CA1064930A - Substituted benzamides and derivatives thereof - Google Patents

Substituted benzamides and derivatives thereof

Info

Publication number
CA1064930A
CA1064930A CA254,480A CA254480A CA1064930A CA 1064930 A CA1064930 A CA 1064930A CA 254480 A CA254480 A CA 254480A CA 1064930 A CA1064930 A CA 1064930A
Authority
CA
Canada
Prior art keywords
group
methoxy
ethyl
hydroxyethyl
sulphamoyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA254,480A
Other languages
English (en)
French (fr)
Inventor
Michel Thominet
Gerard Bulteau
Jacques Acher
Jean-Claude Monier
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Societe dEtudes Scientifiques et Industrielles de lIle de France SA
Original Assignee
Societe dEtudes Scientifiques et Industrielles de lIle de France SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Societe dEtudes Scientifiques et Industrielles de lIle de France SA filed Critical Societe dEtudes Scientifiques et Industrielles de lIle de France SA
Application granted granted Critical
Publication of CA1064930A publication Critical patent/CA1064930A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09Radicals substituted by nitrogen atoms, not forming part of a nitro radical

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Otolaryngology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CA254,480A 1975-06-10 1976-06-09 Substituted benzamides and derivatives thereof Expired CA1064930A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7518001A FR2313935A1 (fr) 1975-06-10 1975-06-10 Nouveaux benzamides substitues, leurs derives et leur procede de preparation

Publications (1)

Publication Number Publication Date
CA1064930A true CA1064930A (en) 1979-10-23

Family

ID=9156239

Family Applications (1)

Application Number Title Priority Date Filing Date
CA254,480A Expired CA1064930A (en) 1975-06-10 1976-06-09 Substituted benzamides and derivatives thereof

Country Status (37)

Country Link
JP (1) JPS6055503B2 (de)
AR (1) AR210888A1 (de)
AT (1) AT358571B (de)
AU (1) AU506001B2 (de)
BE (1) BE842059A (de)
BG (1) BG27360A3 (de)
CA (1) CA1064930A (de)
CH (1) CH596175A5 (de)
CS (1) CS189007B2 (de)
DD (1) DD124380A5 (de)
DE (1) DE2623075A1 (de)
DK (1) DK255276A (de)
EG (1) EG12285A (de)
ES (1) ES448643A1 (de)
FI (1) FI761669A (de)
FR (1) FR2313935A1 (de)
GB (1) GB1500105A (de)
HK (1) HK46979A (de)
HU (1) HU172195B (de)
IE (1) IE43375B1 (de)
IN (1) IN142899B (de)
LU (1) LU75104A1 (de)
MW (1) MW1676A1 (de)
MX (1) MX3580E (de)
NL (1) NL186382C (de)
NO (1) NO146058C (de)
NZ (1) NZ181072A (de)
OA (1) OA05350A (de)
PH (1) PH13912A (de)
PL (2) PL103075B1 (de)
PT (1) PT65164B (de)
RO (1) RO70265A (de)
SE (1) SE415971B (de)
SU (2) SU607551A3 (de)
YU (1) YU39352B (de)
ZA (1) ZA763042B (de)
ZM (1) ZM6576A1 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ186175A (en) * 1977-01-27 1980-03-05 Shionogi & Co Meta-sulphonamidobenzamide derivatives
FR2415099A1 (fr) * 1978-01-20 1979-08-17 Ile De France Nouveaux derives de 4-amino-5-alkylsulfonyl ortho-anisamides, leurs procedes de preparation et leur application comme psychotropes
FR2438650A1 (fr) * 1978-10-11 1980-05-09 Ile De France N-(1-methyl 2-pyrrolidinyl methyl) 2,3-dimethoxy 5-methylsulfamoyl benzamide et ses derives, leurs methodes de preparation et leur application dans le traitement des troubles du bas appareil urinaire
JPS597160A (ja) * 1982-06-28 1984-01-14 ラボラトリーオス・デラグランヘ・エセ・ア N−(1−プロピル−2−ピロリジニルメチル)−2−メトキシ−5−スルフアモイルベンズアミド、その製造方法およびこれを有効成分とする抗うつ剤
US4820715A (en) * 1984-06-28 1989-04-11 Bristol-Myers Company Anti-emetic quinuclidinyl benzamides
US4808624A (en) * 1984-06-28 1989-02-28 Bristol-Myers Company Pharmacologically active substituted benzamides
US5011992A (en) * 1984-06-28 1991-04-30 Bristol-Myers Squibb Company Pharmacologically active substituted benzamides
JP3026845B2 (ja) * 1991-02-20 2000-03-27 日清製粉株式会社 ピペリジン誘導体
US9375486B2 (en) 2012-09-17 2016-06-28 Nektar Therapeutics Oligomer-containing benzamide-based compounds

Also Published As

Publication number Publication date
ATA400176A (de) 1980-02-15
EG12285A (en) 1978-09-30
PH13912A (en) 1980-11-04
NO146058B (no) 1982-04-13
MW1676A1 (en) 1977-10-12
ZA763042B (en) 1977-04-27
CH596175A5 (de) 1978-02-28
PT65164A (fr) 1976-07-01
DD124380A5 (de) 1977-02-16
PL102929B1 (pl) 1979-05-31
YU39352B (en) 1984-10-31
FI761669A (de) 1976-12-11
IN142899B (de) 1977-09-03
AR210888A1 (es) 1977-09-30
MX3580E (es) 1981-03-19
RO70265A (ro) 1981-06-30
AU1436076A (en) 1977-12-01
BE842059A (fr) 1976-11-22
DK255276A (da) 1976-12-11
NO761977L (de) 1976-12-13
OA05350A (fr) 1981-02-28
GB1500105A (en) 1978-02-08
ES448643A1 (es) 1977-07-01
SE415971B (sv) 1980-11-17
JPS5231041A (en) 1977-03-09
NZ181072A (en) 1978-07-28
AU506001B2 (en) 1979-12-13
NO146058C (no) 1982-07-28
PL103075B1 (pl) 1979-05-31
ZM6576A1 (en) 1977-06-21
SU607551A3 (ru) 1978-05-15
IE43375B1 (en) 1981-02-11
IE43375L (en) 1976-12-10
NL186382B (nl) 1990-06-18
NL186382C (nl) 1990-11-16
SE7606424L (sv) 1976-12-11
DE2623075A1 (de) 1976-12-30
JPS6055503B2 (ja) 1985-12-05
NL7606284A (nl) 1976-12-14
PL190247A1 (pl) 1978-03-13
SU645557A3 (ru) 1979-01-30
BG27360A3 (en) 1979-10-12
HU172195B (hu) 1978-06-28
PT65164B (fr) 1977-11-17
YU131876A (en) 1982-06-30
CS189007B2 (en) 1979-03-30
HK46979A (en) 1979-07-20
LU75104A1 (de) 1977-03-09
AT358571B (de) 1980-09-25
FR2313935A1 (fr) 1977-01-07
FR2313935B1 (de) 1979-04-27

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