CN102388055B - 咪唑并[2,1-b][1,3,4]噻二唑衍生物 - Google Patents

咪唑并[2,1-b][1,3,4]噻二唑衍生物 Download PDF

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CN102388055B
CN102388055B CN201080015246.6A CN201080015246A CN102388055B CN 102388055 B CN102388055 B CN 102388055B CN 201080015246 A CN201080015246 A CN 201080015246A CN 102388055 B CN102388055 B CN 102388055B
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CN102388055A (zh
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华金·帕斯托费尔南德斯
吉多·库尔兹
索尼娅·马丁内斯冈萨雷斯
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Research Centre Foundation Of Carlos Three Generations National Cancer
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    • C—CHEMISTRY; METALLURGY
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    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433—Thidiazoles
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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CN201080015246.6A 2009-04-02 2010-04-01 咪唑并[2,1-b][1,3,4]噻二唑衍生物 Expired - Fee Related CN102388055B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09380069.6 2009-04-02
EP09380069 2009-04-02
PCT/GB2010/000674 WO2010112874A1 (en) 2009-04-02 2010-04-01 Imidazo [2, 1-b] [ 1, 3, 4 ] thiadiazole derivatives

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CN102388055A CN102388055A (zh) 2012-03-21
CN102388055B true CN102388055B (zh) 2015-07-29

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US (1) US8815918B2 (https=)
EP (1) EP2414369B1 (https=)
JP (1) JP5615902B2 (https=)
KR (1) KR101727264B1 (https=)
CN (1) CN102388055B (https=)
AU (1) AU2010231162B2 (https=)
BR (1) BRPI1015367B8 (https=)
CA (1) CA2756873C (https=)
CY (1) CY1116880T1 (https=)
DK (1) DK2414369T3 (https=)
EA (1) EA022753B1 (https=)
ES (1) ES2548571T3 (https=)
HR (1) HRP20151126T1 (https=)
HU (1) HUE027964T2 (https=)
IL (1) IL215158A (https=)
MX (1) MX2011010372A (https=)
NZ (1) NZ595674A (https=)
PL (1) PL2414369T3 (https=)
PT (1) PT2414369E (https=)
SG (1) SG175001A1 (https=)
SI (1) SI2414369T1 (https=)
WO (1) WO2010112874A1 (https=)
ZA (1) ZA201107350B (https=)

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