CL2011000317A1 - Combinacion que comprende (1r,2r)-3-(3-dimetilamino-1-etil-2-metil-propil)-fenol y al menos un antiepileptico seleccionado del grupo que consiste de pregabalina, gabapentina, topiramato, lamotrigina, carbamazepina, lacosamida, levetiracetam y retigabina; composicion farmaceutica; forma de dosificacion; util para tratar el dolor. - Google Patents

Combinacion que comprende (1r,2r)-3-(3-dimetilamino-1-etil-2-metil-propil)-fenol y al menos un antiepileptico seleccionado del grupo que consiste de pregabalina, gabapentina, topiramato, lamotrigina, carbamazepina, lacosamida, levetiracetam y retigabina; composicion farmaceutica; forma de dosificacion; util para tratar el dolor.

Info

Publication number
CL2011000317A1
CL2011000317A1 CL2011000317A CL2011000317A CL2011000317A1 CL 2011000317 A1 CL2011000317 A1 CL 2011000317A1 CL 2011000317 A CL2011000317 A CL 2011000317A CL 2011000317 A CL2011000317 A CL 2011000317A CL 2011000317 A1 CL2011000317 A1 CL 2011000317A1
Authority
CL
Chile
Prior art keywords
dimethylamino
phenol
propyl
ethyl
methyl
Prior art date
Application number
CL2011000317A
Other languages
English (en)
Spanish (es)
Inventor
Petra Bloms-Funke
Klaus Schiene
Christoph Thomas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40345058&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2011000317(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of CL2011000317A1 publication Critical patent/CL2011000317A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0021Intradermal administration, e.g. through microneedle arrays, needleless injectors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
CL2011000317A 2008-09-05 2011-02-14 Combinacion que comprende (1r,2r)-3-(3-dimetilamino-1-etil-2-metil-propil)-fenol y al menos un antiepileptico seleccionado del grupo que consiste de pregabalina, gabapentina, topiramato, lamotrigina, carbamazepina, lacosamida, levetiracetam y retigabina; composicion farmaceutica; forma de dosificacion; util para tratar el dolor. CL2011000317A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP08015625 2008-09-05

Publications (1)

Publication Number Publication Date
CL2011000317A1 true CL2011000317A1 (es) 2011-06-17

Family

ID=40345058

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2011000317A CL2011000317A1 (es) 2008-09-05 2011-02-14 Combinacion que comprende (1r,2r)-3-(3-dimetilamino-1-etil-2-metil-propil)-fenol y al menos un antiepileptico seleccionado del grupo que consiste de pregabalina, gabapentina, topiramato, lamotrigina, carbamazepina, lacosamida, levetiracetam y retigabina; composicion farmaceutica; forma de dosificacion; util para tratar el dolor.

Country Status (28)

Country Link
US (1) US20100063148A1 (OSRAM)
EP (2) EP2735338B1 (OSRAM)
JP (4) JP5731387B2 (OSRAM)
KR (3) KR101641519B1 (OSRAM)
CN (2) CN105520924B (OSRAM)
AR (2) AR073361A1 (OSRAM)
AU (3) AU2009289776A1 (OSRAM)
BR (1) BRPI0920521A2 (OSRAM)
CA (1) CA2735857C (OSRAM)
CL (1) CL2011000317A1 (OSRAM)
CO (1) CO6382142A2 (OSRAM)
CY (2) CY1115751T1 (OSRAM)
DK (2) DK2331210T3 (OSRAM)
EC (1) ECSP11010869A (OSRAM)
ES (2) ES2719900T3 (OSRAM)
HR (2) HRP20140663T1 (OSRAM)
HU (1) HUE043278T2 (OSRAM)
IL (3) IL211135A (OSRAM)
LT (1) LT2735338T (OSRAM)
MX (1) MX2011002339A (OSRAM)
PE (5) PE20142357A1 (OSRAM)
PL (2) PL2735338T3 (OSRAM)
PT (2) PT2331210E (OSRAM)
RU (2) RU2674150C1 (OSRAM)
SI (2) SI2331210T1 (OSRAM)
TR (1) TR201904388T4 (OSRAM)
WO (1) WO2010025931A2 (OSRAM)
ZA (1) ZA201101449B (OSRAM)

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Also Published As

Publication number Publication date
AU2016203053B2 (en) 2018-01-25
PT2735338T (pt) 2019-05-24
IL237392A0 (en) 2015-04-30
PT2331210E (pt) 2014-08-25
US20100063148A1 (en) 2010-03-11
CO6382142A2 (es) 2012-02-15
TR201904388T4 (tr) 2019-05-21
PE20110291A1 (es) 2011-06-04
JP2015096530A (ja) 2015-05-21
EP2735338B1 (en) 2019-02-06
KR101851120B1 (ko) 2018-04-23
ES2719900T3 (es) 2019-07-16
CA2735857C (en) 2019-05-28
PL2735338T3 (pl) 2019-07-31
JP2017071636A (ja) 2017-04-13
JP2012501986A (ja) 2012-01-26
CN102159284B (zh) 2015-12-09
CY1115751T1 (el) 2017-01-25
RU2571501C2 (ru) 2015-12-20
AU2016203053A1 (en) 2016-06-02
EP2331210B1 (en) 2014-07-09
AU2018202879B2 (en) 2020-03-12
JP2019131578A (ja) 2019-08-08
BRPI0920521A2 (pt) 2018-01-16
ES2513394T3 (es) 2014-10-27
AU2009289776A1 (en) 2010-03-11
CN102159284A (zh) 2011-08-17
HRP20190500T1 (hr) 2019-08-09
PE20142371A1 (es) 2015-02-04
DK2735338T3 (en) 2019-04-23
CN105520924A (zh) 2016-04-27
IL211135A (en) 2017-09-28
WO2010025931A3 (en) 2010-06-17
IL237391A (en) 2017-12-31
CN105520924B (zh) 2019-04-09
AR073361A1 (es) 2010-11-03
HUE043278T2 (hu) 2019-08-28
EP2735338A1 (en) 2014-05-28
SI2735338T1 (sl) 2019-04-30
HK1159011A1 (en) 2012-07-27
HRP20140663T1 (hr) 2014-10-10
IL211135A0 (en) 2011-04-28
RU2674150C1 (ru) 2018-12-05
AR117613A2 (es) 2021-08-18
PL2331210T3 (pl) 2014-12-31
KR20170048602A (ko) 2017-05-08
KR101641519B1 (ko) 2016-07-21
RU2011112444A (ru) 2012-10-10
SI2331210T1 (sl) 2014-10-30
HK1198145A1 (en) 2015-03-13
MX2011002339A (es) 2011-04-04
AU2018202879A1 (en) 2018-05-17
PE20142357A1 (es) 2015-02-04
LT2735338T (lt) 2019-04-10
EP2331210A2 (en) 2011-06-15
IL237391A0 (en) 2015-04-30
ECSP11010869A (es) 2011-04-29
IL237392B (en) 2019-08-29
KR20160086981A (ko) 2016-07-20
CY1121492T1 (el) 2020-05-29
PE20142372A1 (es) 2015-02-04
KR101730924B1 (ko) 2017-04-27
KR20110057144A (ko) 2011-05-31
PE20190914A1 (es) 2019-06-26
JP5731387B2 (ja) 2015-06-10
WO2010025931A2 (en) 2010-03-11
CA2735857A1 (en) 2010-03-11
ZA201101449B (en) 2011-10-26
DK2331210T3 (da) 2014-08-11

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