CA2472204A1 - N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases - Google Patents

N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases Download PDF

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Publication number
CA2472204A1
CA2472204A1 CA002472204A CA2472204A CA2472204A1 CA 2472204 A1 CA2472204 A1 CA 2472204A1 CA 002472204 A CA002472204 A CA 002472204A CA 2472204 A CA2472204 A CA 2472204A CA 2472204 A1 CA2472204 A1 CA 2472204A1
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CA
Canada
Prior art keywords
pyrazinyl
methoxy
dichloro
benzenesulphonamide
chloro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002472204A
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English (en)
French (fr)
Inventor
Andrew Baxter
Timothy Johnson
Nicholas Kindon
Bryan Roberts
Michael Stocks
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0200119A external-priority patent/SE0200119D0/xx
Priority claimed from SE0201857A external-priority patent/SE0201857D0/xx
Application filed by Individual filed Critical Individual
Publication of CA2472204A1 publication Critical patent/CA2472204A1/en
Abandoned legal-status Critical Current

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

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  • Health & Medical Sciences (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
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  • Virology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
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  • Urology & Nephrology (AREA)
  • Hematology (AREA)
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  • Gynecology & Obstetrics (AREA)
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  • AIDS & HIV (AREA)
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CA002472204A 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases Abandoned CA2472204A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
SE0200119-6 2002-01-16
SE0200119A SE0200119D0 (sv) 2002-01-16 2002-01-16 Novel compounds
SE0201857A SE0201857D0 (sv) 2002-06-17 2002-06-17 Novel compounds
SE0201857-0 2002-06-17
PCT/SE2003/000041 WO2003059893A1 (en) 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases

Publications (1)

Publication Number Publication Date
CA2472204A1 true CA2472204A1 (en) 2003-07-24

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CA002472204A Abandoned CA2472204A1 (en) 2002-01-16 2003-01-14 N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases

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US (2) US7662825B2 (enExample)
EP (1) EP1467976B1 (enExample)
JP (1) JP4504021B2 (enExample)
KR (1) KR20040073566A (enExample)
CN (1) CN100357275C (enExample)
AR (1) AR038179A1 (enExample)
AT (1) ATE534635T1 (enExample)
AU (1) AU2003201802A1 (enExample)
BR (1) BR0306922A (enExample)
CA (1) CA2472204A1 (enExample)
CO (1) CO5640137A2 (enExample)
ES (1) ES2375107T3 (enExample)
IL (1) IL162678A0 (enExample)
IS (1) IS7348A (enExample)
MX (1) MXPA04006806A (enExample)
NO (1) NO20043370L (enExample)
NZ (1) NZ533750A (enExample)
PL (1) PL371432A1 (enExample)
RU (1) RU2312105C9 (enExample)
TW (1) TWI328007B (enExample)
WO (1) WO2003059893A1 (enExample)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
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EP1541563A4 (en) * 2002-07-10 2007-11-07 Ono Pharmaceutical Co ANTAGONIST OF CCR4 AND CORRESPONDING MEDICINAL USE
GB0217431D0 (en) 2002-07-27 2002-09-04 Astrazeneca Ab Novel compounds
DE60318219T2 (de) 2002-08-24 2009-01-15 Astrazeneca Ab PYRIMIDINDERIVATE ALS MODULATOREN DER AKTIVITuT VON CHEMOKINREZEPTOREN
SE0301653D0 (sv) * 2003-06-05 2003-06-05 Astrazeneca Ab Novel compounds
SE0302304D0 (sv) * 2003-08-27 2003-08-27 Astrazeneca Ab Novel compounds
US7732442B2 (en) 2003-09-05 2010-06-08 Ono Pharmaceutical Co., Ltd. Chemokine receptor antagonist and medical use thereof
GB0401269D0 (en) * 2004-01-21 2004-02-25 Astrazeneca Ab Compounds
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