CN102285947B - 卡巴他赛的合成方法 - Google Patents
卡巴他赛的合成方法 Download PDFInfo
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- CN102285947B CN102285947B CN201110162562.2A CN201110162562A CN102285947B CN 102285947 B CN102285947 B CN 102285947B CN 201110162562 A CN201110162562 A CN 201110162562A CN 102285947 B CN102285947 B CN 102285947B
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- borneol
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- cabazitaxel
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/582—Recycling of unreacted starting or intermediate materials
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
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CN201110162562.2A CN102285947B (zh) | 2011-06-17 | 2011-06-17 | 卡巴他赛的合成方法 |
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CN201110162562.2A CN102285947B (zh) | 2011-06-17 | 2011-06-17 | 卡巴他赛的合成方法 |
Publications (2)
Publication Number | Publication Date |
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CN102285947A CN102285947A (zh) | 2011-12-21 |
CN102285947B true CN102285947B (zh) | 2014-12-03 |
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CN201110162562.2A Active CN102285947B (zh) | 2011-06-17 | 2011-06-17 | 卡巴他赛的合成方法 |
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CN (1) | CN102285947B (zh) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102408397B (zh) * | 2011-10-19 | 2014-08-20 | 上海贝美医药科技有限公司 | 紫杉烷类衍生物及其制备方法 |
WO2013111157A1 (en) * | 2012-01-03 | 2013-08-01 | Shilpa Medicare Limited | Process for preparing amorphous cabazitaxel |
CN102659721B (zh) * | 2012-04-19 | 2014-08-06 | 信泰制药(苏州)有限公司 | 一种卡巴他赛的合成方法 |
CN102675257B (zh) * | 2012-05-10 | 2014-07-02 | 上海金和生物技术有限公司 | 一种卡巴他赛晶体及其制备方法 |
CN102775434B (zh) * | 2012-08-21 | 2015-04-08 | 江苏红豆杉生物科技股份有限公司 | 一种7,10-二甲氧基紫杉烷化合物中间体的合成方法 |
CN102898406B (zh) * | 2012-11-02 | 2014-12-03 | 上海金和生物技术有限公司 | 一种卡巴他赛晶体及其制备方法 |
CA2889448C (en) | 2012-11-09 | 2021-07-06 | Intas Pharmaceuticals Limited | Process for the preparation of cabazitaxel and its intermediates |
KR101407353B1 (ko) * | 2012-12-04 | 2014-06-17 | 주식회사 삼양바이오팜 | 10-디아세틸바카틴 iii으로부터 카바지탁셀을 고수율로 제조하는 새로운 방법 및 이를 위한 신규 중간체 |
CN103058960B (zh) * | 2012-12-12 | 2014-12-10 | 江苏奥赛康药业股份有限公司 | 卡巴他赛多晶型形式及其制备方法 |
CN103044364B (zh) * | 2013-01-07 | 2016-01-20 | 重庆泰濠制药有限公司 | 一种卡巴他赛无定形晶及其制备方法 |
WO2014199401A2 (en) * | 2013-06-14 | 2014-12-18 | Hetero Research Foundation | Process for cabazitaxel |
CN106632158B (zh) * | 2013-08-28 | 2018-11-06 | 江苏恒瑞医药股份有限公司 | 7β,10β-二甲氧基-10-去乙酰基浆果赤霉素III的制备方法 |
CN105461664A (zh) * | 2014-08-21 | 2016-04-06 | 中国医学科学院药物研究所 | 卡巴他赛晶n5型物质及制备方法和其组合物与用途 |
CN105504047A (zh) * | 2016-02-16 | 2016-04-20 | 苏州博源医疗科技有限公司 | 卡巴他赛免疫原、特异性抗体和检测试剂及其制备方法 |
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2011
- 2011-06-17 CN CN201110162562.2A patent/CN102285947B/zh active Active
Non-Patent Citations (2)
Title |
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Gunda I. Georg等.Synthesis, Conformational Analysis, and Biological Evaluation of Heteroaromatic Taxanes.《J. Org. Chem. 1996》.1996,第61卷(第8期),2664-2676. * |
Synthesis, Conformational Analysis, and Biological Evaluation of Heteroaromatic Taxanes;Gunda I. Georg等;《J. Org. Chem. 1996》;19961231;第61卷(第8期);2664-2676 * |
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Publication number | Publication date |
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CN102285947A (zh) | 2011-12-21 |
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Address after: 213016 Baiyun District, Changzhou, Jiangsu Patentee after: Changzhou University Address before: Gehu Lake Road Wujin District 213164 Jiangsu city of Changzhou province No. 1 Patentee before: Changzhou University |
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