DK142621B - Analogifremgangsmåde til fremstilling af pyrimido(4,5-b)quinolin-4(3H)-on-2-carboxylsyre-forbindelser eller farmaceutisk acceptable kationsalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af pyrimido(4,5-b)quinolin-4(3H)-on-2-carboxylsyre-forbindelser eller farmaceutisk acceptable kationsalte deraf. Download PDF

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Publication number
DK142621B
DK142621B DK200974AA DK200974A DK142621B DK 142621 B DK142621 B DK 142621B DK 200974A A DK200974A A DK 200974AA DK 200974 A DK200974 A DK 200974A DK 142621 B DK142621 B DK 142621B
Authority
DK
Denmark
Prior art keywords
quinoline
decomp
mixture
ethyl
filtered
Prior art date
Application number
DK200974AA
Other languages
Danish (da)
English (en)
Other versions
DK142621C (no
Inventor
Saul Bernard Kadin
Hans-Jurgen Ernst Hess
Thomas Henry Althuis
Leonard Joseph Czuba
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Priority to DK387377A priority Critical patent/DK387377A/da
Priority to DK387477A priority patent/DK387477A/da
Publication of DK142621B publication Critical patent/DK142621B/da
Application granted granted Critical
Publication of DK142621C publication Critical patent/DK142621C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK200974AA 1973-04-13 1974-04-10 Analogifremgangsmåde til fremstilling af pyrimido(4,5-b)quinolin-4(3H)-on-2-carboxylsyre-forbindelser eller farmaceutisk acceptable kationsalte deraf. DK142621B (da)

Priority Applications (2)

Application Number Priority Date Filing Date Title
DK387377A DK387377A (da) 1973-04-13 1977-08-31 Analogifremgangsmade til fremstilling af 2-alkylpyrimido-(4,5-b)quinolin-4(3h)-onforbindelser
DK387477A DK387477A (da) 1973-04-13 1977-08-31 Analogifremgangsmade til fremstilling af 2-hydroxyethyl-7,8-dimethoxypyrimido(4,5b)-quinolin-4(3h)-on-2-carboxylat

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35102573A 1973-04-13 1973-04-13
US35102573 1973-04-13

Publications (2)

Publication Number Publication Date
DK142621B true DK142621B (da) 1980-12-01
DK142621C DK142621C (no) 1981-08-03

Family

ID=23379271

Family Applications (1)

Application Number Title Priority Date Filing Date
DK200974AA DK142621B (da) 1973-04-13 1974-04-10 Analogifremgangsmåde til fremstilling af pyrimido(4,5-b)quinolin-4(3H)-on-2-carboxylsyre-forbindelser eller farmaceutisk acceptable kationsalte deraf.

Country Status (23)

Country Link
JP (1) JPS5018481A (no)
AR (3) AR205342A1 (no)
AT (1) AT342596B (no)
BE (1) BE813571A (no)
BG (1) BG25988A3 (no)
CA (1) CA1027945A (no)
CH (1) CH619950A5 (no)
DD (1) DD111207A5 (no)
DE (1) DE2418498A1 (no)
DK (1) DK142621B (no)
ES (1) ES425238A1 (no)
FI (1) FI55658C (no)
FR (1) FR2225166B1 (no)
GB (1) GB1458205A (no)
HU (1) HU171157B (no)
IE (1) IE41673B1 (no)
IL (1) IL44569A (no)
LU (1) LU69855A1 (no)
NL (1) NL170285C (no)
NO (1) NO139735C (no)
RO (1) RO64918A (no)
YU (1) YU36960B (no)
ZA (1) ZA742351B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4011324A (en) * 1976-01-20 1977-03-08 Pfizer Inc. Esters and amides of pyrimido[4,5-b]quinolin-4(3H)-one-2-carboxylic acids as antiulcer agents
DE2757915A1 (de) * 1976-12-28 1978-07-06 Mitsubishi Yuka Pharma Pyrimidochinoxalinderivate, verfahren zur herstellung derselben und arzneimittel zur behandlung von allergischem asthma
JPS59210071A (ja) * 1982-12-30 1984-11-28 バイオメジヤ−・インコ−ポレ−テツド 抗ウイルス作用を有する化合物
DE68908786T2 (de) * 1988-06-16 1994-03-17 Smith Kline French Lab Condensierte Pyrimidinderivate, Verfahren und Zwischenprodukte zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen.
FR2682378B1 (fr) * 1991-10-10 1995-04-07 Bellon Laboratoires Nouveaux derives de l'acide fluoroquinoleine carboxylique-3 et leur preparation.
FR2703681B1 (fr) * 1993-04-08 1995-05-12 Bellon Labor Sa Roger Procede de preparation de fluoro-6-halogeno-2 quinoleine
EP1556379A4 (en) * 2002-10-16 2007-06-13 Smithkline Beecham Corp CHEMICAL COMPOUNDS
EP4039753A4 (en) * 2019-09-30 2023-03-22 FUJIFILM Corporation COLORED RESIN PARTICLE DISPERSION, INK, INK SET, INKJET TEXTILE PRINTING METHOD, OIL-SOLUBLE DYE PRODUCTION METHOD, AND TEXTILE PRINTED ARTICLE

Also Published As

Publication number Publication date
AU6750074A (en) 1975-10-09
GB1458205A (en) 1976-12-08
CH619950A5 (en) 1980-10-31
YU36960B (en) 1984-08-31
DE2418498A1 (de) 1974-11-07
NL170285C (nl) 1982-10-18
YU101674A (en) 1982-06-18
HU171157B (hu) 1977-11-28
FI55658B (fi) 1979-05-31
FI55658C (fi) 1979-09-10
NO741231L (no) 1974-10-15
NO139735C (no) 1979-05-02
ES425238A1 (es) 1976-05-16
IE41673B1 (en) 1980-02-27
BE813571A (fr) 1974-10-11
DD111207A5 (no) 1975-02-05
NL7404894A (no) 1974-10-15
FR2225166A1 (no) 1974-11-08
IE41673L (en) 1974-10-13
AR205342A1 (es) 1976-04-30
NL170285B (nl) 1982-05-17
AT342596B (de) 1978-04-10
BG25988A3 (no) 1979-01-12
DK142621C (no) 1981-08-03
CA1027945A (en) 1978-03-14
LU69855A1 (no) 1974-11-21
FR2225166B1 (no) 1977-06-03
ZA742351B (en) 1975-04-30
NO139735B (no) 1979-01-22
AR205556A1 (es) 1976-05-14
ATA315174A (de) 1977-08-15
IL44569A0 (en) 1974-06-30
IL44569A (en) 1979-05-31
JPS5018481A (no) 1975-02-26
AR207459A1 (es) 1976-10-08
RO64918A (ro) 1980-01-15

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