CH619950A5 - Process for the preparation of condensed pyrimidines - Google Patents

Process for the preparation of condensed pyrimidines Download PDF

Info

Publication number
CH619950A5
CH619950A5 CH511074A CH511074A CH619950A5 CH 619950 A5 CH619950 A5 CH 619950A5 CH 511074 A CH511074 A CH 511074A CH 511074 A CH511074 A CH 511074A CH 619950 A5 CH619950 A5 CH 619950A5
Authority
CH
Switzerland
Prior art keywords
group
mixture
alkyl
quinoline
ethyl
Prior art date
Application number
CH511074A
Other languages
English (en)
French (fr)
Inventor
Thomas Henry Althuis
Leonard Joseph Czuba
Saul Bernard Kadin
Hans-Jurgen Ernst Hess
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CH619950A5 publication Critical patent/CH619950A5/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CH511074A 1973-04-13 1974-04-11 Process for the preparation of condensed pyrimidines CH619950A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US35102573A 1973-04-13 1973-04-13

Publications (1)

Publication Number Publication Date
CH619950A5 true CH619950A5 (en) 1980-10-31

Family

ID=23379271

Family Applications (1)

Application Number Title Priority Date Filing Date
CH511074A CH619950A5 (en) 1973-04-13 1974-04-11 Process for the preparation of condensed pyrimidines

Country Status (23)

Country Link
JP (1) JPS5018481A (no)
AR (3) AR205342A1 (no)
AT (1) AT342596B (no)
BE (1) BE813571A (no)
BG (1) BG25988A3 (no)
CA (1) CA1027945A (no)
CH (1) CH619950A5 (no)
DD (1) DD111207A5 (no)
DE (1) DE2418498A1 (no)
DK (1) DK142621B (no)
ES (1) ES425238A1 (no)
FI (1) FI55658C (no)
FR (1) FR2225166B1 (no)
GB (1) GB1458205A (no)
HU (1) HU171157B (no)
IE (1) IE41673B1 (no)
IL (1) IL44569A (no)
LU (1) LU69855A1 (no)
NL (1) NL170285C (no)
NO (1) NO139735C (no)
RO (1) RO64918A (no)
YU (1) YU36960B (no)
ZA (1) ZA742351B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4011324A (en) * 1976-01-20 1977-03-08 Pfizer Inc. Esters and amides of pyrimido[4,5-b]quinolin-4(3H)-one-2-carboxylic acids as antiulcer agents
DE2757915A1 (de) * 1976-12-28 1978-07-06 Mitsubishi Yuka Pharma Pyrimidochinoxalinderivate, verfahren zur herstellung derselben und arzneimittel zur behandlung von allergischem asthma
JPS59210071A (ja) * 1982-12-30 1984-11-28 バイオメジヤ−・インコ−ポレ−テツド 抗ウイルス作用を有する化合物
DE68908786T2 (de) * 1988-06-16 1994-03-17 Smith Kline French Lab Condensierte Pyrimidinderivate, Verfahren und Zwischenprodukte zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen.
FR2682378B1 (fr) * 1991-10-10 1995-04-07 Bellon Laboratoires Nouveaux derives de l'acide fluoroquinoleine carboxylique-3 et leur preparation.
FR2703681B1 (fr) * 1993-04-08 1995-05-12 Bellon Labor Sa Roger Procede de preparation de fluoro-6-halogeno-2 quinoleine
EP1556379A4 (en) * 2002-10-16 2007-06-13 Smithkline Beecham Corp CHEMICAL COMPOUNDS
EP4039753A4 (en) * 2019-09-30 2023-03-22 FUJIFILM Corporation COLORED RESIN PARTICLE DISPERSION, INK, INK SET, INKJET TEXTILE PRINTING METHOD, OIL-SOLUBLE DYE PRODUCTION METHOD, AND TEXTILE PRINTED ARTICLE

Also Published As

Publication number Publication date
AU6750074A (en) 1975-10-09
GB1458205A (en) 1976-12-08
YU36960B (en) 1984-08-31
DE2418498A1 (de) 1974-11-07
NL170285C (nl) 1982-10-18
YU101674A (en) 1982-06-18
HU171157B (hu) 1977-11-28
FI55658B (fi) 1979-05-31
FI55658C (fi) 1979-09-10
NO741231L (no) 1974-10-15
NO139735C (no) 1979-05-02
ES425238A1 (es) 1976-05-16
IE41673B1 (en) 1980-02-27
BE813571A (fr) 1974-10-11
DD111207A5 (no) 1975-02-05
NL7404894A (no) 1974-10-15
FR2225166A1 (no) 1974-11-08
IE41673L (en) 1974-10-13
AR205342A1 (es) 1976-04-30
NL170285B (nl) 1982-05-17
AT342596B (de) 1978-04-10
BG25988A3 (no) 1979-01-12
DK142621C (no) 1981-08-03
DK142621B (da) 1980-12-01
CA1027945A (en) 1978-03-14
LU69855A1 (no) 1974-11-21
FR2225166B1 (no) 1977-06-03
ZA742351B (en) 1975-04-30
NO139735B (no) 1979-01-22
AR205556A1 (es) 1976-05-14
ATA315174A (de) 1977-08-15
IL44569A0 (en) 1974-06-30
IL44569A (en) 1979-05-31
JPS5018481A (no) 1975-02-26
AR207459A1 (es) 1976-10-08
RO64918A (ro) 1980-01-15

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