CN116693447B - 酮酰胺类衍生物及其制药用途 - Google Patents
酮酰胺类衍生物及其制药用途 Download PDFInfo
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- CN116693447B CN116693447B CN202310131329.0A CN202310131329A CN116693447B CN 116693447 B CN116693447 B CN 116693447B CN 202310131329 A CN202310131329 A CN 202310131329A CN 116693447 B CN116693447 B CN 116693447B
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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| EP4488264A4 (en) * | 2022-03-01 | 2026-03-04 | Westvac Biopharma Co Ltd | CETO AMIDE DERIVATIVES AND THEIR PHARMACEUTICAL USE |
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| WO2023165334A1 (zh) * | 2022-03-01 | 2023-09-07 | 成都威斯克生物医药有限公司 | 酮酰胺类衍生物及其制药用途 |
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| CN115698035A (zh) * | 2020-04-10 | 2023-02-03 | 共晶制药公司 | 诺如病毒及冠状病毒复制的抑制剂 |
| PH12022553378A1 (en) * | 2020-06-10 | 2024-03-25 | Univ Leuven Kath | Anti-viral compounds for treating coronavirus, picornavirus, and norovirus infections |
| CN115960088B (zh) * | 2020-07-31 | 2024-07-26 | 四川大学 | 一种新型冠状病毒主蛋白酶的抑制剂及其制备方法和用途 |
| CN114057702B (zh) * | 2020-07-31 | 2022-09-30 | 四川大学 | 一种新型冠状病毒主蛋白酶的抑制剂及其制备方法和用途 |
| US20240083885A1 (en) * | 2020-12-04 | 2024-03-14 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Compositions and methods for inhibiting m pro protease activity and for preventing and treating sars-cov-2 infection |
| WO2022265577A2 (en) * | 2021-06-15 | 2022-12-22 | Agency For Science, Technology And Research | Coronavirus enzyme modulators, methods of synthesis and uses thereof |
| JP2023000996A (ja) * | 2021-06-18 | 2023-01-04 | ラクオリア創薬株式会社 | プロテアーゼ阻害剤としてのケトアミド誘導体 |
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2023
- 2023-02-15 EP EP23762735.1A patent/EP4488264A4/en active Pending
- 2023-02-15 JP JP2023580943A patent/JP2025507472A/ja active Pending
- 2023-02-15 WO PCT/CN2023/076078 patent/WO2023165334A1/zh not_active Ceased
- 2023-02-15 US US18/723,545 patent/US20250064789A1/en active Pending
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| CN116693447A (zh) | 2023-09-05 |
| WO2023165334A1 (zh) | 2023-09-07 |
| EP4488264A4 (en) | 2026-03-04 |
| JP2025507472A (ja) | 2025-03-21 |
| US20250064789A1 (en) | 2025-02-27 |
| EP4488264A1 (en) | 2025-01-08 |
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