CA1204117A - Azolylmethyloxiranes, their preparation and their use as drugs - Google Patents

Azolylmethyloxiranes, their preparation and their use as drugs

Info

Publication number
CA1204117A
CA1204117A CA000426058A CA426058A CA1204117A CA 1204117 A CA1204117 A CA 1204117A CA 000426058 A CA000426058 A CA 000426058A CA 426058 A CA426058 A CA 426058A CA 1204117 A CA1204117 A CA 1204117A
Authority
CA
Canada
Prior art keywords
formula
compound
carbon atoms
above meanings
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000426058A
Other languages
English (en)
French (fr)
Inventor
Bernd Janssen
Norbert Meyer
Friedrich-Wilhelm Kohlmann
Walter Wesenberg
Wolfgang Heberle
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Application granted granted Critical
Publication of CA1204117A publication Critical patent/CA1204117A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/263—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
    • C07C17/2635—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions involving a phosphorus compound, e.g. Wittig synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/08—Compounds containing oxirane rings with hydrocarbon radicals, substituted by halogen atoms, nitro radicals or nitroso radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA000426058A 1982-05-14 1983-04-18 Azolylmethyloxiranes, their preparation and their use as drugs Expired CA1204117A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19823218129 DE3218129A1 (de) 1982-05-14 1982-05-14 Azolylmethyloxirane, ihre herstellung und verwendung als arzneimittel
DEP3218129.9 1982-05-14

Publications (1)

Publication Number Publication Date
CA1204117A true CA1204117A (en) 1986-05-06

Family

ID=6163548

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000426058A Expired CA1204117A (en) 1982-05-14 1983-04-18 Azolylmethyloxiranes, their preparation and their use as drugs

Country Status (5)

Country Link
JP (1) JPS58206585A (da)
CA (1) CA1204117A (da)
DE (1) DE3218129A1 (da)
FI (1) FI77660C (da)
ZA (1) ZA833362B (da)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5057531A (en) * 1988-02-26 1991-10-15 Basf Aktiengesellschaft Azolylmethyloxiranes and fungicides containing these compounds
US5268517A (en) * 1989-07-14 1993-12-07 Basf Aktiengesellschaft Stereoselective preparation of Z-1,2-diarylallyl chlorides and the conversion thereof into azolylmethyloxiranes, and novel intermediates

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3511411A1 (de) 1985-03-29 1986-10-02 Basf Ag, 6700 Ludwigshafen Verwendung von azolylmethyloxiranen zur bekaempfung von viralen erkrankungen
IL78175A (en) * 1985-03-29 1989-10-31 Basf Ag Azolylmethyloxiranes,their preparation and their use as fungicide crop protection agents
DE3907729A1 (de) * 1989-03-10 1990-09-13 Basf Ag Trifluormethylphenylazolylmethyloxirane, verfahren zu ihrer herstellung und deren verwendung als pflanzenschutzmittel
JP2975058B2 (ja) * 1989-07-18 1999-11-10 ビーエーエスエフ アクチェンゲゼルシャフト 新規のｚ―１，２―ジアリール―アリルクロリド及びその立体配置選択的製造方法ならびにこれから製造される新規のクロルメチル―ジアリール―オキシラン
CN101208322A (zh) * 2005-06-27 2008-06-25 马克特辛姆化学工厂有限公司 改进的取代的1-卤代甲基-2-苯基-1-苯基环氧乙烷的合成方法
JP2009541253A (ja) * 2006-06-21 2009-11-26 ビーエーエスエフ ソシエタス・ヨーロピア アゾリルメチルオキシラン、植物病原菌類を防除するためのその使用、およびそれを含む組成物
JP2009541250A (ja) * 2006-06-23 2009-11-26 ビーエーエスエフ ソシエタス・ヨーロピア アゾリルメチルオキシラン、植物病原菌類を防除するためのその使用、およびそれを含む組成物
JP2009541263A (ja) * 2006-06-23 2009-11-26 ビーエーエスエフ ソシエタス・ヨーロピア アゾリルメチルオキシラン、植物病原菌類を防除するためのその使用、およびそれを含む組成物
CN101484446B (zh) * 2006-07-05 2011-07-13 巴斯夫欧洲公司 唑基甲基环氧乙烷及其在防治植物病原性真菌中的用途和包含所述化合物的试剂
CN101484450B (zh) * 2006-07-05 2011-08-03 巴斯夫欧洲公司 唑基甲基环氧乙烷及其在防治植物病原性真菌中的用途和包含所述化合物的试剂
EP2046780A1 (de) * 2006-07-24 2009-04-15 Basf Se Azolylmethyloxirane, ihre verwendung zur bekämpfung von pflanzenpathogenen pilzen sowie sie enthaltende mittel
WO2008012234A2 (de) * 2006-07-25 2008-01-31 Basf Se Azolylmethyloxirane, ihre verwendung zur bekämpfung von pflanzenpathogenen pilzen sowie sie enthaltende mittel
US7994340B2 (en) * 2006-12-22 2011-08-09 Basf Se Azolylmethyloxiranes, their use for controlling phytopathogenic fungi, and compositions comprising them
EA201000950A1 (ru) * 2007-12-19 2011-02-28 Басф Се Азолилметилоксираны, их применение, а также содержащие их средства
WO2009077497A2 (de) * 2007-12-19 2009-06-25 Basf Se Azolylmethyloxirane, ihre verwendung sowie sie enthaltende mittel
JP2011506543A (ja) * 2007-12-19 2011-03-03 ビーエーエスエフ ソシエタス・ヨーロピア アゾリルメチルオキシラン、その使用及びそれを含む薬剤
WO2009077471A2 (de) * 2007-12-19 2009-06-25 Basf Se Azolylmethyloxirane, ihre verwendung sowie sie enthaltende mittel
EP2746276A1 (en) 2012-12-19 2014-06-25 Basf Se New substituted triazoles and imidazoles and their use as fungicides
WO2014095555A1 (en) 2012-12-19 2014-06-26 Basf Se New substituted triazoles and imidazoles and their use as fungicides
EP2746275A1 (en) 2012-12-19 2014-06-25 Basf Se New substituted triazoles and imidazoles and their use as fungicides
MX2019003713A (es) 2016-09-29 2019-06-24 Bayer Cropscience Ag Derivados de imidazolilmetiloxirano 5-sustituido novedosos.

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5057531A (en) * 1988-02-26 1991-10-15 Basf Aktiengesellschaft Azolylmethyloxiranes and fungicides containing these compounds
US5268517A (en) * 1989-07-14 1993-12-07 Basf Aktiengesellschaft Stereoselective preparation of Z-1,2-diarylallyl chlorides and the conversion thereof into azolylmethyloxiranes, and novel intermediates

Also Published As

Publication number Publication date
JPH0474355B2 (da) 1992-11-26
FI77660C (fi) 1989-04-10
FI831590A0 (fi) 1983-05-09
FI77660B (fi) 1988-12-30
ZA833362B (en) 1984-02-29
FI831590L (fi) 1983-11-15
JPS58206585A (ja) 1983-12-01
DE3218129A1 (de) 1983-11-17

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Legal Events

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