CN108137519A - 合成n-(1，3，4-噁二唑-2-基)芳基甲酰胺的方法 - Google Patents

合成n-(1，3，4-噁二唑-2-基)芳基甲酰胺的方法 Download PDF

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Publication number
CN108137519A
CN108137519A CN201680056686.3A CN201680056686A CN108137519A CN 108137519 A CN108137519 A CN 108137519A CN 201680056686 A CN201680056686 A CN 201680056686A CN 108137519 A CN108137519 A CN 108137519A
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CN
China
Prior art keywords
methyl
formula
alkyl
activator
iii
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN201680056686.3A
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English (en)
Chinese (zh)
Inventor
克里斯蒂安·冯克
阿尔德·尼弗
塞吉尔·帕泽诺克
诺伯特·路伊
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Bayer CropScience AG
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Bayer CropScience AG
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Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Publication of CN108137519A publication Critical patent/CN108137519A/zh
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/113—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/582—Recycling of unreacted starting or intermediate materials

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Laminated Bodies (AREA)
  • Shaping By String And By Release Of Stress In Plastics And The Like (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
CN201680056686.3A 2015-09-28 2016-09-23 合成n-(1，3，4-噁二唑-2-基)芳基甲酰胺的方法 Pending CN108137519A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15187023 2015-09-28
EP15187023.5 2015-09-28
PCT/EP2016/072629 WO2017055175A1 (de) 2015-09-28 2016-09-23 Verfahren zur herstellung von n-(1,3,4-oxadiazol-2-yl)arylcarboxamiden

Publications (1)

Publication Number Publication Date
CN108137519A true CN108137519A (zh) 2018-06-08

Family

ID=54207378

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201680056686.3A Pending CN108137519A (zh) 2015-09-28 2016-09-23 合成n-(1，3，4-噁二唑-2-基)芳基甲酰胺的方法

Country Status (10)

Country Link
US (1) US10189800B2 (https=)
EP (1) EP3356336A1 (https=)
JP (1) JP2018529703A (https=)
KR (1) KR20180059456A (https=)
CN (1) CN108137519A (https=)
BR (1) BR112018006202A2 (https=)
IL (1) IL258320B (https=)
MX (1) MX2018003963A (https=)
TW (1) TW201711566A (https=)
WO (1) WO2017055175A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE060120T2 (hu) * 2017-05-04 2023-01-28 Bayer Cropscience Ag Herbicidként aktív 4-difluormetilbenzoilamid
KR102868734B1 (ko) * 2020-12-17 2025-10-02 주식회사 팜한농 N-(1-메틸-1h-테트라졸-5-일)-2-(((2-메틸-2h-테트라졸-5-일)메톡시)메틸)-6-(트리플루오로메틸)니코틴아마이드의 제조 방법
CN117616016A (zh) * 2021-07-08 2024-02-27 拜耳公司 手性3-亚磺酰基苯甲酸

Citations (6)

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WO2002026731A2 (en) * 2000-09-29 2002-04-04 Millenium Pharmaceuticals, Inc. Quaternary amidino based inhibitors of factor xa
CN102491971A (zh) * 2011-12-19 2012-06-13 北京理工大学 手性[(4-甲基-2-丙基-1h-苯并咪唑-6-酰胺)-1-基]甲基联苯类化合物及其制备方法和用途
CN103282354A (zh) * 2010-09-01 2013-09-04 拜耳知识产权有限责任公司 N-(四唑-5-基)-和n-(三唑-5-基)芳基甲酰胺及其作为除草剂的用途
CN103443107A (zh) * 2011-03-28 2013-12-11 弗·哈夫曼-拉罗切有限公司 噻唑并嘧啶化合物
CN103596946A (zh) * 2011-03-22 2014-02-19 拜耳知识产权有限责任公司 N-(1,3,4-噁二唑-2-基)芳基甲酰胺及其作为除草剂的用途
US20140309112A1 (en) * 2011-11-03 2014-10-16 Bayer Intellectual Property Gmbh Herbicidally active oxime-ether-substituted benzoylamides

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US20080090834A1 (en) 2006-07-06 2008-04-17 Pfizer Inc Selective azole pde10a inhibitor compounds
JP2009091267A (ja) * 2007-10-04 2009-04-30 Kyorin Pharmaceut Co Ltd アミド誘導体及びそれらを有効成分とするスフィンゴシン−１−リン酸−１（ｓ１ｐ１）受容体選択的アゴニスト
MY160399A (en) * 2009-07-06 2017-03-15 Aerpio Therapeutics Inc Compounds, compositions, and methods for preventing metastasis of cancer cells
EP2691399B1 (en) * 2011-03-28 2016-07-13 F.Hoffmann-La Roche Ag Thiazolopyrimidine compounds
JP6110881B2 (ja) 2012-02-21 2017-04-05 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 除草３−（スルフィン−／スルホンイミドイル）−ベンズアミド
CN104955456B (zh) * 2013-01-28 2018-07-03 H.隆德贝克有限公司 作为分拣蛋白抑制剂的n-取代的-5-取代的邻氨甲酰苯甲酸
CA2941215A1 (en) * 2014-03-10 2015-09-17 Meiji Seika Pharma Co., Ltd. Method for producing 2-acyliminopyridine derivative

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002026731A2 (en) * 2000-09-29 2002-04-04 Millenium Pharmaceuticals, Inc. Quaternary amidino based inhibitors of factor xa
CN103282354A (zh) * 2010-09-01 2013-09-04 拜耳知识产权有限责任公司 N-(四唑-5-基)-和n-(三唑-5-基)芳基甲酰胺及其作为除草剂的用途
CN103596946A (zh) * 2011-03-22 2014-02-19 拜耳知识产权有限责任公司 N-(1,3,4-噁二唑-2-基)芳基甲酰胺及其作为除草剂的用途
CN103443107A (zh) * 2011-03-28 2013-12-11 弗·哈夫曼-拉罗切有限公司 噻唑并嘧啶化合物
US20140309112A1 (en) * 2011-11-03 2014-10-16 Bayer Intellectual Property Gmbh Herbicidally active oxime-ether-substituted benzoylamides
CN102491971A (zh) * 2011-12-19 2012-06-13 北京理工大学 手性[(4-甲基-2-丙基-1h-苯并咪唑-6-酰胺)-1-基]甲基联苯类化合物及其制备方法和用途

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
MANABU YASUMOTO ET AL.，: "Self-disproportionation of enantiomers of 3,3,3-trifluorolactic acid amides via sublimation", 《JOURNAL OF FLUORINE CHEMISTRY》 *

Also Published As

Publication number Publication date
IL258320A (en) 2018-05-31
BR112018006202A2 (pt) 2018-10-09
MX2018003963A (es) 2018-06-08
EP3356336A1 (de) 2018-08-08
WO2017055175A1 (de) 2017-04-06
KR20180059456A (ko) 2018-06-04
IL258320B (en) 2019-09-26
TW201711566A (zh) 2017-04-01
US20180273496A1 (en) 2018-09-27
JP2018529703A (ja) 2018-10-11
US10189800B2 (en) 2019-01-29

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Application publication date: 20180608