releasing factor receptor 1 (crfr1) antagonists that decrease p-tau and improve cognition |
| WO2018115010A1 (en) | 2016-12-20 | 2018-06-28 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system containing asenapine and polysiloxane or polyisobutylene |
| ES2769286T3 (es) | 2016-12-20 | 2020-06-25 | Lts Lohmann Therapie Systeme Ag | Sistema terapéutico transdérmico que contiene asenapina |
| ES2881783T3 (es) | 2017-06-26 | 2021-11-30 | Lts Lohmann Therapie Systeme Ag | Sistema terapéutico transdérmico que contiene asenapina y polímero de acrílico y silicona |
| WO2019032720A1 (en) | 2017-08-09 | 2019-02-14 | Sanford Burnham Prebys Medical Discovery Institute | APELIN RECEPTOR AGONISTS AND METHODS OF USE |
| CN118845788A (zh) | 2017-08-14 | 2024-10-29 | 云杉生物科学公司 | 促肾上腺皮质激素释放因子受体拮抗剂 |
| EP3761983A1 (en) | 2018-03-05 | 2021-01-13 | Alkermes Pharma Ireland Limited | Aripiprazole dosing strategy |
| EP4438124A3 (en) | 2018-04-27 | 2024-12-18 | Spruce Biosciences, Inc. | Methods for treating testicular and ovarian adrenal rest tumors |
| CN112533593A (zh) | 2018-06-20 | 2021-03-19 | 罗曼治疗系统股份公司 | 含有阿塞那平的透皮治疗系统 |
| CA3101420A1 (en) | 2018-06-20 | 2019-12-26 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system containing asenapine |
| CA3121920A1 (en) | 2018-12-07 | 2020-06-11 | Neurocrine Biosciences, Inc. | Crf1 receptor antagonist, pharmaceutical formulations and solid forms thereof for the treatment of congenital adrenal hyperplasia |
| JP7623365B2 (ja) | 2019-09-27 | 2025-01-28 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | Crf受容体アンタゴニストおよび使用方法 |
| BR112023002497A2 (pt) | 2020-08-12 | 2023-05-02 | Spruce Biosciences Inc | Métodos e composições para tratamento da síndrome dos ovários policísticos |
| WO2022173333A2 (en) * | 2021-02-10 | 2022-08-18 | Gero Pte. Ltd. | Compounds, compositions and methods for treating age-related diseases and conditions |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL7605526A (nl) * | 1976-05-24 | 1977-11-28 | Akzo Nv | Nieuwe tetracyclische derivaten. |
| TW530047B (en) * | 1994-06-08 | 2003-05-01 | Pfizer | Corticotropin releasing factor antagonists |
| TW477787B (en) * | 1996-08-27 | 2002-03-01 | Pfizer | Pyrido six-membered nitrogen-containing cyclic ring derivatives having corticotropin releasing factor antagonist activity and pharmaceutical composition containing same |
| IL127497A (en) * | 1997-12-18 | 2002-07-25 | Pfizer Prod Inc | Medicinal products containing piperazinyl-heterocyclic compounds for the treatment of psychiatric disorders |
| EP1040831A3 (en) * | 1999-04-02 | 2003-05-02 | Pfizer Products Inc. | Use of corticotropin releasing factor (CRF) antagonists to prevent sudden death |
| US6432989B1 (en) * | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
-
2005
- 2005-02-01 WO PCT/IB2005/000251 patent/WO2005079807A1/en not_active Ceased
- 2005-02-01 EP EP05702400A patent/EP1718311A1/en not_active Withdrawn
- 2005-02-01 CA CA002556160A patent/CA2556160A1/en not_active Abandoned
- 2005-02-01 RU RU2006129307/15A patent/RU2006129307A/ru not_active Application Discontinuation
- 2005-02-01 BR BRPI0507609-9A patent/BRPI0507609A/pt not_active IP Right Cessation
- 2005-02-01 AU AU2005215257A patent/AU2005215257A1/en not_active Abandoned
- 2005-02-01 CN CNA2005800049430A patent/CN1917882A/zh active Pending
- 2005-02-01 JP JP2006552710A patent/JP2007522200A/ja active Pending
- 2005-02-01 KR KR1020067018643A patent/KR20060110006A/ko not_active Ceased
- 2005-02-05 TW TW094103864A patent/TW200538128A/zh unknown
- 2005-02-14 US US11/058,329 patent/US20050209250A1/en not_active Abandoned
-
2006
- 2006-08-10 IL IL177433A patent/IL177433A0/en unknown
- 2006-08-10 ZA ZA200606636A patent/ZA200606636B/en unknown
- 2006-09-08 NO NO20064054A patent/NO20064054L/no not_active Application Discontinuation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI568448B (zh) * | 2010-01-07 | 2017-02-01 | 阿艾克麥斯製藥愛爾蘭有限公司 | 四級銨鹽前藥 |
Also Published As
| Publication number | Publication date |
|---|---|
| NO20064054L (no) | 2006-11-10 |
| CA2556160A1 (en) | 2005-09-01 |
| IL177433A0 (en) | 2006-12-10 |
| RU2006129307A (ru) | 2008-02-20 |
| JP2007522200A (ja) | 2007-08-09 |
| KR20060110006A (ko) | 2006-10-23 |
| TW200538128A (en) | 2005-12-01 |
| AU2005215257A1 (en) | 2005-09-01 |
| WO2005079807A1 (en) | 2005-09-01 |
| ZA200606636B (en) | 2008-01-30 |
| BRPI0507609A (pt) | 2007-07-03 |
| EP1718311A1 (en) | 2006-11-08 |
| US20050209250A1 (en) | 2005-09-22 |
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