CN101928295A - 含有烃基硼酸络合物的抗生素和使用方法 - Google Patents

含有烃基硼酸络合物的抗生素和使用方法 Download PDF

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Publication number
CN101928295A
CN101928295A CN2010101656749A CN201010165674A CN101928295A CN 101928295 A CN101928295 A CN 101928295A CN 2010101656749 A CN2010101656749 A CN 2010101656749A CN 201010165674 A CN201010165674 A CN 201010165674A CN 101928295 A CN101928295 A CN 101928295A
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China
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alkyl
substituted
unsubstituted
aryl
compound
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Pending
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CN2010101656749A
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English (en)
Chinese (zh)
Inventor
万·利
斯蒂芬·J·本科维奇
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Anacor Pharmaceuticals LLC
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Anacor Pharmaceuticals LLC
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Publication of CN101928295A publication Critical patent/CN101928295A/zh
Pending legal-status Critical Current

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/022Boron compounds without C-boron linkages
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN2010101656749A 2002-12-18 2003-12-18 含有烃基硼酸络合物的抗生素和使用方法 Pending CN101928295A (zh)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US43437502P 2002-12-18 2002-12-18
US60/434,375 2002-12-18
US43609502P 2002-12-23 2002-12-23
US60/436,095 2002-12-23
US43784903P 2003-01-03 2003-01-03
US60/437,849 2003-01-03

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CNA2003801089173A Division CN1738802A (zh) 2002-12-18 2003-12-18 含有烃基硼酸络合物的抗生素和使用方法

Publications (1)

Publication Number Publication Date
CN101928295A true CN101928295A (zh) 2010-12-29

Family

ID=32686073

Family Applications (1)

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CN2010101656749A Pending CN101928295A (zh) 2002-12-18 2003-12-18 含有烃基硼酸络合物的抗生素和使用方法

Country Status (11)

Country Link
US (2) US20040224923A1 (https=)
EP (2) EP1980564A1 (https=)
JP (2) JP2006511613A (https=)
KR (1) KR20050084378A (https=)
CN (1) CN101928295A (https=)
AU (1) AU2003299821B2 (https=)
BR (1) BR0317564A (https=)
CA (1) CA2509645A1 (https=)
MX (1) MXPA05006685A (https=)
NZ (1) NZ540870A (https=)
WO (1) WO2004056322A2 (https=)

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CN105473150A (zh) * 2013-08-20 2016-04-06 3M创新有限公司 硼-硅烷聚醚络合物

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WO2006102604A2 (en) * 2005-03-24 2006-09-28 Anacor Pharmaceuticals, Inc. Topical formulations of borinic acid antibodies and their methods of use
CA2635840A1 (en) * 2005-12-28 2007-07-12 Anacor Pharmaceuticals, Inc. Process for manufacturing picolinate borinic esters
KR20080110984A (ko) 2005-12-30 2008-12-22 아나코르 파마슈티칼스 인코포레이티드 보론함유 소분자
PT1988779E (pt) 2006-02-16 2015-09-04 Anacor Pharmaceuticals Inc Moléculas pequenas contendo boro como agentes antiinflamatórios
US20070286822A1 (en) * 2006-06-12 2007-12-13 Anacor Pharmaceuticals Inc. Compounds for the Treatment of Periodontal Disease
RU2008152367A (ru) * 2006-06-12 2010-07-20 Анакор Фармасьютикалз, Инк. (Us) Соединения для лечения периодонтального заболевания
EP2069370A4 (en) * 2006-11-22 2011-05-04 Anacor Pharmaceuticals Inc MICRO-ORGANISMS KILLING COMPOUNDS
KR20150065941A (ko) 2008-03-06 2015-06-15 아나코르 파마슈티칼스 인코포레이티드 소염제로써 붕소가 함유된 소분자
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WO2010045503A1 (en) * 2008-10-15 2010-04-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
WO2010080558A1 (en) * 2008-12-17 2010-07-15 Anacor Pharmaceuticals, Inc. Polymorphs of (s)-3-aminomethyl-7-(3-hydroxy-propoxy)-3h-benzo[c][1,2] oxaborol-1-ol
MX2012001156A (es) 2009-07-28 2012-05-08 Anacor Pharmaceuticals Inc Moleculas que contienen boro trisustituidas.
AP4039A (en) 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
WO2011022337A1 (en) * 2009-08-19 2011-02-24 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110124597A1 (en) * 2009-09-25 2011-05-26 Anacor Pharmaceuticals, Inc. Boron containing small molecules
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US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
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RS64770B1 (sr) 2016-03-07 2023-11-30 Agrofresh Inc Sinergistički postupci upotrebe jedinjenja benzoksaborola i gasova za prezerviranje kao antimikrobnih agenasa za useve
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MA52337A (fr) 2017-03-01 2021-03-03 Anacor Pharmaceuticals Inc Nouveaux analogues d'oxaborole et utilisations de ces derniers
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JP2024509256A (ja) 2021-03-09 2024-02-29 ジュリス ゲルマナス, ヒドロキシキノリン化合物および色素変性剤としての使用方法

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105473150A (zh) * 2013-08-20 2016-04-06 3M创新有限公司 硼-硅烷聚醚络合物

Also Published As

Publication number Publication date
US20080146803A1 (en) 2008-06-19
KR20050084378A (ko) 2005-08-26
EP1581500A2 (en) 2005-10-05
EP1980564A1 (en) 2008-10-15
EP1581500A4 (en) 2008-03-05
CA2509645A1 (en) 2004-07-08
JP2006511613A (ja) 2006-04-06
NZ540870A (en) 2008-09-26
JP2009161540A (ja) 2009-07-23
US20040224923A1 (en) 2004-11-11
WO2004056322A2 (en) 2004-07-08
AU2003299821A1 (en) 2004-07-14
MXPA05006685A (es) 2005-12-14
BR0317564A (pt) 2005-11-22
AU2003299821B2 (en) 2010-02-18
WO2004056322A3 (en) 2004-09-16

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Open date: 20101229