CN1157392C - 在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物 - Google Patents

在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物 Download PDF

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Publication number
CN1157392C
CN1157392C CNB988054132A CN98805413A CN1157392C CN 1157392 C CN1157392 C CN 1157392C CN B988054132 A CNB988054132 A CN B988054132A CN 98805413 A CN98805413 A CN 98805413A CN 1157392 C CN1157392 C CN 1157392C
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azabicyclo
oct
ene
methyl
thienyl
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Expired - Fee Related
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CN1257499A (zh
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D
D·彼得斯
�¶�ɭ
G·M·奥尔森
�������ɭ
S·F·尼尔森
E·O·尼尔森
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NTG Nordic Transport Group AS
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Neurosearch AS
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
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CNB988054132A 1997-05-30 1998-05-29 在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物 Expired - Fee Related CN1157392C (zh)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
DK62797 1997-05-30
DK0627/1997 1997-05-30
DK150297 1997-12-19
DK1502/1997 1997-12-19
DK0408/1998 1998-03-24
DK40898 1998-03-24
DK0534/1998 1998-04-16
DK53498 1998-04-16

Publications (2)

Publication Number Publication Date
CN1257499A CN1257499A (zh) 2000-06-21
CN1157392C true CN1157392C (zh) 2004-07-14

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CNB988054132A Expired - Fee Related CN1157392C (zh) 1997-05-30 1998-05-29 在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物

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US (2) US6645977B1 (enExample)
EP (1) EP0984965B1 (enExample)
JP (1) JP4447663B2 (enExample)
KR (1) KR100589872B1 (enExample)
CN (1) CN1157392C (enExample)
AT (1) ATE267199T1 (enExample)
AU (1) AU745964B2 (enExample)
BR (1) BR9809697A (enExample)
CA (1) CA2289574C (enExample)
CZ (1) CZ298824B6 (enExample)
DE (1) DE69823994T2 (enExample)
DK (1) DK0984965T3 (enExample)
EE (1) EE04057B1 (enExample)
HU (1) HUP0002713A3 (enExample)
IL (2) IL132437A0 (enExample)
IS (1) IS2092B (enExample)
NO (1) NO325513B1 (enExample)
NZ (1) NZ500642A (enExample)
RU (1) RU2186780C2 (enExample)
SK (1) SK284994B6 (enExample)
TR (1) TR199902942T2 (enExample)
WO (1) WO1998054181A1 (enExample)

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CA2289574C (en) 2007-04-24
DE69823994D1 (de) 2004-06-24
KR100589872B1 (ko) 2006-06-15
US20040019207A1 (en) 2004-01-29
SK284994B6 (sk) 2006-04-06
EP0984965A1 (en) 2000-03-15
CZ298824B6 (cs) 2008-02-20
RU2186780C2 (ru) 2002-08-10
IL132437A0 (en) 2001-03-19
ATE267199T1 (de) 2004-06-15
IS2092B (is) 2006-04-12
IS5243A (is) 1999-11-10
HK1027353A1 (en) 2001-01-12
NO995850L (no) 1999-11-29
NO995850D0 (no) 1999-11-29
EE9900529A (et) 2000-06-15
HUP0002713A3 (en) 2001-02-28
AU745964B2 (en) 2002-04-11
JP4447663B2 (ja) 2010-04-07
KR20010013154A (ko) 2001-02-26
CA2289574A1 (en) 1998-12-03
JP2002501514A (ja) 2002-01-15
HUP0002713A2 (hu) 2001-01-29
EP0984965B1 (en) 2004-05-19
DE69823994T2 (de) 2009-09-24
NO325513B1 (no) 2008-05-26
SK162699A3 (en) 2000-07-11
AU7426198A (en) 1998-12-30
IL132437A (en) 2006-12-10
CN1257499A (zh) 2000-06-21
US6964972B2 (en) 2005-11-15
CZ414799A3 (cs) 2000-02-16
EE04057B1 (et) 2003-06-16
TR199902942T2 (xx) 2000-04-21
US6645977B1 (en) 2003-11-11
BR9809697A (pt) 2000-07-11
WO1998054181A1 (en) 1998-12-03
DK0984965T3 (da) 2004-09-27

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