CA3223555A1 - Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton - Google Patents

Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton

Info

Publication number
CA3223555A1
CA3223555A1 CA3223555A CA3223555A CA3223555A1 CA 3223555 A1 CA3223555 A1 CA 3223555A1 CA 3223555 A CA3223555 A CA 3223555A CA 3223555 A CA3223555 A CA 3223555A CA 3223555 A1 CA3223555 A1 CA 3223555A1
Authority
CA
Canada
Prior art keywords
zolmitriptan
microns
microprojections
patch
coating
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3223555A
Other languages
English (en)
Inventor
Mahmoud Ameri
Donald Kellerman
Yi Ao
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Emergex USA Corp
Original Assignee
Emergex USA Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Emergex USA Corp filed Critical Emergex USA Corp
Priority to CA3223555A priority Critical patent/CA3223555A1/fr
Publication of CA3223555A1 publication Critical patent/CA3223555A1/fr
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0021Intradermal administration, e.g. through microneedle arrays, needleless injectors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M37/00Other apparatus for introducing media into the body; Percutany, i.e. introducing medicines into the body by diffusion through the skin
    • A61M37/0015Other apparatus for introducing media into the body; Percutany, i.e. introducing medicines into the body by diffusion through the skin by using microneedles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61MDEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
    • A61M37/00Other apparatus for introducing media into the body; Percutany, i.e. introducing medicines into the body by diffusion through the skin
    • A61M37/0015Other apparatus for introducing media into the body; Percutany, i.e. introducing medicines into the body by diffusion through the skin by using microneedles
    • A61M2037/0023Drug applicators using microneedles

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Dermatology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Anesthesiology (AREA)
  • Medical Informatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Media Introduction/Drainage Providing Device (AREA)
CA3223555A 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton Pending CA3223555A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CA3223555A CA3223555A1 (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
PCT/US2017/048258 WO2019040063A1 (fr) 2017-08-23 2017-08-23 Procédé d'obtention rapide de concentrations thérapeutiques de zolmitriptan pour le traitement de migraines et de céphalées de horton
CA3223555A CA3223555A1 (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton
CA3073442A CA3073442C (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA3073442A Division CA3073442C (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton

Publications (1)

Publication Number Publication Date
CA3223555A1 true CA3223555A1 (fr) 2019-02-28

Family

ID=59829462

Family Applications (2)

Application Number Title Priority Date Filing Date
CA3073442A Active CA3073442C (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton
CA3223555A Pending CA3223555A1 (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CA3073442A Active CA3073442C (fr) 2017-08-23 2017-08-23 Procede d'obtention rapide de concentrations therapeutiques de zolmitriptan pour le traitement de migraines et de cephalees de horton

Country Status (8)

Country Link
EP (1) EP3672570A1 (fr)
JP (2) JP7219384B2 (fr)
KR (2) KR102340393B1 (fr)
CN (1) CN111050749A (fr)
AU (1) AU2017428907B2 (fr)
CA (2) CA3073442C (fr)
IL (1) IL272776B1 (fr)
WO (1) WO2019040063A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3416618A1 (fr) 2016-02-19 2018-12-26 ZP Opco, Inc. Procédé pour obtenir rapidement des concentrations thérapeutiques de triptans pour le traitement de migraines
US11660264B2 (en) 2017-08-23 2023-05-30 Emergex USA Corporation Method of rapidly achieving therapeutic concentrations of triptans for treatment of migraines and cluster headaches
US11660265B2 (en) 2018-06-28 2023-05-30 Emergex USA Corporation Method of rapidly achieving therapeutic concentrations of triptans for treatment of migraines and cluster headaches
US20220241571A1 (en) * 2019-06-06 2022-08-04 Kindeva Drug Delivery L.P. Microarray carrier for microarray applicator
CA3145203A1 (fr) * 2019-06-28 2020-12-30 Passport Technologies, Inc. Systeme de distribution de micro-porosites de triptan
CN114699510A (zh) * 2021-12-29 2022-07-05 浙江湃肽生物有限公司 一种司美格鲁肽微针阵列及其制备方法
CN115887903A (zh) * 2022-12-15 2023-04-04 太平洋康泰科学仪器(济南)有限公司 微针贴片给药组件及给药方法

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5080646A (en) 1988-10-03 1992-01-14 Alza Corporation Membrane for electrotransport transdermal drug delivery
US5169382A (en) 1988-10-03 1992-12-08 Alza Corporation Membrane for electrotransport transdermal drug delivery
US5147296A (en) 1988-10-03 1992-09-15 Alza Corporation Membrane for electrotransport transdermal drug delivery
ES2195151T3 (es) 1996-06-18 2003-12-01 Alza Corp Dispositivo de mejora de aporte o de muestreo de agentes transdermicos.
US5916524A (en) 1997-07-23 1999-06-29 Bio-Dot, Inc. Dispensing apparatus having improved dynamic range
US5743960A (en) 1996-07-26 1998-04-28 Bio-Dot, Inc. Precision metered solenoid valve dispenser
US5738728A (en) 1996-07-26 1998-04-14 Bio Dot, Inc. Precision metered aerosol dispensing apparatus
US5741554A (en) 1996-07-26 1998-04-21 Bio Dot, Inc. Method of dispensing a liquid reagent
EP1037687B8 (fr) 1997-12-11 2008-10-22 Alza Corporation Dispositif renfor ant le flux d'agents transdermiques
ATE221400T1 (de) 1997-12-11 2002-08-15 Alza Corp Vorrichtung zur erhöhung des transdermalen wirkstoffeflusses
DK1037686T3 (da) 1997-12-11 2006-01-02 Alza Corp Apparat til forögelse af transdermal gennemströmning af midler
US6091975A (en) 1998-04-01 2000-07-18 Alza Corporation Minimally invasive detecting device
ES2253278T3 (es) 1999-12-10 2006-06-01 Alza Corporation Dispositivo y procedimiento para mejorar la perforacion cutanea con microprotuberancias.
IL155389A0 (en) 2000-10-13 2003-11-23 Alza Corportion Microprotrusion member retainer for impact applicator
EP1341453B1 (fr) 2000-10-13 2009-04-15 Alza Corporation Dispositif et procede permettant la perforation de la peau au moyen de microprotuberances
WO2002030281A1 (fr) 2000-10-13 2002-04-18 Alza Corporation Applicateur a reseau de microlames produisant un impact
US7419481B2 (en) 2000-10-13 2008-09-02 Alza Corporation Apparatus and method for piercing skin with microprotrusions
IL155583A0 (en) 2000-10-26 2003-11-23 Alza Corp Transdermal drug delivery devices having coated microprotrusions
US6855372B2 (en) 2001-03-16 2005-02-15 Alza Corporation Method and apparatus for coating skin piercing microprojections
BR0209046A (pt) 2001-04-20 2004-11-09 Alza Corp Disposição de microprojeção que possui um agente benéfico contendo revestimento
EP1680154B1 (fr) 2003-10-31 2012-01-04 ALZA Corporation Applicateur a actionnement automatique pour reseau de micro-protuberances
CA2566032A1 (fr) 2004-05-13 2005-12-01 Alza Corporation Appareil et procede pour la delivrance transdermique d'agents a base d'hormone parathyroide
CN101466393A (zh) 2006-03-15 2009-06-24 阿尔扎公司 用于经皮递送甲状旁腺激素药剂以治疗骨质减少的方法
WO2008115586A1 (fr) 2007-03-21 2008-09-25 Alza Corporation Appareil et procédé d'administration transdermique d'un agoniste de triptane
JP6121734B2 (ja) * 2012-02-09 2017-04-26 久光製薬株式会社 マイクロニードル用ゾルミトリプタン含有コーティング組成物及びマイクロニードルデバイス
WO2015017561A1 (fr) 2013-07-30 2015-02-05 Zosano Pharma, Inc. Applicateur extra-plat de tampon de micro-aiguilles
EP3416618A1 (fr) * 2016-02-19 2018-12-26 ZP Opco, Inc. Procédé pour obtenir rapidement des concentrations thérapeutiques de triptans pour le traitement de migraines

Also Published As

Publication number Publication date
CA3073442C (fr) 2024-02-06
EP3672570A1 (fr) 2020-07-01
KR102340393B1 (ko) 2021-12-17
KR20200032170A (ko) 2020-03-25
JP2021500397A (ja) 2021-01-07
IL272776A (en) 2020-04-30
KR20210155817A (ko) 2021-12-23
CA3073442A1 (fr) 2019-02-28
IL272776B1 (en) 2024-02-01
JP2023033378A (ja) 2023-03-10
CN111050749A (zh) 2020-04-21
AU2017428907B2 (en) 2021-12-16
JP7219384B2 (ja) 2023-02-08
AU2017428907A1 (en) 2020-03-05
WO2019040063A1 (fr) 2019-02-28

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20231218

EEER Examination request

Effective date: 20231218

EEER Examination request

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EEER Examination request

Effective date: 20231218