CN104302630A - 作为甲酰肽受体2调节剂的(2-脲基乙酰氨基)烷基衍生物 - Google Patents

作为甲酰肽受体2调节剂的(2-脲基乙酰氨基)烷基衍生物 Download PDF

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CN104302630A
CN104302630A CN201380025558.9A CN201380025558A CN104302630A CN 104302630 A CN104302630 A CN 104302630A CN 201380025558 A CN201380025558 A CN 201380025558A CN 104302630 A CN104302630 A CN 104302630A
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substituted
unsubstituted
amino
hydrogen
alkyl
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R·L·比尔德
T·T·杜昂
J·E·多纳罗
V·维斯瓦纳斯
M·E·贾斯特
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Allergan Inc
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Allergan Inc
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    • C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C309/13—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton
    • C07C309/14—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton containing amino groups bound to the carbon skeleton
    • C07C309/15—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing nitrogen atoms, not being part of nitro or nitroso groups, bound to the carbon skeleton containing amino groups bound to the carbon skeleton the nitrogen atom of at least one of the amino groups being part of any of the groups, X being a hetero atom, Y being any atom
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CN201380025558.9A 2012-04-16 2013-04-16 作为甲酰肽受体2调节剂的(2-脲基乙酰氨基)烷基衍生物 Pending CN104302630A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261624495P 2012-04-16 2012-04-16
US61/624,495 2012-04-16
PCT/US2013/036715 WO2013158597A1 (en) 2012-04-16 2013-04-16 (2-ureidoacetamido)alkyl derivatives as formyl peptide receptor 2 modulators

Publications (1)

Publication Number Publication Date
CN104302630A true CN104302630A (zh) 2015-01-21

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CN201380025558.9A Pending CN104302630A (zh) 2012-04-16 2013-04-16 作为甲酰肽受体2调节剂的(2-脲基乙酰氨基)烷基衍生物

Country Status (11)

Country Link
US (1) US9670150B2 (https=)
EP (1) EP2838887B1 (https=)
JP (1) JP2015520130A (https=)
KR (1) KR20140145203A (https=)
CN (1) CN104302630A (https=)
AU (1) AU2013249474A1 (https=)
CA (1) CA2870356A1 (https=)
ES (1) ES2711363T3 (https=)
NZ (1) NZ700733A (https=)
SG (1) SG11201406629VA (https=)
WO (1) WO2013158597A1 (https=)

Cited By (2)

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Publication number Priority date Publication date Assignee Title
CN109593067A (zh) * 2017-09-30 2019-04-09 暨南大学 四氮唑类分子探针化合物或组合物及其应用
CN109641857A (zh) * 2016-04-12 2019-04-16 阿勒根公司 作为n-甲酰基肽受体调节剂的苯基脲衍生物

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AU2012329098B2 (en) 2011-10-26 2017-08-03 Allergan, Inc. Amide derivatives of N-urea substituted amino acids as formyl peptide receptor like-1 (FPRL-1) receptor modulators
KR102223384B1 (ko) * 2013-03-06 2021-03-05 알러간, 인코포레이티드 피부 질환 치료용 포르밀 펩티드 수용체 2의 항진제의 용도
AU2014225992B2 (en) 2013-03-06 2018-03-22 Allergan, Inc. Use of agonists of formyl peptide receptor 2 for treating ocular inflammatory diseases
RU2703725C1 (ru) * 2013-11-21 2019-10-22 Аллерган, Инк. Производные фенилкарбамата в качестве модуляторов формилпептидного рецептора
NZ720508A (en) 2013-11-28 2019-03-29 Kyorin Seiyaku Kk Urea derivative or pharmacologically acceptable salt thereof
US9604934B2 (en) 2014-01-29 2017-03-28 Allergan, Inc. Urea hydantoin derivatives as formyl peptide modulators
US9663457B2 (en) 2014-04-09 2017-05-30 Allergan, Inc. Carbamoyl hydrazine derivatives as formyl peptide modulators
WO2015179707A1 (en) 2014-05-21 2015-11-26 Allergan, Inc. Imidazole derivatives as formyl peptide receptor modulators
TW201718473A (zh) * 2015-08-05 2017-06-01 歐樂根公司 作為甲醯肽受體１（ｆｐｒ１）選擇性促效劑之苯基脲類似物
WO2018227065A1 (en) * 2017-06-09 2018-12-13 Bristol-Myers Squibb Company Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists
KR102615095B1 (ko) * 2017-06-09 2023-12-15 브리스톨-마이어스 스큅 컴퍼니 피페리디논 포르밀 펩티드 2 수용체 효능제
KR102803660B1 (ko) 2018-03-05 2025-05-02 브리스톨-마이어스 스큅 컴퍼니 페닐피롤리디논 포르밀 펩티드 2 수용체 효능제

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KR102223384B1 (ko) * 2013-03-06 2021-03-05 알러간, 인코포레이티드 피부 질환 치료용 포르밀 펩티드 수용체 2의 항진제의 용도

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109641857A (zh) * 2016-04-12 2019-04-16 阿勒根公司 作为n-甲酰基肽受体调节剂的苯基脲衍生物
CN109593067A (zh) * 2017-09-30 2019-04-09 暨南大学 四氮唑类分子探针化合物或组合物及其应用
CN109593067B (zh) * 2017-09-30 2021-11-26 暨南大学 四氮唑类分子探针化合物或组合物及其应用

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WO2013158597A1 (en) 2013-10-24
US9670150B2 (en) 2017-06-06
CA2870356A1 (en) 2013-10-24
EP2838887A1 (en) 2015-02-25
KR20140145203A (ko) 2014-12-22
JP2015520130A (ja) 2015-07-16
SG11201406629VA (en) 2014-11-27
US20130274230A1 (en) 2013-10-17
AU2013249474A1 (en) 2014-11-06

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