CA2464951C - Spirocyclic 3-phenyl-3-substituted-4-ketolactams and -lactones - Google Patents

Spirocyclic 3-phenyl-3-substituted-4-ketolactams and -lactones Download PDF

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Publication number
CA2464951C
CA2464951C CA2464951A CA2464951A CA2464951C CA 2464951 C CA2464951 C CA 2464951C CA 2464951 A CA2464951 A CA 2464951A CA 2464951 A CA2464951 A CA 2464951A CA 2464951 C CA2464951 C CA 2464951C
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CA
Canada
Prior art keywords
methyl
spp
alkyl
ethyl
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CA2464951A
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English (en)
French (fr)
Other versions
CA2464951A1 (en
Inventor
Reiner Fischer
Astrid Ullmann
Thomas Bretschneider
Mark Wilhelm Drewes
Christoph Erdelen (Deceased)
Dieter Feucht
Udo Reckmann
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Bayer CropScience AG
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Bayer CropScience AG
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Filing date
Publication date
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Publication of CA2464951A1 publication Critical patent/CA2464951A1/en
Application granted granted Critical
Publication of CA2464951C publication Critical patent/CA2464951C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A01N43/12Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings condensed with a carbocyclic ring
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • A01N43/38Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/54Spiro-condensed
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/94Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom spiro-condensed with carbocyclic rings or ring systems, e.g. griseofulvins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/10Spiro-condensed systems

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Furan Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA2464951A 2001-09-24 2002-09-11 Spirocyclic 3-phenyl-3-substituted-4-ketolactams and -lactones Expired - Fee Related CA2464951C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10146910.1 2001-09-24
DE10146910A DE10146910A1 (de) 2001-09-24 2001-09-24 Spirocyclische 3-Phenyl-3-substituierte-4-ketolaktame und -laktone
PCT/EP2002/010158 WO2003029213A1 (de) 2001-09-24 2002-09-11 Spirocyclische 3-phenyl-3-substituierte-4-ketolaktame und -laktone

Publications (2)

Publication Number Publication Date
CA2464951A1 CA2464951A1 (en) 2003-04-10
CA2464951C true CA2464951C (en) 2011-04-19

Family

ID=7700022

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2464951A Expired - Fee Related CA2464951C (en) 2001-09-24 2002-09-11 Spirocyclic 3-phenyl-3-substituted-4-ketolactams and -lactones

Country Status (20)

Country Link
US (2) US7425575B2 (cg-RX-API-DMAC7.html)
EP (2) EP1432680B1 (cg-RX-API-DMAC7.html)
JP (2) JP4532112B2 (cg-RX-API-DMAC7.html)
KR (2) KR100969572B1 (cg-RX-API-DMAC7.html)
CN (4) CN1837194B (cg-RX-API-DMAC7.html)
AR (2) AR036607A1 (cg-RX-API-DMAC7.html)
AT (1) ATE428695T1 (cg-RX-API-DMAC7.html)
BR (1) BR0212984A (cg-RX-API-DMAC7.html)
CA (1) CA2464951C (cg-RX-API-DMAC7.html)
CO (1) CO5580821A2 (cg-RX-API-DMAC7.html)
DE (2) DE10146910A1 (cg-RX-API-DMAC7.html)
EG (1) EG23387A (cg-RX-API-DMAC7.html)
ES (2) ES2323229T3 (cg-RX-API-DMAC7.html)
MX (1) MXPA04002718A (cg-RX-API-DMAC7.html)
PL (1) PL369510A1 (cg-RX-API-DMAC7.html)
RU (1) RU2309146C2 (cg-RX-API-DMAC7.html)
TW (1) TWI310377B (cg-RX-API-DMAC7.html)
UA (1) UA79242C2 (cg-RX-API-DMAC7.html)
WO (1) WO2003029213A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200402259B (cg-RX-API-DMAC7.html)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10146910A1 (de) * 2001-09-24 2003-04-10 Bayer Cropscience Ag Spirocyclische 3-Phenyl-3-substituierte-4-ketolaktame und -laktone
DE10231333A1 (de) 2002-07-11 2004-01-22 Bayer Cropscience Ag Cis-Alkoxysubstituierte spirocyclische 1-H-Pyrrolidin-2,4-dion-Derivate
DE10301805A1 (de) * 2003-01-20 2004-07-29 Bayer Cropscience Ag 3-Phenylsubstituierte-3-substituierte-4-ketolaktame und -laktone
DE10301804A1 (de) * 2003-01-20 2004-07-29 Bayer Cropscience Ag 2,4-Dihalogen-6-(C2-C3-alkyl)-phenyl substituierte Tetramsäure-Derivate
DE10301806A1 (de) * 2003-01-20 2004-07-29 Bayer Cropscience Ag Selektive Herbizide auf Basis von substituierten, cyclischen Dicarbonylverbindungen und Safenern
DE10320782A1 (de) * 2003-05-09 2004-11-25 Bayer Cropscience Ag Substituierte Oxyarene
DE102004001433A1 (de) * 2004-01-09 2005-08-18 Bayer Cropscience Ag cis-Alkoxyspiro-substituierte Tetramsäure-Derivate
DE102004035131A1 (de) * 2004-07-20 2006-02-16 Bayer Cropscience Ag Selektive Insektizide und/oder Akarizide auf Basis von substituierten, cyclischen Dicarbonylverbindungen und Safenern
US20080200499A1 (en) * 2004-07-20 2008-08-21 Reiner Fischer Selective Insecticides and/or Acaricides Based on Substituted Cyclic Dicarbonyl Compounds and Safeners
DE102004047922A1 (de) * 2004-10-01 2006-04-06 Bayer Cropscience Ag Wirkstoffe für die Saatgutbehandlung
DE102006015940A1 (de) * 2006-04-05 2007-10-11 Bayer Cropscience Ag Flüssige Formulierungen im Pflanzenschutz und deren Verwendung
DE102006050148A1 (de) 2006-10-25 2008-04-30 Bayer Cropscience Ag Trifluormethoxy-phenylsubstituierte Tetramsäure-Derivate
DE102006057037A1 (de) * 2006-12-04 2008-06-05 Bayer Cropscience Ag cis-Alkoxyspirocyclische biphenylsubstituierte Tetramsäure-Derivate
FR2923356B1 (fr) * 2007-11-09 2010-01-22 Xeda International Utilisation de solutions d'huile de menthe ou de l-carvone pour le traitement fongicide et/ou antigerminatif des bulbes et/ou tubercules
EP2071952A1 (de) * 2007-12-21 2009-06-24 Bayer CropScience AG Verwendung von Tetramsäurederivaten zur Bekämpfung von Schaderregern durch Angiessen oder Tröpfchenapplikation
CN101235023B (zh) * 2008-03-04 2010-06-02 浙江大学 一种螺螨酯的合成方法
JP5619001B2 (ja) * 2008-07-31 2014-11-05 サノフイ ストレプトスピロール誘導体
WO2011151197A1 (en) * 2010-05-31 2011-12-08 Syngenta Participations Ag 1, 8 -diazaspiro [4.5] decane- 2, 4 -dione derivatives useful as pesticides
WO2011151194A1 (en) * 2010-05-31 2011-12-08 Syngenta Participations Ag 1, 8 -diazaspiro [4.5] decane- 2, 4 -dione derivatives useful as pesticides
TW202002787A (zh) * 2018-04-13 2020-01-16 德商拜耳作物科學股份有限公司 吡咯酮酸(tetramic acid)藉由濕透及滴落施予以控制動物害蟲之用途
WO2019197617A1 (de) * 2018-04-13 2019-10-17 Bayer Cropscience Aktiengesellschaft Verwendung von tetramsäurederivaten zur bekämpfung von tierischen schädlingen durch angiessen, tröpfchenapplikation. pflanzlochbehandlung oder furchenapplikation

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US4430335A (en) * 1983-02-09 1984-02-07 Hoechst-Roussel Pharmaceuticals Inc. Substituted 1-azaspiro[4,5]decanes and their analgesic compositions
DE4216814A1 (de) * 1991-07-16 1993-01-21 Bayer Ag 3-aryl-4-hydroxy-(delta)(pfeil hoch)3(pfeil hoch)-dihydrofuranon- und 3-aryl-4-hydroxy-(delta)(pfeil hoch)3(pfeil hoch)-dihydrothiophenon-derivate
AU666040B2 (en) 1992-10-28 1996-01-25 Bayer Aktiengesellschaft Substituted 1-H-3-aryl-pyrrolidine-2,4-dione derivatives
WO1994029268A1 (de) 1993-06-07 1994-12-22 Bayer Aktiengesellschaft Iodpropargylcarbamate und ihre verwendung als biozide im pflanzen- und materialschutz
ATE208779T1 (de) * 1993-07-02 2001-11-15 Bayer Ag Substituierte spiroheterocyclische 1h-3-aryl- pyrrolidin-2,4-dion-derivate, verfahren zu deren herstellung und deren verwendung als schädlingsbekämpfungsmittel
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EP0809629B1 (de) * 1995-02-13 2004-06-30 Bayer CropScience AG 2-phenylsubstituierte heterocyclische 1,3-ketoenole als herbizide und pestizide
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DE19651686A1 (de) 1996-12-12 1998-06-18 Bayer Ag Neue substituierte Phenylketoenole
JPH10258555A (ja) 1997-03-19 1998-09-29 Citizen Watch Co Ltd ペーパーカッター装置
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JP2000086628A (ja) * 1998-09-11 2000-03-28 Otsuka Chem Co Ltd 3−アリール−3−置換−2,4−ジオン−5員環化合物、その製造法及び該化合物を含有する殺虫、殺ダニ剤
AU771383B2 (en) * 1998-12-08 2004-03-18 Rohm And Haas Company Dirt pickup resistant coating binder and coatings
DE10016544A1 (de) 2000-04-03 2001-10-11 Bayer Ag C2-phenylsubstituierte Ketoenole
DE10146910A1 (de) * 2001-09-24 2003-04-10 Bayer Cropscience Ag Spirocyclische 3-Phenyl-3-substituierte-4-ketolaktame und -laktone

Also Published As

Publication number Publication date
ES2539528T3 (es) 2015-07-01
CN1837194B (zh) 2010-06-16
DE50213460D1 (de) 2009-05-28
BR0212984A (pt) 2004-10-13
JP4532112B2 (ja) 2010-08-25
US8063096B2 (en) 2011-11-22
ES2323229T3 (es) 2009-07-09
JP5231339B2 (ja) 2013-07-10
CN1837194A (zh) 2006-09-27
EG23387A (en) 2005-03-30
KR20040044877A (ko) 2004-05-31
MXPA04002718A (es) 2004-07-05
PL369510A1 (en) 2005-04-18
US7425575B2 (en) 2008-09-16
RU2004112772A (ru) 2005-10-10
EP1432680B1 (de) 2009-04-15
CA2464951A1 (en) 2003-04-10
CN101851243A (zh) 2010-10-06
EP2030969A1 (de) 2009-03-04
TWI310377B (en) 2009-06-01
ZA200402259B (en) 2005-05-25
CN1280272C (zh) 2006-10-18
EP2030969B1 (de) 2015-03-18
AR082924A2 (es) 2013-01-16
JP2005508928A (ja) 2005-04-07
KR100969572B1 (ko) 2010-07-12
CO5580821A2 (es) 2005-11-30
US20080274893A1 (en) 2008-11-06
WO2003029213A9 (de) 2003-11-13
CN101792450A (zh) 2010-08-04
UA79242C2 (en) 2007-06-11
RU2309146C2 (ru) 2007-10-27
US20050032885A1 (en) 2005-02-10
ATE428695T1 (de) 2009-05-15
JP2009235084A (ja) 2009-10-15
KR100995548B1 (ko) 2010-11-19
AR036607A1 (es) 2004-09-22
EP1432680A1 (de) 2004-06-30
WO2003029213A1 (de) 2003-04-10
DE10146910A1 (de) 2003-04-10
KR20090052395A (ko) 2009-05-25
CN1558899A (zh) 2004-12-29

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