CA2488526A1

CA2488526A1 - Stable liquid parenteral parecoxib formulation

Stable liquid parenteral parecoxib formulation Download PDF

Info

Publication number: CA2488526A1
Authority: CA; Canada
Prior art keywords: parecoxib; composition; solvent liquid; salt; amount
Prior art date: 2002-06-26
Legal status : Abandoned

Application number

CA002488526A

Other languages

English (en)

French (fr)

Inventor

Yatin R. Gokarn

Richard Schartman

Current Assignee

Pharmacia LLC

Original Assignee

Individual

Priority date

2002-06-26

Filing date

2003-06-18

Publication date

2004-01-08

2003-06-18 Application filed by Individual filed Critical Individual

2004-01-08 Publication of CA2488526A1 publication Critical patent/CA2488526A1/en

Status Abandoned legal-status Critical Current

Links

239000000203 mixture Substances 0.000 title claims abstract description 232
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229960004662 parecoxib Drugs 0.000 title claims abstract description 121
239000007788 liquid Substances 0.000 title claims abstract description 77
238000009472 formulation Methods 0.000 title description 47
239000002904 solvent Substances 0.000 claims abstract description 106
LNPDTQAFDNKSHK-UHFFFAOYSA-N valdecoxib Chemical compound CC=1ON=C(C=2C=CC=CC=2)C=1C1=CC=C(S(N)(=O)=O)C=C1 LNPDTQAFDNKSHK-UHFFFAOYSA-N 0.000 claims abstract description 70
229960002004 valdecoxib Drugs 0.000 claims abstract description 68
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239000002253 acid Substances 0.000 claims abstract description 35
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