CN101687873A - 具有稠合杂环的11β-羟基类固醇Ⅰ型脱氢酶抑制剂 - Google Patents
具有稠合杂环的11β-羟基类固醇Ⅰ型脱氢酶抑制剂 Download PDFInfo
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- CN101687873A CN101687873A CN200880020554A CN200880020554A CN101687873A CN 101687873 A CN101687873 A CN 101687873A CN 200880020554 A CN200880020554 A CN 200880020554A CN 200880020554 A CN200880020554 A CN 200880020554A CN 101687873 A CN101687873 A CN 101687873A
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Classifications
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- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
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Landscapes
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| US4495108P | 2008-04-15 | 2008-04-15 | |
| US61/044,951 | 2008-04-15 | ||
| PCT/US2008/060395 WO2008130951A1 (en) | 2007-04-17 | 2008-04-16 | Fused heterocyclic 11-beta-hydroxysteroid dehydrogenase type i inhibitors |
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| TW201107329A (en) * | 2009-07-30 | 2011-03-01 | Oncotherapy Science Inc | Fused imidazole derivative having ttk inhibitory action |
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| PH12012501361A1 (en) | 2009-12-31 | 2012-10-22 | Centro Nac De Investigaciones Oncologicas Cnio | Tricyclic compounds for use as kinase inhibitors |
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| US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
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| TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
| TWI526441B (zh) | 2010-08-20 | 2016-03-21 | 中外製藥股份有限公司 | 包含四環化合物的組成物 |
| TWI541243B (zh) * | 2010-09-10 | 2016-07-11 | 拜耳知識產權公司 | 經取代咪唑并嗒 |
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| EP2760862B1 (en) | 2011-09-27 | 2015-10-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| US8785435B2 (en) | 2011-10-20 | 2014-07-22 | Hoffmann-La Roche Inc. | Solid forms |
| SG11201502211QA (en) | 2012-09-25 | 2015-05-28 | Chugai Pharmaceutical Co Ltd | Ret inhibitor |
| US9422290B2 (en) | 2012-11-13 | 2016-08-23 | Boehringer Ingelheim International Gmbh | Triazolopyridazine |
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| US9527835B2 (en) | 2014-02-13 | 2016-12-27 | Incyte Corporation | Cyclopropylamines as LSD1 inhibitors |
| EP3105219B9 (en) | 2014-02-13 | 2018-10-03 | Incyte Corporation | Cyclopropylamines as lsd1 inhibitors |
| PT3105218T (pt) | 2014-02-13 | 2019-12-05 | Incyte Corp | Ciclopropilaminas como inibidores de lsd1 |
| MX386901B (es) | 2014-04-25 | 2025-03-19 | Chugai Pharmaceutical Co Ltd | Formulacion que contiene una gran cantidad de compuesto tetraciclico. |
| CN113416179A (zh) | 2014-04-25 | 2021-09-21 | 中外制药株式会社 | 四环化合物的新结晶 |
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| TWI803187B (zh) | 2014-08-08 | 2023-05-21 | 日商中外製藥股份有限公司 | 包含４環性化合物的非晶質體之固體分散體及製劑 |
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-
2008
- 2008-04-16 US US12/595,524 patent/US8546394B2/en active Active
- 2008-04-16 EP EP08745903.8A patent/EP2142551B1/en not_active Not-in-force
- 2008-04-16 EP EP12163063A patent/EP2474549A1/en not_active Withdrawn
- 2008-04-16 JP JP2010504198A patent/JP2010524953A/ja not_active Withdrawn
- 2008-04-16 CN CN200880020554A patent/CN101687873A/zh active Pending
- 2008-04-16 WO PCT/US2008/060395 patent/WO2008130951A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| US8546394B2 (en) | 2013-10-01 |
| US20100144744A1 (en) | 2010-06-10 |
| EP2474549A1 (en) | 2012-07-11 |
| EP2142551B1 (en) | 2015-10-14 |
| WO2008130951A1 (en) | 2008-10-30 |
| EP2142551A1 (en) | 2010-01-13 |
| JP2010524953A (ja) | 2010-07-22 |
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Application publication date: 20100331 |