CN116600807A - 包含噻吩并吡啶结构的驱虫化合物 - Google Patents

包含噻吩并吡啶结构的驱虫化合物 Download PDF

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Publication number
CN116600807A
CN116600807A CN202180083153.5A CN202180083153A CN116600807A CN 116600807 A CN116600807 A CN 116600807A CN 202180083153 A CN202180083153 A CN 202180083153A CN 116600807 A CN116600807 A CN 116600807A
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CN
China
Prior art keywords
alkyl
hydrogen
alkoxy
independently selected
group
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CN202180083153.5A
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English (en)
Chinese (zh)
Inventor
M·贝格
M·林德
C·施耐德
J·丹兹勒
U·桑德恩
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Intervet International BV
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Intervet International BV
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Publication of CN116600807A publication Critical patent/CN116600807A/zh
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D497/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CN202180083153.5A 2020-12-11 2021-12-10 包含噻吩并吡啶结构的驱虫化合物 Pending CN116600807A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20213297.3 2020-12-11
EP20213297 2020-12-11
PCT/EP2021/085125 WO2022122988A1 (en) 2020-12-11 2021-12-10 Anthelmintic compounds comprising a thienopyridine structure

Publications (1)

Publication Number Publication Date
CN116600807A true CN116600807A (zh) 2023-08-15

Family

ID=73834196

Family Applications (1)

Application Number Title Priority Date Filing Date
CN202180083153.5A Pending CN116600807A (zh) 2020-12-11 2021-12-10 包含噻吩并吡啶结构的驱虫化合物

Country Status (8)

Country Link
US (1) US20240043446A1 (https=)
EP (1) EP4259636A1 (https=)
JP (1) JP2023553428A (https=)
CN (1) CN116600807A (https=)
AU (1) AU2021395477A1 (https=)
CA (1) CA3203279A1 (https=)
MX (1) MX2023006744A (https=)
WO (1) WO2022122988A1 (https=)

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CA3133100A1 (en) 2019-03-19 2020-09-24 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic aza-benzothiophene and aza-benzofuran compounds
KR20230028268A (ko) 2020-05-29 2023-02-28 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 헤테로시클릭 화합물
UY39995A (es) 2021-11-01 2023-05-15 Boehringer Ingelheim Vetmedica GmbH Compuestos de pirrolopiridazina como antihelmínticos
WO2024213752A1 (en) 2023-04-14 2024-10-17 Elanco Animal Health Gmbh Long-term prevention and/or treatment of a disease by slo-1 inhibitors
WO2026078157A2 (en) 2024-10-10 2026-04-16 Elanco Animal Health Gmbh Slo-1 modulators for prevention and/or treatment of a disease

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* Cited by examiner, † Cited by third party
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US5378679A (en) * 1992-08-21 1995-01-03 Basf Aktiengesellschaft Heteroaromatically condensed hydroxypyridonecarboxamides, their preparation and use
CN102413693A (zh) * 2009-05-04 2012-04-11 杜邦公司 磺酰胺杀线虫剂
CN109071545A (zh) * 2016-04-15 2018-12-21 拜耳动物保健有限责任公司 新的吡唑并嘧啶衍生物
CN110582503A (zh) * 2017-04-24 2019-12-17 拜耳公司 作为有害物防治剂的稠合双环杂环化合物衍生物
WO2020131629A1 (en) * 2018-12-18 2020-06-25 Elanco Tiergesundheit Ag Bicyclic derivatives

Also Published As

Publication number Publication date
AU2021395477A1 (en) 2023-06-22
EP4259636A1 (en) 2023-10-18
WO2022122988A1 (en) 2022-06-16
JP2023553428A (ja) 2023-12-21
CA3203279A1 (en) 2022-06-16
MX2023006744A (es) 2023-06-19
US20240043446A1 (en) 2024-02-08
AU2021395477A9 (en) 2024-10-31

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