CA2331870C - Nouveaux composes cycliques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent - Google Patents

Nouveaux composes cycliques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent Download PDF

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CA2331870C
CA2331870C CA002331870A CA2331870A CA2331870C CA 2331870 C CA2331870 C CA 2331870C CA 002331870 A CA002331870 A CA 002331870A CA 2331870 A CA2331870 A CA 2331870A CA 2331870 C CA2331870 C CA 2331870C
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formula
ethyl
group
acid
preparation
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French (fr)
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CA2331870A1 (fr
Inventor
Daniel Lesieur
Frederique Klupsch
Gerald Guillaumet
Marie-Claude Viaud
Michel Langlois
Caroline Bennejean
Pierre Renard
Philippe Delagrange
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Laboratoires Servier SAS
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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    • C07C233/43—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of a saturated carbon skeleton
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US6872851B1 (en) 2005-03-29
AU747301B2 (en) 2002-05-16
CN1304400A (zh) 2001-07-18
NO20005715L (no) 2000-11-13
JP2002514620A (ja) 2002-05-21
DE69933147D1 (de) 2006-10-19
ES2255260T3 (es) 2006-06-16
AU3610399A (en) 1999-11-29
HUP0101813A2 (hu) 2001-11-28
ATE312073T1 (de) 2005-12-15
PL344048A1 (en) 2001-09-24
FR2778662A1 (fr) 1999-11-19
NO20005714D0 (no) 2000-11-13
JP2002514619A (ja) 2002-05-21
HUP0101813A3 (en) 2002-10-28
BR9911771A (pt) 2001-10-02
DK1077927T3 (da) 2006-04-18
US20040002491A1 (en) 2004-01-01
WO1999058496A1 (fr) 1999-11-18
US7183318B2 (en) 2007-02-27
BR9911783A (pt) 2002-12-31
ES2255261T3 (es) 2006-06-16
EP1077927B1 (fr) 2005-12-07
US20050124682A1 (en) 2005-06-09
DE69933147T2 (de) 2006-12-21
DK1077928T3 (da) 2006-04-18
AU3610499A (en) 1999-11-29
NO20005714L (no) 2000-11-13
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US20050059729A1 (en) 2005-03-17
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DE69933149T2 (de) 2006-12-21
HUP0101800A3 (en) 2002-12-28
US6605632B1 (en) 2003-08-12
EP1077928A1 (fr) 2001-02-28
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US7115752B2 (en) 2006-10-03
ATE312072T1 (de) 2005-12-15
CA2331870A1 (fr) 1999-11-18
FR2778662B1 (fr) 2000-06-16
EP1077927A1 (fr) 2001-02-28
EP1077928B1 (fr) 2005-12-07
AU748567B2 (en) 2002-06-06
PL344012A1 (en) 2001-09-24
WO1999058495A1 (fr) 1999-11-18
CN1300277A (zh) 2001-06-20
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US20040002490A1 (en) 2004-01-01
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