BR0317564A - Compostos, composições e métodos para tratar doenças causadas por bactérias ou fungos - Google Patents

Compostos, composições e métodos para tratar doenças causadas por bactérias ou fungos

Info

Publication number
BR0317564A
BR0317564A BR0317564-2A BR0317564A BR0317564A BR 0317564 A BR0317564 A BR 0317564A BR 0317564 A BR0317564 A BR 0317564A BR 0317564 A BR0317564 A BR 0317564A
Authority
BR
Brazil
Prior art keywords
compositions
methods
compounds
fungal diseases
treating bacterial
Prior art date
Application number
BR0317564-2A
Other languages
English (en)
Inventor
Ving Lee
Stephen J Benkovic
Original Assignee
Anacor Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals Inc filed Critical Anacor Pharmaceuticals Inc
Publication of BR0317564A publication Critical patent/BR0317564A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/022—Boron compounds without C-boron linkages
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"COMPOSTOS, COMPOSIçõES E MéTODOS PARA TRATAR DOENçAS CAUSADAS POR BACTéRIAS OU FUNGOS". A estrutura e preparação de antibióticos, incorporando complexos de ácido borínico, são revelados, especialmente hidroxiquinolina, derivados de imidazóis e ácido picolínico, juntamente com composições desses antibióticos e métodos de uso dos antibióticos e composições como agentes bactericidas e fungicidas, bem como agentes terapêuticos para o tratamento de enfermidades causadas por bactérias e fungos.
BR0317564-2A 2002-12-18 2003-12-18 Compostos, composições e métodos para tratar doenças causadas por bactérias ou fungos BR0317564A (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US43437502P 2002-12-18 2002-12-18
US43609502P 2002-12-23 2002-12-23
US43784903P 2003-01-03 2003-01-03
PCT/US2003/040982 WO2004056322A2 (en) 2002-12-18 2003-12-18 Antibiotics containing borinic acid complexes and methods of use

Publications (1)

Publication Number Publication Date
BR0317564A true BR0317564A (pt) 2005-11-22

Family

ID=32686073

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0317564-2A BR0317564A (pt) 2002-12-18 2003-12-18 Compostos, composições e métodos para tratar doenças causadas por bactérias ou fungos

Country Status (11)

Country Link
US (2) US20040224923A1 (pt)
EP (2) EP1980564A1 (pt)
JP (2) JP2006511613A (pt)
KR (1) KR20050084378A (pt)
CN (1) CN101928295A (pt)
AU (1) AU2003299821B2 (pt)
BR (1) BR0317564A (pt)
CA (1) CA2509645A1 (pt)
MX (1) MXPA05006685A (pt)
NZ (1) NZ540870A (pt)
WO (1) WO2004056322A2 (pt)

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US7390806B2 (en) 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
EP1980564A1 (en) * 2002-12-18 2008-10-15 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use
AR049915A1 (es) * 2004-06-14 2006-09-13 Anacor Pharmaceuticals Inc Compuestos con contenido de boro y metodos de uso de los mismos
AR049916A1 (es) * 2004-06-14 2006-09-13 Anacor Pharmaceuticals Inc Usos anti-parasitarios de complejos de acido borinico
DE602005017626D1 (de) 2004-06-14 2009-12-24 Anacor Pharmaceuticals Inc Antivirale verwendung von borinsäurekomplexen
CA2597982C (en) 2005-02-16 2014-07-08 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US7767657B2 (en) 2005-02-16 2010-08-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
CN101522200A (zh) * 2005-03-24 2009-09-02 安纳考尔医药公司 二取代硼酸抗生素局部制剂及其使用方法
JP2009522274A (ja) * 2005-12-28 2009-06-11 アナコール ファーマシューティカルズ，インコーポレイテッド ピコリネートボリン酸エステル類の製造方法
SI2719388T1 (sl) 2006-02-16 2019-06-28 Anacor Pharmaceuticals, Inc. Majhne molekule, polnjene z borom, kot učinkovine proti vnetjem
WO2007146965A2 (en) * 2006-06-12 2007-12-21 Anacor Pharmaceuticals, Inc. Compounds for the treatment of periodontal disease
US20070286822A1 (en) * 2006-06-12 2007-12-13 Anacor Pharmaceuticals Inc. Compounds for the Treatment of Periodontal Disease
EP2069370A4 (en) * 2006-11-22 2011-05-04 Anacor Pharmaceuticals Inc MICROORGANISM DESTRUCTIVE COMPOUNDS
MX2010009765A (es) 2008-03-06 2013-07-12 Anacor Pharmaceuticals Inc Moleculas pequeñas que contienen boro como agentes anti-inflamatorios.
EP2285384A4 (en) * 2008-05-12 2012-04-25 Anacor Pharmaceuticals Inc BORN SMALL MOLECULES
EP2348863A4 (en) 2008-09-04 2012-03-07 Anacor Pharmaceuticals Inc BORN SMALL MOLECULES
WO2010028005A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US9493489B2 (en) 2008-10-15 2016-11-15 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
EP2378886A4 (en) 2008-12-17 2012-08-29 Anacor Pharmaceuticals Inc (S) -3-Aminomethyl-7- (3-hydroxypropoxy) -3H-benzo [c] [1,2] oxaborole-1-OL-POLYMORPHS
BR112012001987A2 (pt) 2009-07-28 2015-09-01 Anacor Pharmaceuticals Inc Composto, combinação, formulação farmacêutica, uso de um composto, uma combinação ou um sal farmaceuticamente aceitável dos mesmos, e, métodos para tratar uma infecção bacteriana, para matar ou inibir o crescimento de uma bactéria, e para inibir uma beta-lactamase.
AP4039A (en) 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
WO2011022337A1 (en) * 2009-08-19 2011-02-24 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110124597A1 (en) * 2009-09-25 2011-05-26 Anacor Pharmaceuticals, Inc. Boron containing small molecules
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110212918A1 (en) 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
AP2012006482A0 (en) 2010-03-19 2012-10-31 Anacor Pharmacueticals Inc Boron-containing small molecules as anti-protozoalagent
JP5952280B2 (ja) 2010-09-07 2016-07-13 アナコール ファーマシューティカルズ，インコーポレーテッド 細菌感染治療用のベンゾオキサボロール誘導体
CN107646865B (zh) 2013-01-30 2020-07-03 美国陶氏益农公司 苯硼酸半酯作为挥发性抗微生物剂在肉类、植物或植物部分上的用途
US8669207B1 (en) 2013-01-30 2014-03-11 Dow Agrosciences, Llc. Compounds and compositions
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US9585396B2 (en) 2013-01-30 2017-03-07 Agrofresh Inc. Volatile applications against pathogens
BR112016003692B1 (pt) * 2013-08-20 2022-02-08 3M Innovative Properties Company Complexo poliéter boro-silano
KR101756785B1 (ko) * 2015-03-10 2017-07-12 한국화학연구원 4배위 유기 붕소 화합물의 제조방법
TW201735792A (zh) 2016-03-07 2017-10-16 農業保鮮股份有限公司 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法
US11447506B2 (en) 2016-05-09 2022-09-20 Anacor Pharmaceuticals, Inc. Crystal forms of crisaborole in free form and preparation method and use thereof
IL248149B (en) 2016-09-29 2020-03-31 Garti Nissim Formulations of dilutable cannabinoids and processes for their preparation
IL248150B (en) 2016-09-29 2018-05-31 Garti Nissim A method for selective extraction of cannabinoid from plant origin
EA201992153A1 (ru) * 2016-10-05 2020-02-25 Зе Глобал Эллайенс Фо Тб Драг Девелопмент, Инк. Гетероарилтрифторборатные соединения для лечения микобактериальных инфекций
US10961261B2 (en) 2017-03-01 2021-03-30 Anacor Pharmaceuticals, Inc. Oxaborole analogs and uses thereof
US10973835B2 (en) * 2017-03-09 2021-04-13 The Penn State Research Foundation Boron-containing small molecules for inhibiting activity of a receptor-like protein tyrosine phosphatase
EP3840637A4 (en) * 2018-08-20 2022-05-18 Senseonics, Incorporated INDUCED DRUG RELEASE TO REDUCE ANALYTE INDICATOR DEGRADATION IN VIVO
EP4204012A1 (en) 2020-08-31 2023-07-05 Pfizer Inc. Methods of protecting rna
WO2022192385A1 (en) * 2021-03-09 2022-09-15 Germannas Juris Hyrdroxyquinoline compounds and methods of use as pigment modifying agents

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US7390806B2 (en) * 2002-12-18 2008-06-24 Anacor Pharmaceuticals, Inc. Antibiotics containing borinic acid complexes and methods of use

Also Published As

Publication number Publication date
EP1980564A1 (en) 2008-10-15
WO2004056322A3 (en) 2004-09-16
MXPA05006685A (es) 2005-12-14
US20040224923A1 (en) 2004-11-11
CN101928295A (zh) 2010-12-29
US20080146803A1 (en) 2008-06-19
EP1581500A2 (en) 2005-10-05
AU2003299821B2 (en) 2010-02-18
NZ540870A (en) 2008-09-26
KR20050084378A (ko) 2005-08-26
WO2004056322A2 (en) 2004-07-08
JP2009161540A (ja) 2009-07-23
JP2006511613A (ja) 2006-04-06
CA2509645A1 (en) 2004-07-08
EP1581500A4 (en) 2008-03-05
AU2003299821A1 (en) 2004-07-14

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08L Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette]

Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 9A E 10A ANUIDADES.

B08I Publication cancelled [chapter 8.9 patent gazette]

Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2257 DE 08/04/2014 POR TER SIDO INDEVIDA.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 9A, 10A, 11A, 12A, 13A, 14A, 15A E 16A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2602 DE 17-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.