CA2506236C - Compositions and uses of dalbavancin for treatment of bacterial infections - Google Patents
Compositions and uses of dalbavancin for treatment of bacterial infections Download PDFInfo
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- CA2506236C CA2506236C CA2506236A CA2506236A CA2506236C CA 2506236 C CA2506236 C CA 2506236C CA 2506236 A CA2506236 A CA 2506236A CA 2506236 A CA2506236 A CA 2506236A CA 2506236 C CA2506236 C CA 2506236C
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- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/14—Peptides containing saccharide radicals; Derivatives thereof, e.g. bleomycin, phleomycin, muramylpeptides or vancomycin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
- A61K31/704—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
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- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Immunology (AREA)
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- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| US49648303P | 2003-08-19 | 2003-08-19 | |
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| PCT/US2003/036127 WO2004045636A1 (en) | 2002-11-18 | 2003-11-14 | Methods of administering dalbavancin for treatment of bacterial infections |
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| US7119061B2 (en) * | 2002-11-18 | 2006-10-10 | Vicuron Pharmaceuticals, Inc. | Dalbavancin compositions for treatment of bacterial infections |
| US20060074014A1 (en) * | 2002-11-18 | 2006-04-06 | Vicuron Pharmaceuticals Inc. | Dalbavancin compositions for treatment of bacterial infections |
| US20090062182A1 (en) * | 2007-08-29 | 2009-03-05 | Protia, Llc | Deuterium-enriched dalbavancin |
| US8389583B2 (en) * | 2008-05-23 | 2013-03-05 | Zurex Pharma, Inc. | Antimicrobial compositions and methods of use |
| US20110132607A1 (en) * | 2009-12-07 | 2011-06-09 | Schlumberger Technology Corporation | Apparatus and Technique to Communicate With a Tubing-Conveyed Perforating Gun |
| KR102237887B1 (ko) | 2013-03-15 | 2021-04-07 | 멜린타 서브시디어리 코프. | 항생제를 사용하여 과체중 및 비만 환자에서 감염을 치료하는 방법 |
| JP6540705B2 (ja) | 2013-12-19 | 2019-07-10 | ジーイー・ヘルスケア・バイオサイエンス・アクチボラグ | 生物学的液体処理システムのための遠隔操作弁 |
| EP3169345B1 (en) | 2014-07-17 | 2025-01-29 | Melinta Therapeutics, LLC | High purity oritavancin and method of producing same |
| HRP20200101T1 (hr) | 2014-11-06 | 2020-04-03 | Xellia Pharmaceuticals Aps | Glikopeptidni pripravci |
| WO2016140981A1 (en) * | 2015-03-02 | 2016-09-09 | Colonaryconcepts Llc | Compounds and methods for peg metabolite and peg breakdown product assays |
| US10071141B2 (en) | 2015-05-08 | 2018-09-11 | Spectral Platforms, Inc. | Albumin-based non-covalent complexes and methods of use thereof |
| US20200171124A1 (en) | 2016-04-15 | 2020-06-04 | Lupin Limited | Topical compositions for ophthalmic and otic use |
| MX2019011119A (es) | 2017-03-20 | 2019-12-19 | Spectral Platforms Inc | Metodos espectroscopicos para detectar y caracterizar microorganismos. |
| CA3069679A1 (en) * | 2017-07-10 | 2019-01-17 | Contrafect Corporation | Blood component potentiation of lytic protein anti-bacterial activity and methods and uses thereof |
| CN110183519B (zh) * | 2019-05-06 | 2023-04-11 | 大邦(湖南)生物制药有限公司 | 一种达巴万星关键中间体a40926的分离纯化方法 |
| CN112480214B (zh) * | 2020-12-14 | 2023-03-28 | 成都雅途生物技术有限公司 | 一种达巴万星关键中间体a40926的制备方法 |
| EP4014965A1 (en) | 2020-12-16 | 2022-06-22 | EVER Valinject GmbH | Aqueous solution |
| WO2022148868A1 (en) | 2021-01-11 | 2022-07-14 | Xellia Pharmaceuticals Aps | Synthesis process |
| CN115215926A (zh) * | 2022-08-12 | 2022-10-21 | 丽珠集团福州福兴医药有限公司 | 达巴万星母核及其纯化方法、达巴万星及其合成方法 |
| AU2023359653A1 (en) * | 2022-10-12 | 2025-05-29 | Hikma Pharmaceuticals Usa Inc. | Liquid dalbavancin composition |
| JP2025533237A (ja) * | 2022-10-12 | 2025-10-03 | ヒクマ ファーマシューティカルズ ユーエスエイ インコーポレイテッド | 液体ダルババンシン組成物 |
| EP4431083A1 (en) | 2023-03-16 | 2024-09-18 | Adalvo Limited | Formulation of dalbavancin |
| EP4431084A1 (en) | 2023-03-16 | 2024-09-18 | Adalvo Limited | Formulation of dalbavancin |
| WO2025158262A1 (en) | 2024-01-23 | 2025-07-31 | Lupin Limited | Stable pharmaceutical compositions of dalbavancin as ready-to-dilute formulation |
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| FI73697C (fi) * | 1982-06-08 | 1987-11-09 | Lepetit Spa | Foerfarande foer framstaellning av individuella faktorer 1, 2, 3, 4 och 5 av teikomysin a2. |
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| GB8425685D0 (en) | 1984-10-11 | 1984-11-14 | Lepetit Spa | Antibiotic a 40926 complex |
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| US5004605A (en) * | 1987-12-10 | 1991-04-02 | Cetus Corporation | Low pH pharmaceutical compositions of recombinant β-interferon |
| FR2628269B1 (fr) * | 1988-03-04 | 1990-07-27 | Sgs Thomson Microelectronics | Dispositif de demarrage progressif d'une alimentation a decoupage |
| EP0376041B1 (en) | 1988-12-27 | 1996-02-28 | GRUPPO LEPETIT S.p.A. | C63-Amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy-teicoplanins |
| IE64155B1 (en) | 1989-03-29 | 1995-07-12 | Lepetit Spa | New substituted alkylamide derivatives of teicoplanin |
| JPH03193735A (ja) | 1989-12-22 | 1991-08-23 | Shionogi & Co Ltd | グリコペプチド系抗生物質の安定化組成物 |
| US5030619A (en) * | 1990-04-16 | 1991-07-09 | Miles Inc. | Synergistic fungicidal composition |
| US5606036A (en) | 1991-03-27 | 1997-02-25 | Gruppo Lepetit Spa | Antibiotic A 40926 ester derivatives |
| JP2783722B2 (ja) * | 1991-07-12 | 1998-08-06 | 麒麟麦酒株式会社 | スピカマイシン誘導体およびそれを含む抗腫瘍剤 |
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| EP0596929B1 (en) | 1991-07-29 | 1995-07-26 | GRUPPO LEPETIT S.p.A. | Amide derivatives of antibiotic a 40926 |
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- 2003-11-14 PT PT03789744T patent/PT1565201T/pt unknown
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- 2003-11-14 JP JP2004570384A patent/JP5519090B2/ja not_active Expired - Lifetime
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- 2003-11-14 WO PCT/US2003/036127 patent/WO2004045636A1/en not_active Ceased
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- 2003-11-14 US US10/493,558 patent/US20050090433A1/en not_active Abandoned
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- 2004-04-16 US US10/828,483 patent/US20040198715A1/en not_active Abandoned
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- 2004-09-15 US US10/942,197 patent/US20050032721A1/en not_active Abandoned
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2009
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