CN103958496B - 制备n‑取代的1h‑吡唑‑5‑甲酸盐化合物及其衍生物的方法 - Google Patents

制备n‑取代的1h‑吡唑‑5‑甲酸盐化合物及其衍生物的方法 Download PDF

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Publication number
CN103958496B
CN103958496B CN201280056937.XA CN201280056937A CN103958496B CN 103958496 B CN103958496 B CN 103958496B CN 201280056937 A CN201280056937 A CN 201280056937A CN 103958496 B CN103958496 B CN 103958496B
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alkoxy
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CN103958496A (zh
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M·多奇纳赫勒
K·科尔博尔
P·德施姆克
F·凯泽
M·拉克
T·弗拉塞托
G·维奇
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10—Spiro-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CN201280056937.XA 2011-11-21 2012-11-20 制备n‑取代的1h‑吡唑‑5‑甲酸盐化合物及其衍生物的方法 Expired - Fee Related CN103958496B (zh)

Applications Claiming Priority (5)

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US201161561975P 2011-11-21 2011-11-21
EP11189973.8 2011-11-21
EP11189973 2011-11-21
US61/561,975 2011-11-21
PCT/EP2012/073128 WO2013076092A1 (en) 2011-11-21 2012-11-20 Process for preparing n-substituted 1h-pyrazole-5-carboxylate compounds and derivatives thereof

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CN103958496A CN103958496A (zh) 2014-07-30
CN103958496B true CN103958496B (zh) 2017-05-24

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US (1) US9556141B2 (enExample)
EP (1) EP2782910B1 (enExample)
JP (1) JP6067733B2 (enExample)
KR (1) KR20140100474A (enExample)
CN (1) CN103958496B (enExample)
AU (1) AU2012342564A1 (enExample)
BR (1) BR112014012243A2 (enExample)
ES (1) ES2565821T3 (enExample)
IL (1) IL232277A (enExample)
IN (1) IN2014CN03469A (enExample)
MX (1) MX2014005870A (enExample)
WO (1) WO2013076092A1 (enExample)

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IL232277A0 (en) 2014-07-01
BR112014012243A2 (pt) 2017-05-30
CN103958496A (zh) 2014-07-30
MX2014005870A (es) 2014-06-23
WO2013076092A1 (en) 2013-05-30
EP2782910B1 (en) 2016-02-03
AU2012342564A1 (en) 2014-06-12
JP2014533677A (ja) 2014-12-15
US9556141B2 (en) 2017-01-31
US20150087843A1 (en) 2015-03-26
KR20140100474A (ko) 2014-08-14
JP6067733B2 (ja) 2017-01-25
IN2014CN03469A (enExample) 2015-07-03
ES2565821T3 (es) 2016-04-07
EP2782910A1 (en) 2014-10-01
IL232277A (en) 2017-03-30

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