CN114728933B - 5-ht2a受体抑制剂或反向激动剂及其制备方法和应用 - Google Patents

5-ht2a受体抑制剂或反向激动剂及其制备方法和应用 Download PDF

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CN114728933B
CN114728933B CN202180006171.3A CN202180006171A CN114728933B CN 114728933 B CN114728933 B CN 114728933B CN 202180006171 A CN202180006171 A CN 202180006171A CN 114728933 B CN114728933 B CN 114728933B
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straight
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branched alkyl
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CN114728933A (zh
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张睿
叶亮
马明旭
王文艳
代玉森
田京伟
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Shandong Luye Pharmaceutical Co Ltd
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CN115605202B (zh) 2020-03-26 2025-10-28 盐野义制药株式会社 具有血清素受体结合活性的芳香族杂环衍生物
US20240083872A1 (en) * 2020-12-28 2024-03-14 Shionogi & Co., Ltd. Cyclic amine derivatives having serotonin receptor binding activity
AU2023319750A1 (en) * 2022-08-03 2025-02-13 Luye Innomind Pharma Shijiazhuang Co., Ltd. 5-ht2a receptor inverse agonist, and preparation method therefor and use thereof
CN115850204B (zh) * 2022-11-26 2024-01-19 烟台大学 四氢苯并噻吩衍生物及其制备方法和应用
WO2025162237A1 (zh) * 2024-02-02 2025-08-07 绿叶嘉奥制药石家庄有限公司 一种5-ht2a受体反向激动剂的盐型、晶型及其制备方法和应用

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CN1675201A (zh) * 2002-06-24 2005-09-28 阿卡蒂亚药品公司 N－取代哌啶衍生物作为血清素受体试剂
CN109111385A (zh) * 2017-06-23 2019-01-01 上海翰森生物医药科技有限公司 5-ht2a受体抑制剂及其制备方法和应用
WO2019040107A1 (en) * 2017-08-21 2019-02-28 Acadia Pharmaceuticals Inc. COMPOUNDS, CORRESPONDING SALTS AND METHODS FOR THE TREATMENT OF DISEASES
CN115605202A (zh) * 2020-03-26 2023-01-13 盐野义制药株式会社（Jp） 具有血清素受体结合活性的芳香族杂环衍生物

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