CA2920457A1 - Anti-acne compositions comprising bile acid-fatty acid conjugates - Google Patents
Anti-acne compositions comprising bile acid-fatty acid conjugates Download PDFInfo
- Publication number
- CA2920457A1 CA2920457A1 CA2920457A CA2920457A CA2920457A1 CA 2920457 A1 CA2920457 A1 CA 2920457A1 CA 2920457 A CA2920457 A CA 2920457A CA 2920457 A CA2920457 A CA 2920457A CA 2920457 A1 CA2920457 A1 CA 2920457A1
- Authority
- CA
- Canada
- Prior art keywords
- acid
- composition
- acne
- fabac
- fatty acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361863454P | 2013-08-08 | 2013-08-08 | |
| US61/863,454 | 2013-08-08 | ||
| PCT/IL2014/050718 WO2015019359A1 (en) | 2013-08-08 | 2014-08-07 | Anti-acne compositions comprising bile acid-fatty acid conjugates |
Publications (1)
| Publication Number | Publication Date |
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| CA2920457A1 true CA2920457A1 (en) | 2015-02-12 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2920457A Abandoned CA2920457A1 (en) | 2013-08-08 | 2014-08-07 | Anti-acne compositions comprising bile acid-fatty acid conjugates |
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| Country | Link |
|---|---|
| US (1) | US20160175324A1 (enExample) |
| EP (1) | EP3030229B1 (enExample) |
| JP (1) | JP2016527307A (enExample) |
| CN (1) | CN105611919A (enExample) |
| AU (1) | AU2014304079A1 (enExample) |
| CA (1) | CA2920457A1 (enExample) |
| WO (1) | WO2015019359A1 (enExample) |
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|---|---|---|---|---|
| IL227890A0 (en) * | 2013-08-08 | 2014-01-30 | Galderm Therapeutics Ltd | Antiaging compounds containing bile acid and fatty acid conjugates |
| WO2016199137A1 (en) | 2015-06-10 | 2016-12-15 | Galmed Research And Development Ltd. | Low dose compositions of aramchol salts |
| US11571431B2 (en) | 2013-12-04 | 2023-02-07 | Galmed Research And Development Ltd | Aramchol salts |
| US10016456B2 (en) * | 2014-07-18 | 2018-07-10 | Dabney Patents, L.L.C. | Methods for treating acne vulgaris |
| IL243707A0 (en) | 2016-01-20 | 2016-05-01 | Galmed Res And Dev Ltd | Treatment to regulate the microbiota in the intestine |
| KR20180036580A (ko) | 2016-09-30 | 2018-04-09 | 주식회사 유스바이오팜 | 수가용화(水加溶化)된 우르소데옥시콜산을 함유하는 염증성 피부질환 또는 중증 소양증 예방 또는 치료용 조성물 |
| WO2018062922A1 (ko) * | 2016-09-30 | 2018-04-05 | 주식회사 유스바이오팜 | 수가용화된 우르소데옥시콜산을 함유하는 염증성 피부질환 또는 중증 소양증 예방 또는 치료용 조성물 |
| US11197870B2 (en) | 2016-11-10 | 2021-12-14 | Galmed Research And Development Ltd | Treatment for hepatic fibrosis |
| WO2019044852A1 (ja) * | 2017-08-31 | 2019-03-07 | 株式会社資生堂 | レチノイドの副作用に対する感受性の決定方法 |
| CN109503693B (zh) * | 2018-12-12 | 2021-04-06 | 合肥工业大学 | 一种利用胆酸为原料合成Aramchol的工艺 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3860712A (en) * | 1973-04-16 | 1975-01-14 | Sterling Drug Inc | Composition and method for treatment of acne or seborrhea |
| IT8167097A0 (it) * | 1981-01-26 | 1981-01-26 | Unilever Nv | Composizione cosmetica per il trattamento della pelle o dei capelli |
| IL123998A (en) * | 1998-04-08 | 2004-09-27 | Galmed Int Ltd | Conjugates of bile salts and pharmaceutical preparations containing them |
| US7759348B2 (en) * | 2003-07-30 | 2010-07-20 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives and their use as therapeutic agents |
| ES2296463B1 (es) * | 2005-07-13 | 2009-02-16 | Universidade De Santiago Compostela | Nuevos amidoderivados de acidos billares funcionalizados en la posicion 3 del anillo a. procedimientos para su obtencion y aplicaciones. |
| ES2352098T3 (es) * | 2007-08-08 | 2011-02-15 | Graceway Pharmaceuticals, Llc | Derivado de fenoxi-pirrolidina y su uso y composiciones. |
| WO2009060452A2 (en) * | 2007-11-08 | 2009-05-14 | Galmed International Ltd. | Methods and compositions for treating biliary cholesterol crystallization and related conditions |
| FR2940281B1 (fr) * | 2008-12-22 | 2011-04-01 | Fabre Pierre Dermo Cosmetique | Ester de diol et d'acide gras polyinsature comme agent anti-acne |
| US8937194B2 (en) * | 2008-12-31 | 2015-01-20 | Nitromega Corp. | Topical compositions containing nitro fatty acids |
| WO2010086864A1 (en) * | 2009-02-02 | 2010-08-05 | Galmed International Ltd. | Methods and compositions for treating alzheimer's disease |
| IL227890A0 (en) * | 2013-08-08 | 2014-01-30 | Galderm Therapeutics Ltd | Antiaging compounds containing bile acid and fatty acid conjugates |
-
2014
- 2014-08-07 CA CA2920457A patent/CA2920457A1/en not_active Abandoned
- 2014-08-07 US US14/910,485 patent/US20160175324A1/en not_active Abandoned
- 2014-08-07 EP EP14834482.3A patent/EP3030229B1/en active Active
- 2014-08-07 JP JP2016532792A patent/JP2016527307A/ja active Pending
- 2014-08-07 WO PCT/IL2014/050718 patent/WO2015019359A1/en not_active Ceased
- 2014-08-07 AU AU2014304079A patent/AU2014304079A1/en not_active Abandoned
- 2014-08-07 CN CN201480055619.0A patent/CN105611919A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| CN105611919A (zh) | 2016-05-25 |
| EP3030229A1 (en) | 2016-06-15 |
| AU2014304079A1 (en) | 2016-02-25 |
| US20160175324A1 (en) | 2016-06-23 |
| WO2015019359A1 (en) | 2015-02-12 |
| EP3030229B1 (en) | 2019-03-13 |
| JP2016527307A (ja) | 2016-09-08 |
| EP3030229A4 (en) | 2017-03-22 |
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