CN113302175A - 双环化合物 - Google Patents

双环化合物 Download PDF

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CN113302175A
CN113302175A CN201980088541.5A CN201980088541A CN113302175A CN 113302175 A CN113302175 A CN 113302175A CN 201980088541 A CN201980088541 A CN 201980088541A CN 113302175 A CN113302175 A CN 113302175A
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substituted
unsubstituted
pharmaceutically acceptable
compound
acceptable salt
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CN201980088541.5A
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Chinese (zh)
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安德烈·W·康拉迪
特蕾西·紫玲·汤·林
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Vivas Treatment Co
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Vivas Treatment Co
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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CN114181039A (zh) * 2021-12-23 2022-03-15 凯美克(上海)医药科技有限公司 一种4,4-二苯基-3-丁烯-1-醇的合成方法
CN114539080A (zh) * 2022-03-02 2022-05-27 八叶草健康产业研究院(厦门)有限公司 一种2-(2-氨基-6-氯苯基)-乙酸钠的制备方法
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EP3917911A1 (en) * 2019-01-31 2021-12-08 Kyorin Pharmaceutical Co., Ltd. 15-pgdh inhibitors
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IL301691A (en) 2020-09-30 2023-05-01 Univ Leuven Kath 1,2,3,4-tetrahydroquinoline derivatives as inhibitors of the yap/taz-tead activation for treating cancer
WO2022120355A1 (en) 2020-12-02 2022-06-09 Ikena Oncology, Inc. Tead degraders and uses thereof
CA3205726A1 (en) 2021-01-25 2022-07-28 Alfredo C. Castro Combination of a 3-(imidazol-4-yl)-4-(amino)-benzenesulfonamide tead inhibitor with an egfr inhibitor and/or mek inhibitor for use in the treatment of lung cancer
WO2022233442A1 (en) * 2021-02-10 2022-11-10 Merck Patent Gmbh 2,8-dihydropyrazolo[3,4-b]indole derivatives for use in the treatment of cancer
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