CA2364281A1 - Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils - Google Patents

Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils Download PDF

Info

Publication number
CA2364281A1
CA2364281A1 CA002364281A CA2364281A CA2364281A1 CA 2364281 A1 CA2364281 A1 CA 2364281A1 CA 002364281 A CA002364281 A CA 002364281A CA 2364281 A CA2364281 A CA 2364281A CA 2364281 A1 CA2364281 A1 CA 2364281A1
Authority
CA
Canada
Prior art keywords
group
c4alkyl
hydrogen
groups
optionally substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002364281A
Other languages
English (en)
French (fr)
Inventor
Venkataraman Kameswaran
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2364281A1 publication Critical patent/CA2364281A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/04—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms
    • C07C275/20—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an unsaturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/06—1,3-Oxazines; Hydrogenated 1,3-oxazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CA002364281A 1999-02-16 2000-02-14 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils Abandoned CA2364281A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25066099A 1999-02-16 1999-02-16
US09/250,660 1999-02-16
PCT/US2000/003731 WO2000049002A1 (en) 1999-02-16 2000-02-14 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils

Publications (1)

Publication Number Publication Date
CA2364281A1 true CA2364281A1 (en) 2000-08-24

Family

ID=22948652

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002364281A Abandoned CA2364281A1 (en) 1999-02-16 2000-02-14 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils

Country Status (11)

Country Link
EP (1) EP1169308A1 (cs)
JP (1) JP4619542B2 (cs)
KR (1) KR20020000140A (cs)
CN (1) CN1344259A (cs)
AU (1) AU2759800A (cs)
CA (1) CA2364281A1 (cs)
CZ (1) CZ20012948A3 (cs)
HU (1) HUP0201942A3 (cs)
IL (1) IL144776A0 (cs)
MX (1) MXPA01008188A (cs)
WO (1) WO2000049002A1 (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105211076A (zh) * 2015-10-31 2016-01-06 许自协 一种抑制水稻细菌性谷枯病菌生长的化合物
CN105175403A (zh) * 2015-10-31 2015-12-23 许自协 一种抑制菜豆细菌性萎蔫病菌生长的化合物
CN105198870A (zh) * 2015-10-31 2015-12-30 许自协 一种抑制玉米内州萎蔫病菌生长的化合物
CN105384732A (zh) * 2015-10-31 2016-03-09 许自协 一种抑制水稻细菌性条斑病菌生长的化合物
CN105211077A (zh) * 2015-10-31 2016-01-06 许自协 一种抑制番茄细菌性叶斑病菌生长的化合物
CN105165847A (zh) * 2015-10-31 2015-12-23 许自协 一种抑制苜蓿细菌性萎蔫病菌生长的化合物
CN105330654A (zh) * 2015-11-01 2016-02-17 许自协 一种抑制向日葵白锈病菌生长的化合物
CN105211078A (zh) * 2015-11-01 2016-01-06 许自协 一种抑制落叶松枯梢病菌生长的化合物
CN105330655A (zh) * 2015-11-01 2016-02-17 许自协 一种抑制黄瓜黑星病菌生长的化合物
CN105153138A (zh) * 2015-11-01 2015-12-16 许自协 一种抑制李黑节病菌生长的化合物
CN105165849A (zh) * 2015-11-02 2015-12-23 许自协 一种抑制小麦矮腥黑穗病菌生长的化合物
CN105165848A (zh) * 2015-11-02 2015-12-23 许自协 一种抑制香蕉枯萎病菌生长的化合物
CN105211079A (zh) * 2015-11-02 2016-01-06 许自协 一种抑制大豆茎褐腐病菌生长的化合物
ES2900867T3 (es) 2016-05-24 2022-03-18 Basf Se Uracilpiridina herbicida
US11292784B2 (en) 2017-11-27 2022-04-05 Basf Se Crystalline forms of ethyl 2-[[3-[[3- chloro-5-fluoro-6-[3-methyl-2,6-dioxo-4-(trifluoromethyl)pyrimidin-1-yl]-2-pyridyl]oxy] acetate
WO2023161172A1 (de) 2022-02-22 2023-08-31 Bayer Aktiengesellschaft Substituierte n-benzoesäureuracile sowie deren salze und ihre verwendung als herbizide wirkstoffe
EP4230621A1 (de) 2022-02-22 2023-08-23 Bayer AG Substituierte n-benzoesäureuracile sowie deren salze und ihre verwendung als herbizide wirkstoffe
EP4230620A1 (de) 2022-02-22 2023-08-23 Bayer Aktiengesellschaft Substituierte n-amino-n´-benzoesäureuracile sowie deren salze und ihre verwendung als herbizide wirkstoffe

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK366887A (da) * 1986-07-31 1988-05-13 Hoffmann La Roche Pyrimidinderivater
EP0260621A3 (de) * 1986-09-18 1989-03-15 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft 3-Aryluracil-enoläther und deren Verwendung zur Unkrautbekämpfung
KR920700211A (ko) * 1989-06-09 1992-02-19 베르너 벨데크 헤테로 고리 화합물
IL125947A0 (en) * 1997-09-17 1999-04-11 American Cyanamid Co 3-(1,2-benzisothiazol- and isoxazol-5-yl)-2,4(1h,3h)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-yl)-4(3)-pyrimidinone or thione herbicidal agents
DE19750195A1 (de) * 1997-11-13 1999-05-20 Bayer Ag Verfahren zur Herstellung von Ar(alk)yluracilen, neue Zwischenprodukte hierfür und Verfahren zu deren Herstellung
EP0985670A1 (en) * 1998-08-13 2000-03-15 American Cyanamid Company 1-(3-Heterocyclylphenyl)isothiourea, -isourea, -guanidine and -amidine compounds as herbicides

Also Published As

Publication number Publication date
HUP0201942A3 (en) 2002-12-28
CN1344259A (zh) 2002-04-10
EP1169308A1 (en) 2002-01-09
MXPA01008188A (es) 2003-07-21
IL144776A0 (en) 2002-06-30
JP4619542B2 (ja) 2011-01-26
AU2759800A (en) 2000-09-04
CZ20012948A3 (cs) 2002-07-17
JP2002537289A (ja) 2002-11-05
KR20020000140A (ko) 2002-01-04
HUP0201942A2 (en) 2002-09-28
WO2000049002A1 (en) 2000-08-24

Similar Documents

Publication Publication Date Title
CA2364281A1 (en) Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils
TWI534137B (zh) 抗感染劑及其用途
JP5931683B2 (ja) 抗感染症ピリミジンおよびその使用
AU737864B2 (en) 3-(1,2-benzisothiazol-and isoxazol-5-yl)-2,4(1H,3H)- pyrimidinedione or thione and 3-(1,2-benzisothiazol-and isoxazol-5-yl)-4(3H)-pyrimidinone or thione herbicidal agents
AU2002352015B2 (en) 5-phenylpyrimidines, agents comprising the same, method for production and use thereof
US6355796B1 (en) Processes and intermediate compounds for the preparation of 2-(N,N-disubstituted) amino-4-(perfluoroalkyl)-1, 3- oxazin-6-one and 6-(perfluoroalkyl) uracil compounds
CA2362990A1 (en) Process for the preparation of 6-(perfluoroalkyl)uracil compounds
JPH07278119A (ja) ２−アリールピリミジンおよびそれを使用する除草剤
US6191275B1 (en) Process for the preparation of 6-(perfluoroalkyl) uracil compounds form urea compounds
CA2362996A1 (en) Process for the preparation of 6-(perfluoroalkyl)uracil compounds from carbamate compounds
CA2363000A1 (en) Process for the preparation of 6-(perfluoroalkyl) uracil compounds from urea compounds
Novakov et al. Synthesis of 2-[(ω-phthalimidoalkyl) sulfanyl]-pyrimidin-4 (3 H)-ones, their cytotoxicity and in vitro activity against HIV-1/2
US6313295B1 (en) Process for the preparation of 6-(perfluoroalkyl) uracil compounds from carbamate compounds

Legal Events

Date Code Title Description
FZDE Discontinued