CN1026320C - 氮杂环烷衍生物的制备方法 - Google Patents

氮杂环烷衍生物的制备方法 Download PDF

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Publication number
CN1026320C
CN1026320C CN91108088A CN91108088A CN1026320C CN 1026320 C CN1026320 C CN 1026320C CN 91108088 A CN91108088 A CN 91108088A CN 91108088 A CN91108088 A CN 91108088A CN 1026320 C CN1026320 C CN 1026320C
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CN
China
Prior art keywords
ketone
organic solvent
integer
decyl
add
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CN91108088A
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English (en)
Chinese (zh)
Other versions
CN1061592A (zh
Inventor
齐田胜
井上寿孝
八谷照美
八寻重德
野田宽治
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hisamitsu Pharmaceutical Co Inc
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Hisamitsu Pharmaceutical Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hisamitsu Pharmaceutical Co Inc filed Critical Hisamitsu Pharmaceutical Co Inc
Publication of CN1061592A publication Critical patent/CN1061592A/zh
Application granted granted Critical
Publication of CN1026320C publication Critical patent/CN1026320C/zh
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C07D211/76—Oxygen atoms attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/08—Oxygen atoms
    • C07D223/10—Oxygen atoms attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Catalysts (AREA)
CN91108088A 1990-10-31 1991-10-23 氮杂环烷衍生物的制备方法 Expired - Lifetime CN1026320C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2291876A JPH07595B2 (ja) 1990-10-31 1990-10-31 アザシクロアルカン誘導体の製造方法
JP291876/90 1990-10-31

Publications (2)

Publication Number Publication Date
CN1061592A CN1061592A (zh) 1992-06-03
CN1026320C true CN1026320C (zh) 1994-10-26

Family

ID=17774584

Family Applications (1)

Application Number Title Priority Date Filing Date
CN91108088A Expired - Lifetime CN1026320C (zh) 1990-10-31 1991-10-23 氮杂环烷衍生物的制备方法

Country Status (11)

Country Link
US (1) US5371238A (enExample)
EP (1) EP0555483B1 (enExample)
JP (1) JPH07595B2 (enExample)
KR (1) KR960014349B1 (enExample)
CN (1) CN1026320C (enExample)
AT (1) ATE199372T1 (enExample)
AU (1) AU638613B2 (enExample)
CA (1) CA2089880C (enExample)
DE (1) DE69132547T2 (enExample)
ES (1) ES2154632T3 (enExample)
WO (1) WO1992007827A1 (enExample)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0643390B2 (ja) * 1986-04-08 1994-06-08 久光製薬株式会社 アザシクロアルカン誘導体
JPS6330466A (ja) * 1986-07-24 1988-02-09 Hisamitsu Pharmaceut Co Inc アザシクロアルカン化合物

Also Published As

Publication number Publication date
US5371238A (en) 1994-12-06
ES2154632T3 (es) 2001-04-16
AU638613B2 (en) 1993-07-01
CA2089880A1 (en) 1992-05-01
CA2089880C (en) 2002-01-29
CN1061592A (zh) 1992-06-03
KR930702294A (ko) 1993-09-08
WO1992007827A1 (fr) 1992-05-14
DE69132547T2 (de) 2001-06-13
ATE199372T1 (de) 2001-03-15
AU8762491A (en) 1992-05-26
EP0555483B1 (en) 2001-02-28
EP0555483A4 (enExample) 1994-03-23
JPH07595B2 (ja) 1995-01-11
DE69132547D1 (de) 2001-04-05
JPH04169571A (ja) 1992-06-17
KR960014349B1 (ko) 1996-10-15
EP0555483A1 (en) 1993-08-18

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Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
C14 Grant of patent or utility model
GR01 Patent grant
C15 Extension of patent right duration from 15 to 20 years for appl. with date before 31.12.1992 and still valid on 11.12.2001 (patent law change 1993)
OR01 Other related matters
C17 Cessation of patent right
CX01 Expiry of patent term

Expiration termination date: 20111023

Granted publication date: 19941026