AU2021395477A1 - Anthelmintic compounds comprising a thienopyridine structure - Google Patents

Anthelmintic compounds comprising a thienopyridine structure Download PDF

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Publication number
AU2021395477A1
AU2021395477A1 AU2021395477A AU2021395477A AU2021395477A1 AU 2021395477 A1 AU2021395477 A1 AU 2021395477A1 AU 2021395477 A AU2021395477 A AU 2021395477A AU 2021395477 A AU2021395477 A AU 2021395477A AU 2021395477 A1 AU2021395477 A1 AU 2021395477A1
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AU
Australia
Prior art keywords
alkyl
hydrogen
alkoxy
independently selected
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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AU2021395477A
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English (en)
Other versions
AU2021395477A9 (en
Inventor
Michael Berger
Michael Linder
Carolin SCHNEIDER
Ulrich Sondern
Janina TÄNZLER
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Intervet International BV
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Intervet International BV
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Publication date
Application filed by Intervet International BV filed Critical Intervet International BV
Publication of AU2021395477A1 publication Critical patent/AU2021395477A1/en
Publication of AU2021395477A9 publication Critical patent/AU2021395477A9/en
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D497/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
AU2021395477A 2020-12-11 2021-12-10 Anthelmintic compounds comprising a thienopyridine structure Pending AU2021395477A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20213297 2020-12-11
EP20213297.3 2020-12-11
PCT/EP2021/085125 WO2022122988A1 (en) 2020-12-11 2021-12-10 Anthelmintic compounds comprising a thienopyridine structure

Publications (2)

Publication Number Publication Date
AU2021395477A1 true AU2021395477A1 (en) 2023-06-22
AU2021395477A9 AU2021395477A9 (en) 2024-10-31

Family

ID=73834196

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2021395477A Pending AU2021395477A1 (en) 2020-12-11 2021-12-10 Anthelmintic compounds comprising a thienopyridine structure

Country Status (8)

Country Link
US (1) US20240043446A1 (https=)
EP (1) EP4259636A1 (https=)
JP (1) JP2023553428A (https=)
CN (1) CN116600807A (https=)
AU (1) AU2021395477A1 (https=)
CA (1) CA3203279A1 (https=)
MX (1) MX2023006744A (https=)
WO (1) WO2022122988A1 (https=)

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KR20230028268A (ko) 2020-05-29 2023-02-28 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 헤테로시클릭 화합물
US11999742B2 (en) 2021-11-01 2024-06-04 Boehringer Ingelheim Vetmedica Gmbh Substituted pyrrolo[1,2-b]pyridazines as anthelmintics
WO2024213752A1 (en) 2023-04-14 2024-10-17 Elanco Animal Health Gmbh Long-term prevention and/or treatment of a disease by slo-1 inhibitors
WO2026078157A2 (en) 2024-10-10 2026-04-16 Elanco Animal Health Gmbh Slo-1 modulators for prevention and/or treatment of a disease

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Also Published As

Publication number Publication date
MX2023006744A (es) 2023-06-19
US20240043446A1 (en) 2024-02-08
EP4259636A1 (en) 2023-10-18
CA3203279A1 (en) 2022-06-16
JP2023553428A (ja) 2023-12-21
WO2022122988A1 (en) 2022-06-16
CN116600807A (zh) 2023-08-15
AU2021395477A9 (en) 2024-10-31

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