CN102046176B - 5-ht3受体调节剂、其制备方法和用途 - Google Patents

5-ht3受体调节剂、其制备方法和用途 Download PDF

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CN102046176B
CN102046176B CN2009801197635A CN200980119763A CN102046176B CN 102046176 B CN102046176 B CN 102046176B CN 2009801197635 A CN2009801197635 A CN 2009801197635A CN 200980119763 A CN200980119763 A CN 200980119763A CN 102046176 B CN102046176 B CN 102046176B
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methyl
quinuclidine
chemical compound
indazole
carboxylate
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CN102046176A (zh
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D·D·曼宁
C·L·乔菲
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Curia Global Inc
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Albany Molecular Research Inc
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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CN2009801197635A 2008-05-29 2009-05-28 5-ht3受体调节剂、其制备方法和用途 Active CN102046176B (zh)

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US5701408P 2008-05-29 2008-05-29
US61/057014 2008-05-29
PCT/US2009/045484 WO2009155054A2 (en) 2008-05-29 2009-05-28 5-ht3 receptor modulators, methods of making, and use thereof

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EP (1) EP2310019A4 (https=)
JP (1) JP5465241B2 (https=)
KR (1) KR101653707B1 (https=)
CN (1) CN102046176B (https=)
AU (1) AU2009260469B2 (https=)
BR (1) BRPI0913188A2 (https=)
CA (1) CA2724449C (https=)
IL (1) IL208939A (https=)
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WO2022110052A1 (zh) * 2020-11-27 2022-06-02 科岭源生物科技(深圳)有限公司 一种含氮杂环类5-ht3受体调节剂及其制备方法和用途
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