JP2006511613A - ボロン酸複合体を含む抗生物質および使用法 - Google Patents
ボロン酸複合体を含む抗生物質および使用法 Download PDFInfo
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- JP2006511613A JP2006511613A JP2005502662A JP2005502662A JP2006511613A JP 2006511613 A JP2006511613 A JP 2006511613A JP 2005502662 A JP2005502662 A JP 2005502662A JP 2005502662 A JP2005502662 A JP 2005502662A JP 2006511613 A JP2006511613 A JP 2006511613A
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- alkyl
- substituted
- aryl
- unsubstituted
- benzyl
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- CZDYPVPMEAXLPK-UHFFFAOYSA-N tetramethylsilane Chemical compound C[Si](C)(C)C CZDYPVPMEAXLPK-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/022—Boron compounds without C-boron linkages
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43437502P | 2002-12-18 | 2002-12-18 | |
| US43609502P | 2002-12-23 | 2002-12-23 | |
| US43784903P | 2003-01-03 | 2003-01-03 | |
| PCT/US2003/040982 WO2004056322A2 (en) | 2002-12-18 | 2003-12-18 | Antibiotics containing borinic acid complexes and methods of use |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009021716A Division JP2009161540A (ja) | 2002-12-18 | 2009-02-02 | ボロン酸複合体を含む抗生物質および使用法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2006511613A true JP2006511613A (ja) | 2006-04-06 |
Family
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
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| JP2005502662A Withdrawn JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
| JP2009021716A Withdrawn JP2009161540A (ja) | 2002-12-18 | 2009-02-02 | ボロン酸複合体を含む抗生物質および使用法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2009021716A Withdrawn JP2009161540A (ja) | 2002-12-18 | 2009-02-02 | ボロン酸複合体を含む抗生物質および使用法 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20040224923A1 (https=) |
| EP (2) | EP1581500A4 (https=) |
| JP (2) | JP2006511613A (https=) |
| KR (1) | KR20050084378A (https=) |
| CN (1) | CN101928295A (https=) |
| AU (1) | AU2003299821B2 (https=) |
| BR (1) | BR0317564A (https=) |
| CA (1) | CA2509645A1 (https=) |
| MX (1) | MXPA05006685A (https=) |
| NZ (1) | NZ540870A (https=) |
| WO (1) | WO2004056322A2 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018511584A (ja) * | 2015-03-10 | 2018-04-26 | コリア リサーチ インスティテュート オブ ケミカル テクノロジー | ４配位有機ホウ素化合物の製造方法 |
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| JP4138662B2 (ja) | 2002-01-10 | 2008-08-27 | ザ・ペンシルバニア・ステイト・リサーチ・フアウンデイシヨン | アルキルジアリールボリネートおよび錯化ジアリールボロン酸を調製するための方法。 |
| JP2006511613A (ja) * | 2002-12-18 | 2006-04-06 | アナコア ファーマシューティカルズ インコーポレイテッド | ボロン酸複合体を含む抗生物質および使用法 |
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| DE602005017626D1 (de) | 2004-06-14 | 2009-12-24 | Anacor Pharmaceuticals Inc | Antivirale verwendung von borinsäurekomplexen |
| NZ578297A (en) * | 2005-02-16 | 2010-11-26 | Anacor Pharmaceuticals Inc | Boron-containing small molecules |
| BRPI0609728A2 (pt) * | 2005-03-24 | 2010-04-20 | Anacor Pharmaceuticals Inc | formulações tópicas de antibióticos de ácido borìnico e métodos de uso do mesmo |
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| EP1976536A4 (en) | 2005-12-30 | 2011-03-02 | Anacor Pharmaceuticals Inc | SMALL MOLECULES CONTAINING BORON |
| ME02188B (me) | 2006-02-16 | 2016-02-20 | Anacor Pharmaceuticals Inc | Mali molekuli koji sadrže boron kao antiinflamatorni agensi |
| US20070286822A1 (en) * | 2006-06-12 | 2007-12-13 | Anacor Pharmaceuticals Inc. | Compounds for the Treatment of Periodontal Disease |
| RU2008152367A (ru) * | 2006-06-12 | 2010-07-20 | Анакор Фармасьютикалз, Инк. (Us) | Соединения для лечения периодонтального заболевания |
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| WO2017155879A1 (en) | 2016-03-07 | 2017-09-14 | Agrofresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
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| EP3576747A4 (en) * | 2017-03-09 | 2020-12-16 | The Penn State Research Foundation | SMALL MOLECULES CONTAINING BORON TO INHIBIT THE ACTIVITY OF A RECEPTOR-TYPE PROTEIN TYROSINE PHOSPHATASE |
| CN112867436A (zh) * | 2018-08-20 | 2021-05-28 | 传感技术股份有限公司 | 用于减少体内分析物指示物降解的调节药物释放 |
| EP4204012A1 (en) | 2020-08-31 | 2023-07-05 | Pfizer Inc. | Methods of protecting rna |
| JP2024509256A (ja) | 2021-03-09 | 2024-02-29 | ジュリス ゲルマナス， | ヒドロキシキノリン化合物および色素変性剤としての使用方法 |
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-
2003
- 2003-12-18 JP JP2005502662A patent/JP2006511613A/ja not_active Withdrawn
- 2003-12-18 MX MXPA05006685A patent/MXPA05006685A/es active IP Right Grant
- 2003-12-18 EP EP03800095A patent/EP1581500A4/en not_active Withdrawn
- 2003-12-18 WO PCT/US2003/040982 patent/WO2004056322A2/en not_active Ceased
- 2003-12-18 CN CN2010101656749A patent/CN101928295A/zh active Pending
- 2003-12-18 EP EP08155302A patent/EP1980564A1/en not_active Withdrawn
- 2003-12-18 KR KR1020057011194A patent/KR20050084378A/ko not_active Ceased
- 2003-12-18 AU AU2003299821A patent/AU2003299821B2/en not_active Ceased
- 2003-12-18 CA CA002509645A patent/CA2509645A1/en not_active Abandoned
- 2003-12-18 US US10/740,304 patent/US20040224923A1/en not_active Abandoned
- 2003-12-18 NZ NZ540870A patent/NZ540870A/en not_active IP Right Cessation
- 2003-12-18 BR BR0317564-2A patent/BR0317564A/pt not_active IP Right Cessation
-
2007
- 2007-09-06 US US11/851,259 patent/US20080146803A1/en not_active Abandoned
-
2009
- 2009-02-02 JP JP2009021716A patent/JP2009161540A/ja not_active Withdrawn
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US5318947A (en) * | 1989-10-18 | 1994-06-07 | Hoechst Aktiengesellschaft | Method for controlling harmful plants in rice with 2-benzoyl-1,3-cyclohexanedione derivatives |
| US5348947A (en) * | 1993-05-07 | 1994-09-20 | American Cyanamid Company | Diarylboron ester and thioester fungicidal agents |
| JPH0952893A (ja) * | 1995-08-10 | 1997-02-25 | Yoshitomi Pharmaceut Ind Ltd | キノロンカルボン酸誘導体の工業的な製造法およびその合成中間体 |
| WO2000044387A1 (fr) * | 1999-01-29 | 2000-08-03 | Nitto Kasei Co., Ltd. | Composes organobores presentant une activite de coccidiostats |
| JP2002322007A (ja) * | 2001-04-27 | 2002-11-08 | Shionogi & Co Ltd | 有機ホウ素化合物を含有する植物用殺線虫剤 |
| JP2005515229A (ja) * | 2002-01-10 | 2005-05-26 | ザ・ペンシルバニア・ステイト・リサーチ・フアウンデイシヨン | アルキルジアリールボリネートおよび錯化ジアリールボロン酸を調製するための方法。 |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018511584A (ja) * | 2015-03-10 | 2018-04-26 | コリア リサーチ インスティテュート オブ ケミカル テクノロジー | ４配位有機ホウ素化合物の製造方法 |
| US10689403B2 (en) | 2015-03-10 | 2020-06-23 | Korea Research Institute Of Chemical Technology | Method for preparing four-coordinated organic boron compound |
Also Published As
| Publication number | Publication date |
|---|---|
| US20080146803A1 (en) | 2008-06-19 |
| CA2509645A1 (en) | 2004-07-08 |
| BR0317564A (pt) | 2005-11-22 |
| CN101928295A (zh) | 2010-12-29 |
| WO2004056322A3 (en) | 2004-09-16 |
| US20040224923A1 (en) | 2004-11-11 |
| WO2004056322A2 (en) | 2004-07-08 |
| MXPA05006685A (es) | 2005-12-14 |
| EP1581500A4 (en) | 2008-03-05 |
| AU2003299821A1 (en) | 2004-07-14 |
| NZ540870A (en) | 2008-09-26 |
| JP2009161540A (ja) | 2009-07-23 |
| AU2003299821B2 (en) | 2010-02-18 |
| EP1581500A2 (en) | 2005-10-05 |
| EP1980564A1 (en) | 2008-10-15 |
| KR20050084378A (ko) | 2005-08-26 |
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