CN104640858B - 环醚吡唑-4-基-杂环基-甲酰胺化合物及使用方法 - Google Patents

环醚吡唑-4-基-杂环基-甲酰胺化合物及使用方法 Download PDF

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CN104640858B
CN104640858B CN201380048262.9A CN201380048262A CN104640858B CN 104640858 B CN104640858 B CN 104640858B CN 201380048262 A CN201380048262 A CN 201380048262A CN 104640858 B CN104640858 B CN 104640858B
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methyl
amino
bases
nitro
compound
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CN104640858A (zh
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W.布莱卡比
J.伯奇
A.J.霍奇斯
A.夏普
M.孙
X.王
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F Hoffmann La Roche AG
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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CN201380048262.9A 2012-09-26 2013-09-25 环醚吡唑-4-基-杂环基-甲酰胺化合物及使用方法 Active CN104640858B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261705791P 2012-09-26 2012-09-26
US61/705,791 2012-09-26
US201361864882P 2013-08-12 2013-08-12
US61/864,882 2013-08-12
PCT/EP2013/069892 WO2014048939A1 (en) 2012-09-26 2013-09-25 Cyclic ether pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use

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CN104640858B true CN104640858B (zh) 2018-11-06

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