CA3140641A1 - Formulations d'imatinib, leur fabrication et leurs utilisations - Google Patents
Formulations d'imatinib, leur fabrication et leurs utilisations Download PDFInfo
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- CA3140641A1 CA3140641A1 CA3140641A CA3140641A CA3140641A1 CA 3140641 A1 CA3140641 A1 CA 3140641A1 CA 3140641 A CA3140641 A CA 3140641A CA 3140641 A CA3140641 A CA 3140641A CA 3140641 A1 CA3140641 A1 CA 3140641A1
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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Abstract
L'invention concerne des formulations d'imatinib inhalables, leur fabrication et leurs utilisations. Les compositions et les méthodes de l'invention permettent de résoudre les problèmes posés par les traitements de la HTAP à base d'imatinib grâce à l'utilisation de formulations et de mécanismes d'administration spécialisés. Plus particulièrement, l'invention reconnaît que la forme cristalline et la composition polymorphe de médicaments tels que l'imatinib et ses sels peuvent exercer des effets significatifs sur la solubilité, l'administration, l'absorption et le métabolisme des médicaments.
Applications Claiming Priority (17)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962849056P | 2019-05-16 | 2019-05-16 | |
| US201962849058P | 2019-05-16 | 2019-05-16 | |
| US201962849059P | 2019-05-16 | 2019-05-16 | |
| US201962849054P | 2019-05-16 | 2019-05-16 | |
| US62/849,058 | 2019-05-16 | ||
| US62/849,059 | 2019-05-16 | ||
| US62/849,056 | 2019-05-16 | ||
| US62/849,054 | 2019-05-16 | ||
| US201962877575P | 2019-07-23 | 2019-07-23 | |
| US62/877,575 | 2019-07-23 | ||
| US201962942408P | 2019-12-02 | 2019-12-02 | |
| US62/942,408 | 2019-12-02 | ||
| US202062958481P | 2020-01-08 | 2020-01-08 | |
| US62/958,481 | 2020-01-08 | ||
| US202062984037P | 2020-03-02 | 2020-03-02 | |
| US62/984,037 | 2020-03-02 | ||
| PCT/US2020/032872 WO2020232236A1 (fr) | 2019-05-16 | 2020-05-14 | Formulations d'imatinib, leur fabrication et leurs utilisations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3140641A1 true CA3140641A1 (fr) | 2020-11-19 |
Family
ID=73228465
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3140641A Pending CA3140641A1 (fr) | 2019-05-16 | 2020-05-14 | Formulations d'imatinib, leur fabrication et leurs utilisations |
Country Status (14)
| Country | Link |
|---|---|
| US (13) | US20200360279A1 (fr) |
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| JP2023550407A (ja) * | 2020-11-17 | 2023-12-01 | ユナイテッド セラピューティクス コーポレイション | 肺高血圧向けの吸入式イマチニブ |
| WO2022109458A1 (fr) * | 2020-11-23 | 2022-05-27 | Aerovate Therapeutics, Inc. | Formulations d'imatinib, fabrication et utilisations de celles-ci |
| EP4274577A1 (fr) * | 2021-01-06 | 2023-11-15 | InCarda Therapeutics, Inc. | Formulation d'imatinib inhalable |
| KR102634754B1 (ko) * | 2021-07-07 | 2024-02-08 | 애니머스큐어 주식회사 | 이마티닙을 포함하는 근육 질환의 예방 또는 치료용 조성물 |
| WO2023147868A1 (fr) * | 2022-02-04 | 2023-08-10 | Justus-Liebig-Universität Giessen | Imatinib inhalé pour le traitement de l'hypertension pulmonaire |
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- 2020-05-14 WO PCT/US2020/032874 patent/WO2020232238A1/fr active Application Filing
- 2020-05-14 BR BR112021023014A patent/BR112021023014A2/pt unknown
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- 2020-05-14 EP EP20806383.4A patent/EP3968963A4/fr active Pending
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