CL2014000992A1 - Preparacion de liberacion sostenida que comprende pioglitazona o una sal de esta; metodo de preparacion; uso para prevenir y/o retardar el inicio o suprimir la progresion de la enfermedad de alzheimer. - Google Patents

Preparacion de liberacion sostenida que comprende pioglitazona o una sal de esta; metodo de preparacion; uso para prevenir y/o retardar el inicio o suprimir la progresion de la enfermedad de alzheimer.

Info

Publication number
CL2014000992A1
CL2014000992A1 CL2014000992A CL2014000992A CL2014000992A1 CL 2014000992 A1 CL2014000992 A1 CL 2014000992A1 CL 2014000992 A CL2014000992 A CL 2014000992A CL 2014000992 A CL2014000992 A CL 2014000992A CL 2014000992 A1 CL2014000992 A1 CL 2014000992A1
Authority
CL
Chile
Prior art keywords
preparation
pioglitazone
alzheimer
onset
progression
Prior art date
Application number
CL2014000992A
Other languages
English (en)
Spanish (es)
Inventor
Yumiko Ishii
Yutaka Tanque
Yusuke Murakawa
Kaoru Takenaka
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47178262&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2014000992(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of CL2014000992A1 publication Critical patent/CL2014000992A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biomedical Technology (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CL2014000992A 2011-10-21 2014-04-17 Preparacion de liberacion sostenida que comprende pioglitazona o una sal de esta; metodo de preparacion; uso para prevenir y/o retardar el inicio o suprimir la progresion de la enfermedad de alzheimer. CL2014000992A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2011232302 2011-10-21

Publications (1)

Publication Number Publication Date
CL2014000992A1 true CL2014000992A1 (es) 2014-09-05

Family

ID=47178262

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2014000992A CL2014000992A1 (es) 2011-10-21 2014-04-17 Preparacion de liberacion sostenida que comprende pioglitazona o una sal de esta; metodo de preparacion; uso para prevenir y/o retardar el inicio o suprimir la progresion de la enfermedad de alzheimer.

Country Status (30)

Country Link
US (1) US9907789B2 (cg-RX-API-DMAC7.html)
EP (1) EP2768487B1 (cg-RX-API-DMAC7.html)
JP (1) JP6093762B2 (cg-RX-API-DMAC7.html)
KR (1) KR20140081826A (cg-RX-API-DMAC7.html)
CN (1) CN104039313A (cg-RX-API-DMAC7.html)
AP (1) AP2014007645A0 (cg-RX-API-DMAC7.html)
AR (1) AR088398A1 (cg-RX-API-DMAC7.html)
AU (1) AU2012326976B2 (cg-RX-API-DMAC7.html)
BR (1) BR112014008744A2 (cg-RX-API-DMAC7.html)
CA (1) CA2852417A1 (cg-RX-API-DMAC7.html)
CL (1) CL2014000992A1 (cg-RX-API-DMAC7.html)
CO (1) CO6960544A2 (cg-RX-API-DMAC7.html)
CR (1) CR20140213A (cg-RX-API-DMAC7.html)
DO (1) DOP2014000077A (cg-RX-API-DMAC7.html)
EA (1) EA201490840A1 (cg-RX-API-DMAC7.html)
EC (1) ECSP14013328A (cg-RX-API-DMAC7.html)
IL (1) IL232114A0 (cg-RX-API-DMAC7.html)
IN (1) IN2014DN03169A (cg-RX-API-DMAC7.html)
MA (1) MA35717B1 (cg-RX-API-DMAC7.html)
MX (1) MX2014004679A (cg-RX-API-DMAC7.html)
NZ (1) NZ624275A (cg-RX-API-DMAC7.html)
PE (1) PE20141189A1 (cg-RX-API-DMAC7.html)
PH (1) PH12014500856A1 (cg-RX-API-DMAC7.html)
SG (2) SG2014012025A (cg-RX-API-DMAC7.html)
TN (1) TN2014000152A1 (cg-RX-API-DMAC7.html)
TW (1) TW201323018A (cg-RX-API-DMAC7.html)
UA (1) UA113858C2 (cg-RX-API-DMAC7.html)
UY (1) UY34403A (cg-RX-API-DMAC7.html)
WO (1) WO2013058409A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA201403103B (cg-RX-API-DMAC7.html)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112014008744A2 (pt) 2011-10-21 2017-04-18 Takeda Pharmaceuticals Co preparação de libertação prolongada, e, métodos para produzir uma preparação de liberação prolongada, e para prevenir e/ou retardar o início ou suprimir a progressão da doença de alzheimer
SG11201401189WA (en) 2012-04-20 2014-09-26 Gilead Sciences Inc Benzothiazol- 6 -yl acetic acid derivatives and their use for treating an hiv infection
US20150141517A1 (en) * 2013-11-15 2015-05-21 Shin-Etsu Chemical Co., Ltd. Granulated composite, rapid release tablet and method for producing same
KR102485766B1 (ko) 2019-12-11 2023-01-09 한국유나이티드제약 주식회사 생체이용률이 향상된 피오글리타존 함유 약학조성물
UY39094A (es) * 2020-02-27 2021-07-30 Hk Inno N Corp Composición farmacéutica que comprende compuesto derivado de bencimidazol
JP2023066053A (ja) * 2021-10-28 2023-05-15 東和薬品株式会社 放出制御医薬組成物
WO2025064867A1 (en) * 2023-09-21 2025-03-27 Yuva Biosciences, Inc. Delivery system for mitochondrial health enhancers

Family Cites Families (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4810502A (en) 1987-02-27 1989-03-07 Alza Corporation Pseudoephedrine brompheniramine therapy
US4820522A (en) 1987-07-27 1989-04-11 Mcneilab, Inc. Oral sustained release acetaminophen formulation and process
JPH0624991A (ja) 1991-06-20 1994-02-01 Tokyo Tanabe Co Ltd ウルソデスオキシコール酸持続性製剤
JPH0624959A (ja) 1991-10-04 1994-02-01 Bayer Yakuhin Kk 胃内浮遊型薬物徐放性固形製剤
DK0661045T3 (da) 1992-09-18 2002-10-28 Yamanouchi Pharma Co Ltd Hydrogelpræparat med forsinket frigivelse
JPH06316517A (ja) 1993-02-22 1994-11-15 Grelan Pharmaceut Co Ltd 放出制御製剤
AU8532798A (en) 1997-06-13 1998-12-30 Roland Bodmeier Compounds which delay the release of active substances
US6191154B1 (en) * 1998-11-27 2001-02-20 Case Western Reserve University Compositions and methods for the treatment of Alzheimer's disease, central nervous system injury, and inflammatory diseases
WO2003013609A1 (fr) 2001-08-03 2003-02-20 Takeda Chemical Industries, Ltd. Medicaments a liberation continue
US9060941B2 (en) 2002-09-20 2015-06-23 Actavis, Inc. Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
EP2604266A1 (en) 2002-09-20 2013-06-19 Andrx Labs Llc Novel pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
JP4493970B2 (ja) 2002-10-16 2010-06-30 武田薬品工業株式会社 持続性製剤
MY148805A (en) 2002-10-16 2013-05-31 Takeda Pharmaceutical Controlled release preparation
IN192749B (cg-RX-API-DMAC7.html) 2002-11-15 2004-05-15 Ranbaxy Lab Ltd
US7442387B2 (en) 2003-03-06 2008-10-28 Astellas Pharma Inc. Pharmaceutical composition for controlled release of active substances and manufacturing method thereof
EP1607088B1 (en) 2003-03-17 2019-02-27 Takeda Pharmaceutical Company Limited Controlled release composition
JP4933033B2 (ja) 2003-03-17 2012-05-16 武田薬品工業株式会社 放出制御組成物
JP2005015477A (ja) 2003-06-06 2005-01-20 Takeda Chem Ind Ltd 固形製剤
CA2528164A1 (en) 2003-06-06 2004-12-16 Takeda Pharmaceutical Company Limited Solid preparation
US20060003002A1 (en) 2003-11-03 2006-01-05 Lipocine, Inc. Pharmaceutical compositions with synchronized solubilizer release
WO2005099760A1 (ja) 2004-04-14 2005-10-27 Takeda Pharmaceutical Company Limited 固形製剤
MX2007002375A (es) 2004-08-31 2007-04-23 Pfizer Prod Inc Formas de dosificacion de liberacion controlada combinando liberacion inmediata y liberacion sostenida de un farmaco de baja solubilidad.
TW200803851A (en) 2005-09-22 2008-01-16 Sb Pharmco Inc Pharmaceutical composition for improvement of cognitive function
WO2007054976A2 (en) 2005-11-08 2007-05-18 Panacea Biotec Ltd. Lipid based controlled release pharmaceutical composition
AU2006328328B2 (en) 2005-12-22 2012-08-30 Takeda Pharmaceutical Company Limited Solid preparation containing an insulin sensitizer
AU2007232836B2 (en) 2006-03-30 2012-12-06 Nippon Zoki Pharmaceutical Co., Ltd. Solid pharmaceutical preparation
JP2009534292A (ja) 2006-04-27 2009-09-24 武田薬品工業株式会社 塩酸ピオグリタゾンを有するアンジオテンシンii拮抗薬の医薬組成物
DK2120878T3 (da) 2007-02-09 2014-11-03 Alphapharm Pty Ltd Doseringsform indeholdende to aktive farmaceutiske ingredienser i forskellige fysiske former
TW200914006A (en) * 2007-07-12 2009-04-01 Takeda Pharmaceutical Coated preparation
CN101269040A (zh) 2008-05-16 2008-09-24 北京正大绿洲医药科技有限公司 盐酸吡格列酮缓释滴丸及其制备方法
US8445190B2 (en) 2008-09-30 2013-05-21 The Trustees Of The University Of Pennsylvania Method of inhibiting biomaterial-induced procoagulant activity using complement inhibitors
TWI478712B (zh) 2008-09-30 2015-04-01 Astellas Pharma Inc 釋控性醫藥組成物
WO2011049309A2 (ko) 2009-10-09 2011-04-28 영진약품공업 주식회사 속효성과 지속성을 동시에 갖는 약제학적 조성물
JP2011232302A (ja) 2010-04-30 2011-11-17 Ricoh Elemex Corp 画像検査方法及び画像検査装置
CN101884627B (zh) * 2010-07-07 2012-01-25 青岛黄海制药有限责任公司 盐酸吡格列酮胃内滞留缓释片及其制备方法
KR102171747B1 (ko) * 2011-01-10 2020-11-04 진판델 파마슈티컬스 인코포레이티드 알츠하이머 병 치료를 위한 방법 및 약품
BR112014008744A2 (pt) 2011-10-21 2017-04-18 Takeda Pharmaceuticals Co preparação de libertação prolongada, e, métodos para produzir uma preparação de liberação prolongada, e para prevenir e/ou retardar o início ou suprimir a progressão da doença de alzheimer
KR20160056691A (ko) 2014-11-12 2016-05-20 삼성에스디아이 주식회사 이차전지

Also Published As

Publication number Publication date
AU2012326976A1 (en) 2014-05-29
KR20140081826A (ko) 2014-07-01
SG2014012025A (en) 2014-06-27
EP2768487A1 (en) 2014-08-27
DOP2014000077A (es) 2014-07-15
BR112014008744A2 (pt) 2017-04-18
ECSP14013328A (es) 2014-05-31
ZA201403103B (en) 2015-08-26
UY34403A (es) 2013-05-31
CO6960544A2 (es) 2014-05-30
IN2014DN03169A (cg-RX-API-DMAC7.html) 2015-05-22
WO2013058409A1 (en) 2013-04-25
AR088398A1 (es) 2014-05-28
CN104039313A (zh) 2014-09-10
MA35717B1 (fr) 2014-12-01
US20140248362A1 (en) 2014-09-04
AU2012326976B2 (en) 2017-08-17
CR20140213A (es) 2014-06-18
EP2768487B1 (en) 2020-06-03
JP6093762B2 (ja) 2017-03-08
SG10201700121YA (en) 2017-03-30
MX2014004679A (es) 2014-08-01
IL232114A0 (en) 2014-06-30
EA201490840A1 (ru) 2014-08-29
PE20141189A1 (es) 2014-09-24
AP2014007645A0 (en) 2014-05-31
PH12014500856A1 (en) 2014-05-19
UA113858C2 (uk) 2017-03-27
CA2852417A1 (en) 2013-04-25
NZ624275A (en) 2016-09-30
TN2014000152A1 (en) 2015-09-30
AU2012326976A2 (en) 2014-06-12
JP2014530802A (ja) 2014-11-20
US9907789B2 (en) 2018-03-06
TW201323018A (zh) 2013-06-16

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