CN106478497B - 作为ttx-s阻滞剂的芳胺衍生物 - Google Patents

作为ttx-s阻滞剂的芳胺衍生物 Download PDF

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CN106478497B
CN106478497B CN201610833742.1A CN201610833742A CN106478497B CN 106478497 B CN106478497 B CN 106478497B CN 201610833742 A CN201610833742 A CN 201610833742A CN 106478497 B CN106478497 B CN 106478497B
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methyl
pyridin
isonicotinamide
ethyl
trifluoroethoxy
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CN106478497A (zh
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山岸龙也
川村清
新野义政
森田干雄
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Raqualia Pharma Inc
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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CN201610833742.1A 2010-10-18 2011-10-18 作为ttx-s阻滞剂的芳胺衍生物 Active CN106478497B (zh)

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US39401710P 2010-10-18 2010-10-18
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US41800210P 2010-11-30 2010-11-30
US61/418,002 2010-11-30
US201161522792P 2011-08-12 2011-08-12
US61/522,792 2011-08-12
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US (1) US9302991B2 (https=)
EP (1) EP2630122B1 (https=)
JP (2) JP2013543480A (https=)
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CN (2) CN106478497B (https=)
BR (1) BR112013009365B1 (https=)
CA (1) CA2813708C (https=)
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EP2630122B1 (en) * 2010-10-18 2016-11-30 RaQualia Pharma Inc Arylamide derivatives as ttx-s blockers
MX2014001862A (es) * 2011-09-12 2014-05-30 Hoffmann La Roche 5-cicloalquil-o 5-heterociclil-nicotinamidas.
IN2014MN01982A (https=) * 2012-04-25 2015-07-10 Raqualia Pharma Inc
KR102090944B1 (ko) * 2012-04-25 2020-03-19 라퀄리아 파마 인코포레이티드 Ttx-s 차단제로서의 피롤로피리디논 유도체
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BR112013009365B1 (pt) 2021-10-26
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