BRPI9811826B8 - processos para a preparação de monossacarídeos - Google Patents

processos para a preparação de monossacarídeos

Info

Publication number
BRPI9811826B8
BRPI9811826B8 BRPI9811826A BR9811826A BRPI9811826B8 BR PI9811826 B8 BRPI9811826 B8 BR PI9811826B8 BR PI9811826 A BRPI9811826 A BR PI9811826A BR 9811826 A BR9811826 A BR 9811826A BR PI9811826 B8 BRPI9811826 B8 BR PI9811826B8
Authority
BR
Brazil
Prior art keywords
preparation
monosaccharides
processes
improved
antiparasitic
Prior art date
Application number
BRPI9811826A
Other languages
English (en)
Other versions
BR9811826A (pt
BR9811826B1 (pt
Inventor
Nigel Derek Arthur Walshe
Selena Jane Cambers
Original Assignee
Ah Usa 42 Llc
Pfizer
Zoetis Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ah Usa 42 Llc, Pfizer, Zoetis Llc filed Critical Ah Usa 42 Llc
Publication of BR9811826A publication Critical patent/BR9811826A/pt
Publication of BR9811826B1 publication Critical patent/BR9811826B1/pt
Publication of BRPI9811826B8 publication Critical patent/BRPI9811826B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

patente de invenção: <b>"processo melhorado para agente antiparasítico"<d>. processo melhorado para a preparação do composto antiparasítico monossacarídeo de 25-ciclohexil-22,23-dihidro-5-hidroxiimino-avermectina b1 a partir de doramectina e intermediários para esse processo e solvatos cristalinos do mesmo derivados.
BRPI9811826A 1997-08-05 1998-07-23 processos para a preparação de monossacarídeos BRPI9811826B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9716567.4A GB9716567D0 (en) 1997-08-05 1997-08-05 Process
GB9716567.4 1997-08-05
PCT/EP1998/004931 WO1999007721A1 (en) 1997-08-05 1998-07-23 Improved process for antiparasitic agent

Publications (3)

Publication Number Publication Date
BR9811826A BR9811826A (pt) 2000-08-15
BR9811826B1 BR9811826B1 (pt) 2015-02-03
BRPI9811826B8 true BRPI9811826B8 (pt) 2016-09-13

Family

ID=10817038

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9811826A BRPI9811826B8 (pt) 1997-08-05 1998-07-23 processos para a preparação de monossacarídeos

Country Status (35)

Country Link
US (1) US6906184B1 (pt)
EP (1) EP1003764B1 (pt)
JP (1) JP3476476B2 (pt)
KR (1) KR100336060B1 (pt)
CN (2) CN1161369C (pt)
AP (1) AP1217A (pt)
AR (1) AR016388A1 (pt)
AT (1) ATE238333T1 (pt)
AU (1) AU731854B2 (pt)
BR (1) BRPI9811826B8 (pt)
CA (1) CA2296109C (pt)
CZ (1) CZ296906B6 (pt)
DE (1) DE69813830T2 (pt)
DK (1) DK1003764T3 (pt)
EA (1) EA002103B1 (pt)
ES (1) ES2192334T3 (pt)
GB (1) GB9716567D0 (pt)
HK (1) HK1030610A1 (pt)
HR (1) HRP20000054B1 (pt)
HU (1) HU228202B1 (pt)
ID (1) ID24505A (pt)
IL (2) IL133628A0 (pt)
MA (1) MA24628A1 (pt)
MY (1) MY116766A (pt)
NO (1) NO996521L (pt)
NZ (1) NZ501969A (pt)
OA (1) OA11278A (pt)
PL (1) PL191259B1 (pt)
PT (1) PT1003764E (pt)
SK (1) SK283899B6 (pt)
TW (2) TW530059B (pt)
UA (1) UA56244C2 (pt)
WO (1) WO1999007721A1 (pt)
YU (1) YU72399A (pt)
ZA (1) ZA986970B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100998906B1 (ko) 2003-01-20 2010-12-09 엘지전자 주식회사 기록된 정지 영상의 재생을 관리하기 위한 데이터 구조를갖는 기록 매체, 그에 따른 기록 및 재생 방법 및 장치
CN103360444B (zh) * 2012-04-03 2016-05-11 浙江海正药业股份有限公司 抗寄生虫药赛拉菌素的合成新工艺
CN105061457B (zh) * 2015-08-20 2016-06-22 湖北宏中药业股份有限公司 一种米尔贝肟的合成方法
EP3150618A1 (en) 2015-09-29 2017-04-05 Virbac Process for the preparation of selamectin
EA201992125A1 (ru) 2017-03-17 2020-03-16 КРКА, д.д., НОВО МЕСТО Стабильная ветеринарная композиция для местного применения
CN107118247B (zh) * 2017-06-14 2019-07-26 博瑞生物医药（苏州）股份有限公司 塞拉菌素的制备方法
CN107021990B (zh) * 2017-06-14 2019-07-12 博瑞生物医药（苏州）股份有限公司 高纯度塞拉菌素的制备方法
CN109734760A (zh) * 2018-11-01 2019-05-10 丽珠集团新北江制药股份有限公司 一种多拉菌素杂质的制备方法
CN112830945A (zh) * 2019-11-22 2021-05-25 东莞市东阳光动物保健药品有限公司 一种大环内酯类化合物的制备方法
CN111116692A (zh) * 2020-01-14 2020-05-08 北大方正集团有限公司 一种高纯度塞拉菌素的合成方法
CN114106071A (zh) * 2021-11-11 2022-03-01 浙江荣耀生物科技股份有限公司 一种塞拉菌素的合成方法
WO2023203038A1 (en) 2022-04-19 2023-10-26 Syngenta Crop Protection Ag Insect, acarina and nematode pest control

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CS262673B2 (cs) * 1985-07-27 1989-03-14 Pfizer Způsob výroby nových derivátů avermectinu
DE3883408T2 (de) * 1987-01-23 1993-12-09 Pfizer Verfahren zur Herstellung von Avermectinen und die verwendeten Kulturen.
US5015630A (en) * 1989-01-19 1991-05-14 Merck & Co., Inc. 5-oxime avermectin derivatives
NZ233680A (en) * 1989-05-17 1995-02-24 Beecham Group Plc Avermectins and milbemycins and compositions thereof
GB9300883D0 (en) * 1993-01-18 1993-03-10 Pfizer Ltd Antiparasitic agents
US5380838A (en) * 1993-10-08 1995-01-10 Merck & Co. Inc. Stable solvates of avermectin compounds
US5587362A (en) * 1994-01-28 1996-12-24 Univ. Of Ga Research Foundation L-nucleosides

Also Published As

Publication number Publication date
CN1161369C (zh) 2004-08-11
US6906184B1 (en) 2005-06-14
JP3476476B2 (ja) 2003-12-10
MA24628A1 (fr) 1999-04-01
CN1528774A (zh) 2004-09-15
TW200300762A (en) 2003-06-16
HUP0003399A2 (hu) 2001-02-28
AU731854B2 (en) 2001-04-05
IL156463A (en) 2006-12-31
TW530059B (en) 2003-05-01
CN1266437A (zh) 2000-09-13
CZ200095A3 (cs) 2000-05-17
NO996521D0 (no) 1999-12-28
PT1003764E (pt) 2003-07-31
BR9811826A (pt) 2000-08-15
EA002103B1 (ru) 2001-12-24
IL133628A0 (en) 2001-04-30
PL191259B1 (pl) 2006-04-28
ID24505A (id) 2000-07-20
PL338557A1 (en) 2000-11-06
DE69813830T2 (de) 2003-11-06
AR016388A1 (es) 2001-07-04
GB9716567D0 (en) 1997-10-08
KR20010022592A (ko) 2001-03-26
SK283899B6 (sk) 2004-04-06
AU9339698A (en) 1999-03-01
NO996521L (no) 2000-02-03
EA199901056A1 (ru) 2000-06-26
EP1003764B1 (en) 2003-04-23
BR9811826B1 (pt) 2015-02-03
HUP0003399A3 (en) 2003-05-28
CA2296109C (en) 2003-11-04
DE69813830D1 (de) 2003-05-28
AP9801311A0 (en) 1998-09-30
DK1003764T3 (da) 2003-06-30
ATE238333T1 (de) 2003-05-15
HRP20000054A2 (en) 2000-12-31
NZ501969A (en) 2002-03-01
KR100336060B1 (ko) 2002-05-10
MY116766A (en) 2004-03-31
YU72399A (pt) 2002-08-12
ZA986970B (en) 2000-02-04
AP1217A (en) 2003-10-20
CA2296109A1 (en) 1999-02-18
CN1303094C (zh) 2007-03-07
WO1999007721A1 (en) 1999-02-18
JP2000511943A (ja) 2000-09-12
HRP20000054B1 (en) 2003-04-30
CZ296906B6 (cs) 2006-07-12
EP1003764A1 (en) 2000-05-31
ES2192334T3 (es) 2003-10-01
OA11278A (en) 2003-07-31
SK1372000A3 (en) 2000-06-12
UA56244C2 (uk) 2003-05-15
HK1030610A1 (en) 2001-05-11
HU228202B1 (en) 2013-01-28

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B25A Requested transfer of rights approved

Owner name: AH USA 42 LLC (US)

B25D Requested change of name of applicant approved

Owner name: ZOETIS LLC (US)

B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 03/02/2015, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]

Free format text: REFERENTE AO DESPACHO 16.1 PUBLICADO NA RPI 2300 DE 03.02.2015, QUANTO AO ENDERECO DO TITULAR

B25A Requested transfer of rights approved
B25G Requested change of headquarter approved