JP6067733B2 - N置換1h−ピラゾール−5−カルボキシラート化合物及びその誘導体を製造する方法 - Google Patents

N置換1h−ピラゾール−5−カルボキシラート化合物及びその誘導体を製造する方法 Download PDF

Info

Publication number
JP6067733B2
JP6067733B2 JP2014541709A JP2014541709A JP6067733B2 JP 6067733 B2 JP6067733 B2 JP 6067733B2 JP 2014541709 A JP2014541709 A JP 2014541709A JP 2014541709 A JP2014541709 A JP 2014541709A JP 6067733 B2 JP6067733 B2 JP 6067733B2
Authority
JP
Japan
Prior art keywords
compound
alkyl
groups
formula
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
JP2014541709A
Other languages
English (en)
Japanese (ja)
Other versions
JP2014533677A (ja
Inventor
ドシュナル,マクシミリアン
ケルバー,カルステン
デシュムク,プラサント
カイザー,フローリアン
ラック,ミヒャエル
フラッセット,ティモ
ビーチ,ジェマ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Publication of JP2014533677A publication Critical patent/JP2014533677A/ja
Application granted granted Critical
Publication of JP6067733B2 publication Critical patent/JP6067733B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
JP2014541709A 2011-11-21 2012-11-20 N置換1h−ピラゾール−5−カルボキシラート化合物及びその誘導体を製造する方法 Expired - Fee Related JP6067733B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161561975P 2011-11-21 2011-11-21
EP11189973.8 2011-11-21
US61/561,975 2011-11-21
EP11189973 2011-11-21
PCT/EP2012/073128 WO2013076092A1 (en) 2011-11-21 2012-11-20 Process for preparing n-substituted 1h-pyrazole-5-carboxylate compounds and derivatives thereof

Publications (2)

Publication Number Publication Date
JP2014533677A JP2014533677A (ja) 2014-12-15
JP6067733B2 true JP6067733B2 (ja) 2017-01-25

Family

ID=48469152

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014541709A Expired - Fee Related JP6067733B2 (ja) 2011-11-21 2012-11-20 N置換1h−ピラゾール−5−カルボキシラート化合物及びその誘導体を製造する方法

Country Status (12)

Country Link
US (1) US9556141B2 (enExample)
EP (1) EP2782910B1 (enExample)
JP (1) JP6067733B2 (enExample)
KR (1) KR20140100474A (enExample)
CN (1) CN103958496B (enExample)
AU (1) AU2012342564A1 (enExample)
BR (1) BR112014012243A2 (enExample)
ES (1) ES2565821T3 (enExample)
IL (1) IL232277A (enExample)
IN (1) IN2014CN03469A (enExample)
MX (1) MX2014005870A (enExample)
WO (1) WO2013076092A1 (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2014001605A (es) 2011-08-12 2014-05-01 Basf Se Proceso para la preparacion de compuestos de cloruro de 1h - pirazol - 5 - carbonilo n - sustituidos.
IN2014CN03469A (enExample) 2011-11-21 2015-07-03 Basf Se
AU2014242984A1 (en) 2013-03-28 2015-10-22 Basf Se Process for preparing sulfimines and their in-situ conversion into n-(2-amino-benzoyl)-sulfimines
BR112015027591A2 (pt) * 2013-05-17 2017-07-25 Basf Se processos para a preparação de um ácido, de um cloreto e de um composto de sulfimina
BR112015031945A2 (pt) * 2013-06-20 2017-07-25 Basf Se processos para a preparação de compostos
WO2016071243A1 (en) * 2014-11-05 2016-05-12 Basf Se Process for preparing halogenated alkenone ethers and their use in the synthesis of anthranilamide pesticides
WO2016091674A1 (en) 2014-12-12 2016-06-16 Basf Se Use of cyclaniliprole on cultivated plants
US11297837B2 (en) 2016-02-19 2022-04-12 Basf Se Pesticidally activi mixtures comprising anthranilamide compounds
MX2019002204A (es) * 2016-08-22 2019-09-19 Basf Se Proceso para preparar bifenilos sustituidos.
US11124528B2 (en) * 2017-04-27 2021-09-21 Basf Se Process for preparing optically active 2,3-dihydrothiazolo[3,2-A]pyrimidin-4-ium compounds
TWI903299B (zh) 2018-03-08 2025-11-01 美商英塞特公司 作為PI3K-γ抑制劑之胺基吡嗪二醇化合物
WO2020010003A1 (en) 2018-07-02 2020-01-09 Incyte Corporation AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS
US20220267296A1 (en) * 2019-10-18 2022-08-25 Fmc Corporation Methods for the preparation of 5-bromo-2-(3-chloro-pyridin-2-yl)-2h-pyrazole-3-carboxylic acid
TW202241859A (zh) * 2021-01-29 2022-11-01 美商富曼西公司 用於製備5-溴-2-(3-氯-吡啶-2-基)-2h-吡唑-3-甲酸之方法

Family Cites Families (57)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4544654A (en) 1984-03-20 1985-10-01 Schering A.G. Substituted sulfonamidobenzamides, antiarrhythmic agents and compositions thereof
US6136983A (en) 1995-06-05 2000-10-24 Rhone-Poulenc Agrochimie Pesticidal sulfur compounds
TW436485B (en) * 1997-08-01 2001-05-28 American Cyanamid Co Substituted quinazoline derivatives
MY138097A (en) 2000-03-22 2009-04-30 Du Pont Insecticidal anthranilamides
MXPA03007935A (es) 2001-03-05 2003-12-04 Du Pont Agentes de diamina heterociclica de control de animales invertebrados daninos.
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
TWI325302B (en) 2001-08-13 2010-06-01 Du Pont Benzoxazinone compounds
ATE396985T1 (de) 2001-08-15 2008-06-15 Du Pont Orthosubstituierte arylamide zur bekämpfung von wirbellosen schädlingen
EP1417176B1 (en) 2001-08-16 2008-12-17 E.I. Du Pont De Nemours And Company Substituted anthranilamides for controlling invertebrate pests
TWI283164B (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
EP1511733A2 (en) 2002-06-13 2005-03-09 E.I. Du Pont De Nemours And Company Pyrazole and pyrrole carboxamide insecticides
WO2004110351A2 (en) * 2003-05-14 2004-12-23 Anadys Pharmaceuticals, Inc. Heterocyclic compounds for treating hepatitis c virus
DE102004031100A1 (de) 2004-06-28 2006-01-12 Bayer Cropscience Ag Anthranilamide
MY140912A (en) * 2004-07-26 2010-01-29 Du Pont Mixtures of anthranilamide invertebrate pest control agents
TWI363756B (en) 2004-12-07 2012-05-11 Du Pont Method for preparing n-phenylpyrazole-1-carboxamides
US8143292B2 (en) * 2005-07-07 2012-03-27 Basf Se N-Thio-anthranilamid compounds and their use as pesticides
DE102005044108A1 (de) * 2005-09-15 2007-03-29 Bayer Cropscience Ag Dioxazin- und Oxdiazin-substituierte Arylamide
JP2007077106A (ja) 2005-09-16 2007-03-29 Sumitomo Chemical Co Ltd N−ピリジルアミド化合物とその用途
DK1937664T3 (da) * 2005-10-14 2011-07-18 Sumitomo Chemical Co Hydrazidforbindelse og pesticid anvendelse af den samme
HUP0600573A2 (en) 2006-07-12 2008-06-30 Laszlo Pirity Multifunction safety foil, especially fire-prevention foil
JP2009544616A (ja) 2006-07-21 2009-12-17 武田薬品工業株式会社 アミド化合物
JP5507045B2 (ja) * 2006-12-15 2014-05-28 石原産業株式会社 アントラニルアミド系化合物の製造方法
DE102007003036A1 (de) 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
JP2008280336A (ja) 2007-04-11 2008-11-20 Sumitomo Chemical Co Ltd アミド化合物の製造方法
CL2008000979A1 (es) 2007-04-11 2008-10-17 Sumitomo Chemical Co Proceso para producir un compuesto derivado de 2-piridin-2-il-2h-pirazol-3-fenilamida; compuestos intermediarios; el compuesto en si; composicion plaguicida que contiene a dicho compuesto; uso de dicho compuesto como plaguicida; y metodo para control
JP2008280341A (ja) 2007-04-12 2008-11-20 Sumitomo Chemical Co Ltd ヒドラジド化合物およびその防除用途
CA2687611A1 (en) 2007-05-24 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Novel sulphoximine-substituted quinoline and quinazoline derivatives as kinase inhibitors
TWI431000B (zh) 2008-03-05 2014-03-21 Du Pont 製備2-胺基-5-氰基苯甲酸衍生物之方法
WO2009156090A2 (de) 2008-06-26 2009-12-30 Bayer Cropscience Aktiengesellschaft Insektizide schwefel-derivatisierte 1-azinylpyrazole
EP2321262A1 (de) 2008-08-14 2011-05-18 Bayer CropScience AG Insektizide 4-phenyl-1h-pyrazole
EP2266973A1 (de) 2009-05-29 2010-12-29 Bayer CropScience AG Pyrazinylpyrazole
AR078947A1 (es) 2009-11-11 2011-12-14 Bayer Cropscience Ag Compuestos de diazinil-pirazolilo y procesos de preparacion de los mismos
WO2011064188A1 (en) 2009-11-27 2011-06-03 Basf Se Insecticidal methods using nitrogen-containing heteroaromatic compounds
MX2014001605A (es) * 2011-08-12 2014-05-01 Basf Se Proceso para la preparacion de compuestos de cloruro de 1h - pirazol - 5 - carbonilo n - sustituidos.
BR112014003217A2 (pt) 2011-08-12 2017-04-25 Basf Se composto, forma cristalina do composto, combinação pesticida, composição agrícola ou veterinária, método para combater ou controlar pragas invertebradas, método para proteger plantas em crescimento e método para a proteção de sementes
BR112014003186A2 (pt) 2011-08-12 2017-04-04 Basf Se composto da fórmula geral (i), combinação pesticida, composição agrícola ou veterinária, método para combater ou controlar pragas invertebradas, método para a proteção de plantas e sementes, semente, uso de um composto e método para tratar um animal
BR112014003220A2 (pt) 2011-08-12 2017-03-01 Basf Se composto de fórmula (i), processo para preparar um composto de fórmula i e v, uso do composto de fórmula i, método para controlar uma praga invertebrada, forma cristalina, uso das formas cristalinas e método para controlar uma praga invertebrada
CN109255735A (zh) 2011-11-18 2019-01-22 松下知识产权经营株式会社 菜谱提示系统以及菜谱提示方法
IN2014CN03469A (enExample) 2011-11-21 2015-07-03 Basf Se
WO2013113789A1 (en) 2012-02-02 2013-08-08 Basf Se N-thio-anthranilamide compounds and their use as pesticides
US9334238B2 (en) 2012-03-30 2016-05-10 Basf Se N-substituted pyridinylidenes for combating animal pests
AU2013255894A1 (en) 2012-05-04 2014-11-13 Basf Se Substituted pyrazole-containing compounds and their use as pesticides
WO2013174645A1 (en) 2012-05-24 2013-11-28 Basf Se N-thio-anthranilamide compounds and their use as pesticides
MX2015004175A (es) 2012-10-01 2015-06-10 Basf Se Uso de compuestos de n-tio-antranilamida en plantas cultivadas.
WO2014053407A1 (en) 2012-10-01 2014-04-10 Basf Se N-thio-anthranilamide compounds and their use as pesticides
WO2014053401A2 (en) 2012-10-01 2014-04-10 Basf Se Method of improving plant health
US20150250175A1 (en) 2012-10-01 2015-09-10 Basf Se Pesticidally active mixtures comprising anthranilamide compounds
BR112015003035A2 (pt) 2012-10-01 2017-12-05 Basf Se métodos para o controle de insetos, para a proteção de uma cultura e para o controle da resistência
WO2014053403A1 (en) 2012-10-01 2014-04-10 Basf Se Method of controlling insecticide resistant insects
JP2015535837A (ja) 2012-10-01 2015-12-17 ビーエーエスエフ ソシエタス・ヨーロピアBasf Se 土壌処理施用方法および種子処理施用方法におけるアントラニルアミド化合物の使用
WO2014053402A1 (en) 2012-10-01 2014-04-10 Basf Se Method for controlling non-crop pests
WO2014053405A1 (en) 2012-10-01 2014-04-10 Basf Se Pesticidally active mixtures comprising anthranilamide compounds
WO2014079820A1 (en) 2012-11-22 2014-05-30 Basf Se Use of anthranilamide compounds for reducing insect-vectored viral infections
EP2958908B1 (en) 2013-02-20 2018-12-19 Basf Se Anthranilamide compounds, their mixtures and the use thereof as pesticides
WO2014128136A1 (en) 2013-02-20 2014-08-28 Basf Se Anthranilamide compounds and their use as pesticides
AU2014242984A1 (en) 2013-03-28 2015-10-22 Basf Se Process for preparing sulfimines and their in-situ conversion into n-(2-amino-benzoyl)-sulfimines
BR112015027591A2 (pt) 2013-05-17 2017-07-25 Basf Se processos para a preparação de um ácido, de um cloreto e de um composto de sulfimina

Also Published As

Publication number Publication date
EP2782910B1 (en) 2016-02-03
ES2565821T3 (es) 2016-04-07
CN103958496A (zh) 2014-07-30
JP2014533677A (ja) 2014-12-15
US20150087843A1 (en) 2015-03-26
CN103958496B (zh) 2017-05-24
BR112014012243A2 (pt) 2017-05-30
WO2013076092A1 (en) 2013-05-30
MX2014005870A (es) 2014-06-23
IL232277A (en) 2017-03-30
AU2012342564A1 (en) 2014-06-12
KR20140100474A (ko) 2014-08-14
IN2014CN03469A (enExample) 2015-07-03
EP2782910A1 (en) 2014-10-01
IL232277A0 (en) 2014-07-01
US9556141B2 (en) 2017-01-31

Similar Documents

Publication Publication Date Title
JP6067733B2 (ja) N置換1h−ピラゾール−5−カルボキシラート化合物及びその誘導体を製造する方法
JP5955961B2 (ja) N−置換1h−ピラゾール5−カルボニルクロリド化合物を製造するための方法
JP2016518433A (ja) N置換1h−ピラゾール−5−カルボン酸化合物及びその誘導体を製造する方法
JP2014500865A (ja) 置換イソオキサゾリン化合物及びそれらの前駆体4−クロロベンズアルデヒドオキシム、4−ブロモベンズアルデヒドオキシム又は4−ヨードベンズアルデヒドオキシムを製造するための方法
US20160229820A1 (en) Process for preparing substituted isatoic acid anhydride compounds and derivatives thereof
WO2016071243A1 (en) Process for preparing halogenated alkenone ethers and their use in the synthesis of anthranilamide pesticides
JP2016522234A (ja) ピリジルヒドラジンからピリジルピラゾール化合物及びその誘導体を製造するための方法
KR102790425B1 (ko) 안트라닐산 디아미드의 새로운 제조 방법
JP2016520539A (ja) スルフィミンの製造方法およびそれらのN−(2−アミノ−ベンゾイル)−スルフィミンへのin−situ転化
WO2015162260A1 (en) Process for preparing anthranilamide esters and derivatives

Legal Events

Date Code Title Description
A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20151118

A977 Report on retrieval

Free format text: JAPANESE INTERMEDIATE CODE: A971007

Effective date: 20160630

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20160726

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20161026

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20161122

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20161221

R150 Certificate of patent or registration of utility model

Ref document number: 6067733

Country of ref document: JP

Free format text: JAPANESE INTERMEDIATE CODE: R150

LAPS Cancellation because of no payment of annual fees