CA2666177A1 - Acylaminoimidazoles and acylaminothiazoles - Google Patents

Acylaminoimidazoles and acylaminothiazoles Download PDF

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Publication number
CA2666177A1
CA2666177A1 CA002666177A CA2666177A CA2666177A1 CA 2666177 A1 CA2666177 A1 CA 2666177A1 CA 002666177 A CA002666177 A CA 002666177A CA 2666177 A CA2666177 A CA 2666177A CA 2666177 A1 CA2666177 A1 CA 2666177A1
Authority
CA
Canada
Prior art keywords
alkyl
substituents
another
substituted
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002666177A
Other languages
English (en)
French (fr)
Inventor
Marcus Bauser
Anja Buchmueller
Georges Von Degenfeld
Elke Dittrich-Wengenroth
Christoph Gerdes
Mark Jean Gnoth
Dirk Gottschling
Stefan Heitmeier
Martin Hendrix
Johannes Koebberling
Dieter Lang
Ulrich Rester
Uwe Saatmann
Adrian Tersteegen
Astrid Bruens
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
Original Assignee
Bayer Schering Pharma Aktiengesellschaft
Marcus Bauser
Anja Buchmueller
Georges Von Degenfeld
Elke Dittrich-Wengenroth
Christoph Gerdes
Mark Jean Gnoth
Dirk Gottschling
Stefan Heitmeier
Martin Hendrix
Johannes Koebberling
Dieter Lang
Ulrich Rester
Uwe Saatmann
Adrian Tersteegen
Astrid Bruens
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Aktiengesellschaft, Marcus Bauser, Anja Buchmueller, Georges Von Degenfeld, Elke Dittrich-Wengenroth, Christoph Gerdes, Mark Jean Gnoth, Dirk Gottschling, Stefan Heitmeier, Martin Hendrix, Johannes Koebberling, Dieter Lang, Ulrich Rester, Uwe Saatmann, Adrian Tersteegen, Astrid Bruens filed Critical Bayer Schering Pharma Aktiengesellschaft
Publication of CA2666177A1 publication Critical patent/CA2666177A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88Nitrogen atoms, e.g. allantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
CA002666177A 2006-10-11 2007-10-10 Acylaminoimidazoles and acylaminothiazoles Abandoned CA2666177A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102006048042.2 2006-10-11
DE102006048042A DE102006048042A1 (de) 2006-10-11 2006-10-11 Acylaminoimidazole und Acylaminothiazole
PCT/EP2007/008789 WO2008043533A2 (de) 2006-10-11 2007-10-10 Acylaminoimidazole und acylaminothiazole

Publications (1)

Publication Number Publication Date
CA2666177A1 true CA2666177A1 (en) 2008-04-17

Family

ID=39184814

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002666177A Abandoned CA2666177A1 (en) 2006-10-11 2007-10-10 Acylaminoimidazoles and acylaminothiazoles

Country Status (5)

Country Link
EP (1) EP2079708A2 (de)
JP (1) JP2010505896A (de)
CA (1) CA2666177A1 (de)
DE (1) DE102006048042A1 (de)
WO (1) WO2008043533A2 (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2350002A1 (de) * 2008-10-02 2011-08-03 Abbott Laboratories Neue verbindungen als kalziumkanalblocker
WO2011115813A1 (en) 2010-03-18 2011-09-22 Abbott Laboratories Lactam acetamides as calcium channel blockers
JP2015083542A (ja) * 2012-02-08 2015-04-30 大日本住友製薬株式会社 3位置換プロリン誘導体
IN2014MU00072A (de) * 2014-01-08 2015-08-21 Wockhardt Ltd
IL277071B1 (en) 2018-03-08 2024-03-01 Incyte Corp Aminopyrizine diol compounds as PI3K–y inhibitors
US11046658B2 (en) 2018-07-02 2021-06-29 Incyte Corporation Aminopyrazine derivatives as PI3K-γ inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2842523A1 (fr) * 2002-07-17 2004-01-23 Sanofi Synthelabo Derives d'acylaminothiazole, leur preparation et leur application en therapeutique
RS50595B (sr) * 2004-03-23 2010-05-07 Pfizer Products Incorporated Jedinjenja imidazola za lečenje neurodegenerativnih poremećaja
DE102006001574A1 (de) * 2006-01-12 2007-07-19 Bayer Healthcare Ag Acylaminoimidazole

Also Published As

Publication number Publication date
WO2008043533A2 (de) 2008-04-17
DE102006048042A1 (de) 2008-04-17
WO2008043533A3 (de) 2008-07-03
EP2079708A2 (de) 2009-07-22
JP2010505896A (ja) 2010-02-25

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Legal Events

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