CA1081228A - Amides d'oxazole, d'isoxazole, de thiazole et d'isothiazole - Google Patents

Amides d'oxazole, d'isoxazole, de thiazole et d'isothiazole

Info

Publication number
CA1081228A
CA1081228A CA271,839A CA271839A CA1081228A CA 1081228 A CA1081228 A CA 1081228A CA 271839 A CA271839 A CA 271839A CA 1081228 A CA1081228 A CA 1081228A
Authority
CA
Canada
Prior art keywords
carbon atoms
alkyl
group
compound
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA271,839A
Other languages
English (en)
Inventor
Richard A. Partyka
Ronnie R. Crenshaw
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/658,961 external-priority patent/US4001237A/en
Priority claimed from US05/658,979 external-priority patent/US4001238A/en
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of CA1081228A publication Critical patent/CA1081228A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA271,839A 1976-02-18 1977-02-15 Amides d'oxazole, d'isoxazole, de thiazole et d'isothiazole Expired CA1081228A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/658,961 US4001237A (en) 1976-02-18 1976-02-18 Oxazole, isoxazole, thiazole and isothiazole amides
US05/658,979 US4001238A (en) 1976-02-18 1976-02-18 1,3,4-oxadiazole amides

Publications (1)

Publication Number Publication Date
CA1081228A true CA1081228A (fr) 1980-07-08

Family

ID=27097727

Family Applications (1)

Application Number Title Priority Date Filing Date
CA271,839A Expired CA1081228A (fr) 1976-02-18 1977-02-15 Amides d'oxazole, d'isoxazole, de thiazole et d'isothiazole

Country Status (16)

Country Link
JP (1) JPS584716B2 (fr)
CA (1) CA1081228A (fr)
CH (1) CH635838A5 (fr)
CY (1) CY1122A (fr)
DE (1) DE2707067A1 (fr)
DK (1) DK65177A (fr)
FI (1) FI770485A (fr)
FR (1) FR2348924A1 (fr)
GB (1) GB1533529A (fr)
IE (1) IE44614B1 (fr)
KE (1) KE3155A (fr)
LU (1) LU76802A1 (fr)
MY (1) MY8200110A (fr)
NL (1) NL7701753A (fr)
SE (1) SE7701732L (fr)
YU (4) YU45477A (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5791987A (en) * 1980-11-26 1982-06-08 Sankyo Co Ltd Aminoquinazoline derivative and its preparation
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
US5994294A (en) * 1996-02-02 1999-11-30 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
JP2005538968A (ja) * 2002-06-29 2005-12-22 ツェンタリス ゲゼルシャフト ミット ベシュレンクテル ハフツング アリール−及びヘテロアリールカルボニルピペラジン及び良性及び悪性の腫瘍疾患を治療するためのその使用

Also Published As

Publication number Publication date
IE44614B1 (en) 1982-01-27
FR2348924B1 (fr) 1980-05-09
IE44614L (en) 1977-08-18
FR2348924A1 (fr) 1977-11-18
DK65177A (da) 1977-08-19
DE2707067A1 (de) 1977-08-25
YU45477A (en) 1982-10-31
YU267780A (en) 1983-06-30
CH635838A5 (en) 1983-04-29
LU76802A1 (fr) 1977-09-12
SE7701732L (sv) 1977-08-19
YU161282A (en) 1982-10-31
MY8200110A (en) 1982-12-31
CY1122A (en) 1981-12-04
JPS584716B2 (ja) 1983-01-27
JPS52102286A (en) 1977-08-27
GB1533529A (en) 1978-11-29
AU2242677A (en) 1978-07-06
FI770485A (fr) 1977-08-19
KE3155A (en) 1981-09-18
YU161182A (en) 1982-10-31
NL7701753A (nl) 1977-08-22

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Legal Events

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