CA3018986A1 - Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith - Google Patents
Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith Download PDFInfo
- Publication number
- CA3018986A1 CA3018986A1 CA3018986A CA3018986A CA3018986A1 CA 3018986 A1 CA3018986 A1 CA 3018986A1 CA 3018986 A CA3018986 A CA 3018986A CA 3018986 A CA3018986 A CA 3018986A CA 3018986 A1 CA3018986 A1 CA 3018986A1
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- Canada
- Prior art keywords
- cancer
- purin
- cyclohexanecarboxamide
- substituted
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US201662317412P | 2016-04-01 | 2016-04-01 | |
| US62/317,412 | 2016-04-01 | ||
| PCT/US2017/025252 WO2017173206A1 (en) | 2016-04-01 | 2017-03-31 | Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith |
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|---|---|
| CA3018986A1 true CA3018986A1 (en) | 2017-10-05 |
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| CA3018986A Abandoned CA3018986A1 (en) | 2016-04-01 | 2017-03-31 | Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith |
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| BR (1) | BR112018070163A2 (cg-RX-API-DMAC7.html) |
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| JO3633B1 (ar) | 2015-09-16 | 2020-08-27 | Katholieke Univ Leuven Ku Leuven Research & Development | مشتقات اندول مستبدلة احاديا او ثنائيا بصفتها مانعات للتكاثر الفيروسي لحمى الفنك |
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| MX2018011992A (es) | 2019-01-24 |
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| US20170281633A1 (en) | 2017-10-05 |
| SG10202009589UA (en) | 2020-10-29 |
| EA201892229A1 (ru) | 2019-03-29 |
| EA039392B1 (ru) | 2022-01-21 |
| WO2017173206A1 (en) | 2017-10-05 |
| IL262007B2 (en) | 2023-04-01 |
| KR20180126497A (ko) | 2018-11-27 |
| BR112018070163A2 (pt) | 2019-01-29 |
| US10576085B2 (en) | 2020-03-03 |
| JP2019510066A (ja) | 2019-04-11 |
| EP3436018A4 (en) | 2019-11-13 |
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