CN1041383C - 制备有效抑制妇女排卵的组合物的方法 - Google Patents
制备有效抑制妇女排卵的组合物的方法 Download PDFInfo
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- CN1041383C CN1041383C CN88101379A CN88101379A CN1041383C CN 1041383 C CN1041383 C CN 1041383C CN 88101379 A CN88101379 A CN 88101379A CN 88101379 A CN88101379 A CN 88101379A CN 1041383 C CN1041383 C CN 1041383C
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- 230000001629 suppression Effects 0.000 description 1
- 239000004094 surface-active agent Substances 0.000 description 1
- 238000013268 sustained release Methods 0.000 description 1
- 239000012730 sustained-release form Substances 0.000 description 1
- 208000024891 symptom Diseases 0.000 description 1
- 230000002381 testicular Effects 0.000 description 1
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- 210000004291 uterus Anatomy 0.000 description 1
- 229940044952 vaginal foam Drugs 0.000 description 1
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Images
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Indole Compounds (AREA)
- Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
- Saccharide Compounds (AREA)
- Peptides Or Proteins (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Seeds, Soups, And Other Foods (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US029,229 | 1987-03-23 | ||
| US07/029,229 US4855305A (en) | 1987-03-23 | 1987-03-23 | Compositions and methods of effecting contraception utilizing melatonin |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN88101379A CN88101379A (zh) | 1988-10-05 |
| CN1041383C true CN1041383C (zh) | 1998-12-30 |
Family
ID=21847942
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN88101379A Expired - Fee Related CN1041383C (zh) | 1987-03-23 | 1988-03-23 | 制备有效抑制妇女排卵的组合物的方法 |
Country Status (26)
| Country | Link |
|---|---|
| US (1) | US4855305A (enExample) |
| EP (1) | EP0354921B1 (enExample) |
| JP (2) | JP2965160B2 (enExample) |
| KR (1) | KR890700349A (enExample) |
| CN (1) | CN1041383C (enExample) |
| AT (1) | ATE143807T1 (enExample) |
| AU (3) | AU628784B2 (enExample) |
| BG (1) | BG51075A1 (enExample) |
| BR (1) | BR8807426A (enExample) |
| CA (1) | CA1322527C (enExample) |
| DD (1) | DD269557A5 (enExample) |
| DE (1) | DE3855606T2 (enExample) |
| EG (1) | EG18583A (enExample) |
| ES (1) | ES2009251A6 (enExample) |
| FI (1) | FI894423L (enExample) |
| GR (1) | GR1002146B (enExample) |
| HU (1) | HU208487B (enExample) |
| IL (1) | IL85814A (enExample) |
| IN (1) | IN166946B (enExample) |
| NZ (1) | NZ223989A (enExample) |
| OA (1) | OA09134A (enExample) |
| PH (1) | PH26709A (enExample) |
| PT (1) | PT87053B (enExample) |
| RU (1) | RU2114621C1 (enExample) |
| WO (1) | WO1988007370A1 (enExample) |
| ZA (1) | ZA882079B (enExample) |
Families Citing this family (44)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GR1001395B (el) * | 1987-03-23 | 1993-10-29 | Michael Cohen | Συν?έσεις και μέ?οδοι προς πραγματοποίηση αντισύλληψης. |
| EP0300630A3 (en) * | 1987-07-03 | 1990-03-28 | Schering Agrochemicals Limited | Melatonin for regulating animal reproduction |
| IL87574A0 (en) * | 1987-08-28 | 1989-01-31 | Regulin Ltd | Composition for regulating animal reproduction containing an indole derivative |
| US4945103A (en) * | 1989-01-17 | 1990-07-31 | Michael Cohen | Method of treating pre-menstrual syndrome |
| IN170311B (enExample) * | 1989-01-17 | 1992-03-14 | Cohen Michael | |
| GR900100024A (el) * | 1989-01-17 | 1991-06-07 | Amr Int | Μέθοδος θεραπείας του προεμμηνορροϊκού συνδρόμου. |
| BR9007382A (pt) * | 1989-05-17 | 1992-04-28 | Michael Cohen | Composicoes e metodos de efetuar a contracepcao |
| NZ233697A (en) * | 1989-05-17 | 1996-12-20 | Applied Med Res Ltd | Contraceptive composition comprising a melatonin analogue and a progestogen and/or an estrogen |
| IT1243193B (it) * | 1990-08-10 | 1994-05-24 | Medea Res Srl | Composizioni farmaceutiche orali a base di melatonina |
| EP0483077B1 (en) * | 1990-09-28 | 1995-12-06 | I.F.L.O. S.a.s. di Giorgio e Aldo Laguzzi | A method for carrying out the synthesis of a contraceptive and menstrual cycle controlling drug having oncostatic, antikinetosic, preventive and therapeutic properties for treatment of mammary tumours and melanomas. |
| DE69229490T2 (de) * | 1991-05-09 | 2000-02-17 | Neurim Pharmaceuticals (1991) Ltd., Tel Aviv | Melatonin enthaltende Arzneimittel |
| AU660336B2 (en) * | 1991-10-18 | 1995-06-22 | Alza Corporation | Device for the transdermal administration of melatonin |
| US5196435A (en) * | 1991-11-21 | 1993-03-23 | Eli Lilly And Company | Melatonin derivatives and combinations with antiestrogen compounds for treating mammalian breast carcinoma |
| DK0565296T3 (da) * | 1992-04-07 | 1996-12-09 | Neurim Pharma 1991 | Anvendelse af melatonin til fremstilling af et lægemiddel til behandling af godartet prostatahyperplasi |
| US5792785A (en) * | 1995-11-24 | 1998-08-11 | Equitech Laboratories, Inc. | Method for enhancing pregnancy success in an animal |
| US6403631B1 (en) | 1995-11-24 | 2002-06-11 | Equitech Laboratories, Inc. | Method and compositions for enhancing pregnancy success in an animal |
| US6028064A (en) * | 1996-09-13 | 2000-02-22 | New Life Pharmaceuticals Inc. | Prevention of ovarian cancer by administration of progestin products |
| US6620836B1 (en) * | 1997-01-22 | 2003-09-16 | Jay Patrick | Antiarrhythmic and tranquilizer composition and treatment |
| DE19739916C2 (de) * | 1997-09-11 | 2001-09-13 | Hesch Rolf Dieter | Verwendung einer Kombination aus einem Gestagen und einem Estrogen zur kontinuierlichen Ovulationshemmung und ggf. gleichzeitigen Behandlung und/oder Prophylaxe von Tumoren der Brustdrüsen |
| AU747710B2 (en) | 1997-11-14 | 2002-05-23 | Akzo Nobel N.V. | Progestogen-antiprogestogen regimens |
| US6133453A (en) * | 1998-05-15 | 2000-10-17 | Pharm-Eco Laboratories, Inc. | Method for making substituted indoles |
| US7989436B2 (en) | 2003-07-23 | 2011-08-02 | Duramed Pharmaceuticals, Inc. | Estrogenic compounds and pharmaceutical formulations comprising the same |
| US6855703B1 (en) | 2000-03-10 | 2005-02-15 | Endeavor Pharmaceuticals | Pharmaceutical compositions of conjugated estrogens and methods of analyzing mixtures containing estrogenic compounds |
| US7459445B2 (en) * | 2000-03-10 | 2008-12-02 | Duramed Pharmaceuticals, Inc. | Estrogenic compounds and topical pharmaceutical formulations of the same |
| US6660726B2 (en) | 2000-03-10 | 2003-12-09 | Endeavor Pharmaceuticals | Estrogenic compounds, pharmaceutical compositions thereof, and methods of using same |
| US20040176336A1 (en) * | 2000-03-21 | 2004-09-09 | Rodriguez Gustavo C. | Prevention of ovarian cancer by administration of products that induce biologic effects in the ovarian epithelium |
| US20050113351A1 (en) * | 2000-03-21 | 2005-05-26 | Rodriguez Gustavo C. | Prevention of ovarian cancer by administration of products that induce biologic effects in the ovarian epithelium |
| ES2341090T3 (es) * | 2000-08-30 | 2010-06-15 | Unimed Pharmaceuticals, Llc | Procedimiento para tratar la disfuncion erectil y aumentar la libido en hombres. |
| US6503894B1 (en) | 2000-08-30 | 2003-01-07 | Unimed Pharmaceuticals, Inc. | Pharmaceutical composition and method for treating hypogonadism |
| US20030139384A1 (en) * | 2000-08-30 | 2003-07-24 | Dudley Robert E. | Method for treating erectile dysfunction and increasing libido in men |
| WO2003077900A1 (en) * | 2002-03-14 | 2003-09-25 | Prevention, L.L.C. | A unifying mechanism and methods to prevent cancer and neurodegenerative diseases |
| US6992075B2 (en) * | 2003-04-04 | 2006-01-31 | Barr Laboratories, Inc. | C(14) estrogenic compounds |
| MXPA05010871A (es) * | 2003-04-11 | 2005-11-25 | Barr Lab Inc | Metodos para administrar estrogenos y progestinas. |
| DK1663197T3 (da) | 2003-09-09 | 2008-01-07 | Fumapharm Ag | Anvendelse af fumarsyrederivater til behandling af hjerteinsuffiens og astma |
| MXPA06013418A (es) * | 2004-05-26 | 2007-01-23 | Wyeth Corp | Composiciones y metodos para el tratamiento del trastorno disforico premenstrual. |
| SI1799196T1 (sl) | 2004-10-08 | 2016-10-28 | Forward Pharma A/S | Farmacevtski sestavki z nadzorovanim sproščanjem, obsegajoči ester fumarne kisline |
| RS52671B (sr) | 2005-10-12 | 2013-06-28 | Unimed Pharmaceuticals Llc | Poboljšani gel testosterona i postupak korišćenja |
| CN101516255A (zh) * | 2006-09-13 | 2009-08-26 | 皇家飞利浦电子股份有限公司 | 用于自动调整褪黑素的剂量和/或递送褪黑素的装置 |
| EP2653873B8 (en) | 2007-02-08 | 2022-08-24 | Biogen MA Inc. | Compositions and uses for treating Multiple Sclerosis |
| DE102008036825A1 (de) * | 2008-08-05 | 2010-02-11 | Aicuris Gmbh & Co. Kg | Schwangerschaftsvermeidung durch Gestagene |
| FR2937862B1 (fr) * | 2008-11-03 | 2010-11-19 | Mohammed Ridha Chakroun | Kit contraceptif |
| WO2015144965A1 (es) * | 2014-03-27 | 2015-10-01 | Servicio Andaluz De Salud | Preparación duradera de inyectable de melatonina estable a largo plazo |
| RU2617518C2 (ru) * | 2015-07-01 | 2017-04-25 | Общество с ограниченной ответственностью "Научно-внедренческий центр Агроветзащита" | Способ регулирования полового поведения и контрацепции самок млекопитающих |
| RU2616252C2 (ru) * | 2015-08-04 | 2017-04-13 | Общество с ограниченной ответственностью "Научно-внедренческий центр Агроветзащита" | Способ регулирования полового поведения самцов млекопитающих |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4087444A (en) * | 1976-09-08 | 1978-05-02 | Eli Lilly And Company | Amides as ovulation inhibitors |
| EP0004770B1 (en) * | 1978-04-11 | 1984-06-13 | Efamol Limited | Pharmaceutical and dietary composition comprising gamma-linolenic acids |
| US4425339A (en) * | 1981-04-09 | 1984-01-10 | Syntex (U.S.A.) Inc. | Treatment of menopausal symptoms |
| US4390531A (en) * | 1981-08-10 | 1983-06-28 | Syntex Pharmaceuticals International Ltd. | Method of contraception using peak progestogen dosage |
| US4628051A (en) * | 1983-09-26 | 1986-12-09 | Ortho Pharmaceutical Corporation | Triphasic oral contraceptive |
| US4614807A (en) * | 1984-10-04 | 1986-09-30 | Eli Lilly And Company | 6,7-dihalomelatonins |
| DE3685696T2 (de) * | 1985-03-04 | 1993-01-14 | Cell Eng Ag | Melatoninhaltige mittel sowie deren verwendungen. |
| US4746674A (en) * | 1985-08-27 | 1988-05-24 | Cellena (Cell Engineering) Ag | Melatonin compositions and uses thereof |
| US4997845A (en) * | 1987-02-02 | 1991-03-05 | Eli Lilly And Company | β-alkylmelatonins as ovulation inhibitors |
-
1987
- 1987-03-23 US US07/029,229 patent/US4855305A/en not_active Expired - Lifetime
-
1988
- 1988-03-22 EP EP88904025A patent/EP0354921B1/en not_active Expired - Lifetime
- 1988-03-22 CA CA000562109A patent/CA1322527C/en not_active Expired - Fee Related
- 1988-03-22 HU HU883281A patent/HU208487B/hu not_active IP Right Cessation
- 1988-03-22 FI FI894423A patent/FI894423L/fi not_active Application Discontinuation
- 1988-03-22 AU AU16830/88A patent/AU628784B2/en not_active Ceased
- 1988-03-22 JP JP63503744A patent/JP2965160B2/ja not_active Expired - Fee Related
- 1988-03-22 WO PCT/US1988/000971 patent/WO1988007370A1/en not_active Ceased
- 1988-03-22 DE DE3855606T patent/DE3855606T2/de not_active Expired - Fee Related
- 1988-03-22 RU SU4742272A patent/RU2114621C1/ru not_active IP Right Cessation
- 1988-03-22 BR BR888807426A patent/BR8807426A/pt not_active Application Discontinuation
- 1988-03-22 PH PH36671A patent/PH26709A/en unknown
- 1988-03-22 AT AT88904025T patent/ATE143807T1/de not_active IP Right Cessation
- 1988-03-22 IL IL85814A patent/IL85814A/xx not_active IP Right Cessation
- 1988-03-23 ES ES8800883A patent/ES2009251A6/es not_active Expired
- 1988-03-23 GR GR880100177A patent/GR1002146B/el not_active IP Right Cessation
- 1988-03-23 EG EG166/88A patent/EG18583A/xx active
- 1988-03-23 CN CN88101379A patent/CN1041383C/zh not_active Expired - Fee Related
- 1988-03-23 NZ NZ223989A patent/NZ223989A/xx unknown
- 1988-03-23 PT PT87053A patent/PT87053B/pt not_active IP Right Cessation
- 1988-03-23 DD DD88313924A patent/DD269557A5/de not_active IP Right Cessation
- 1988-03-23 ZA ZA882079A patent/ZA882079B/xx unknown
- 1988-03-28 IN IN197/MAS/88A patent/IN166946B/en unknown
- 1988-11-23 KR KR1019880701526A patent/KR890700349A/ko not_active Ceased
-
1989
- 1989-09-19 OA OA59646A patent/OA09134A/xx unknown
- 1989-09-25 BG BG89841A patent/BG51075A1/bg unknown
-
1991
- 1991-10-31 AU AU86938/91A patent/AU8693891A/en not_active Abandoned
-
1994
- 1994-02-14 AU AU55134/94A patent/AU676523B2/en not_active Ceased
-
1998
- 1998-02-12 JP JP10044264A patent/JPH1171276A/ja active Pending
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| C14 | Grant of patent or utility model | ||
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| C15 | Extension of patent right duration from 15 to 20 years for appl. with date before 31.12.1992 and still valid on 11.12.2001 (patent law change 1993) | ||
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| CF01 | Termination of patent right due to non-payment of annual fee |