BRPI1011888A2 - processo para preparar um composto, e, composição. - Google Patents

processo para preparar um composto, e, composição.

Info

Publication number
BRPI1011888A2
BRPI1011888A2 BRPI1011888A BRPI1011888A BRPI1011888A2 BR PI1011888 A2 BRPI1011888 A2 BR PI1011888A2 BR PI1011888 A BRPI1011888 A BR PI1011888A BR PI1011888 A BRPI1011888 A BR PI1011888A BR PI1011888 A2 BRPI1011888 A2 BR PI1011888A2
Authority
BR
Brazil
Prior art keywords
preparing
compound
composition
Prior art date
Application number
BRPI1011888A
Other languages
English (en)
Portuguese (pt)
Inventor
Karl-Heinz Giselbrecht
Michael Wolberg
Ulfried Felfer
Original Assignee
Rigel Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rigel Pharmaceuticals Inc filed Critical Rigel Pharmaceuticals Inc
Publication of BRPI1011888A2 publication Critical patent/BRPI1011888A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/091Esters of phosphoric acids with hydroxyalkyl compounds with further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
BRPI1011888A 2009-07-02 2010-07-01 processo para preparar um composto, e, composição. BRPI1011888A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27007309P 2009-07-02 2009-07-02
PCT/US2010/040792 WO2011002999A1 (en) 2009-07-02 2010-07-01 Synthesis of n4- (2, 2-dimethyl-4- [ (dihydrogen phosphonoxy ] -3-oxo-5-pyrido [1, 4] oxazin-6-yl)-5-fluoro-n2- (3, 4, 5,-trimethoxyphenyl) -2, 4- pyrimidinediamine disodium salt

Publications (1)

Publication Number Publication Date
BRPI1011888A2 true BRPI1011888A2 (pt) 2016-04-12

Family

ID=42937685

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1011888A BRPI1011888A2 (pt) 2009-07-02 2010-07-01 processo para preparar um composto, e, composição.

Country Status (21)

Country Link
US (3) US8299242B2 (enExample)
EP (1) EP2448950B1 (enExample)
JP (1) JP5739882B2 (enExample)
CN (1) CN102482305B (enExample)
AU (1) AU2010266213B2 (enExample)
BR (1) BRPI1011888A2 (enExample)
CA (1) CA2766801C (enExample)
CY (1) CY1117489T1 (enExample)
DK (1) DK2448950T3 (enExample)
EA (1) EA021657B1 (enExample)
ES (1) ES2565985T3 (enExample)
HR (1) HRP20160319T1 (enExample)
HU (1) HUE027212T2 (enExample)
ME (1) ME02388B (enExample)
PL (1) PL2448950T3 (enExample)
RS (1) RS54679B1 (enExample)
SG (1) SG176799A1 (enExample)
SI (1) SI2448950T1 (enExample)
SM (1) SMT201600084B (enExample)
UA (1) UA108077C2 (enExample)
WO (1) WO2011002999A1 (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5468899B2 (ja) 2006-07-20 2014-04-09 アフィニウム ファーマシューティカルズ, インク. Fabiインヒビターとしてのアクリルアミド誘導体
UA108077C2 (xx) 2009-07-02 2015-03-25 Синтез динатрієвої солі n4-(2,2-диметил-4-$(дигідрофосфонокси)метил]-3-оксо-5-піридо$1,4]оксазин-6-іл)-5-фтор-n2-(3,4,5-триметоксифеніл)-2,4-піримідиндіаміну
US20110206661A1 (en) * 2010-02-24 2011-08-25 Auspex Pharmaceuticals, Inc. Trimethoxyphenyl inhibitors of tyrosine kinase
EP2736487B2 (en) * 2011-07-28 2024-08-28 Rigel Pharmaceuticals, Inc. New (trimethoxyphenylamino)pyrimidinyl formulations
TWI526437B (zh) * 2011-09-09 2016-03-21 台灣神隆股份有限公司 卡巴他賽之結晶型
US8426450B1 (en) * 2011-11-29 2013-04-23 Helsinn Healthcare Sa Substituted 4-phenyl pyridines having anti-emetic effect
MY170437A (en) 2012-06-19 2019-07-31 Debiopharm Int Sa Prodrug derivatives of (e)-n-methyl-n-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide
CN102746337B (zh) * 2012-06-21 2014-12-17 成都苑东药业有限公司 一种2,4-嘧啶二胺类化合物及其制备方法
TW201410657A (zh) 2012-08-02 2014-03-16 Endo Pharmaceuticals Inc 經取代胺基-嘧啶衍生物
LT3083648T (lt) * 2013-12-20 2019-01-25 Rigel Pharmaceuticals, Inc. Farmacinis būdas ir tarpiniai junginiai
PL3419628T3 (pl) 2016-02-26 2021-05-31 Debiopharm International Sa Lek do leczenia zakażeń stopy cukrzycowej
EP3509578B1 (en) 2016-09-08 2022-12-21 Glykon Technologies Group, LLC Monomeric bimetal hydroxycitric acid compounds and methods of making and using the same
JP2020536100A (ja) * 2017-10-04 2020-12-10 セルジーン コーポレイション シス−4−[2−{[(3s,4r)−3−フルオロキサン−4−イル]アミノ}−8−(2,4,6−トリクロロアニリノ)−9h−プリン−9−イル]−1−メチルシクロヘキサン−1−カルボキサミドの製造プロセス
HRP20230437T1 (hr) 2019-02-14 2023-07-07 Debiopharm International S.A. Formulacija afabicina, postupak izrade iste
CN113939306B (zh) 2019-06-14 2024-07-19 德彪药业国际股份公司 用于治疗涉及生物膜的细菌感染的药物及其用途

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US303022A (en) 1884-08-05 Egg-beater
US324087A (en) 1885-08-11 Abel combs
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
US20040024716A1 (en) 2002-04-12 2004-02-05 James Malatesta Mail sorting processes and systems
CN103169708B (zh) 2002-07-29 2018-02-02 里格尔药品股份有限公司 用2,4‑嘧啶二胺化合物治疗或者预防自体免疫性疾病的方法
US7122542B2 (en) 2003-07-30 2006-10-17 Rigel Pharmaceuticals, Inc. Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
US20060047135A1 (en) 2004-08-30 2006-03-02 Chadwick Scott T Process for preparing chloromethyl di-tert-butylphosphate
US7449458B2 (en) * 2005-01-19 2008-11-11 Rigel Pharmaceuticals, Inc. Prodrugs of 2,4-pyrimidinediamine compounds and their uses
US20090114877A1 (en) * 2005-09-13 2009-05-07 Eisai R&D Management Co., Ltd. Composition Containing Stability-Improved Chloromethyl Phosphate Derivatve and Process for Producing Same
US8163902B2 (en) * 2006-11-21 2012-04-24 Rigel Pharmaceuticals, Inc. Prodrugs of 2,4-pyrimidinediamine compounds and their uses
UA108077C2 (xx) 2009-07-02 2015-03-25 Синтез динатрієвої солі n4-(2,2-диметил-4-$(дигідрофосфонокси)метил]-3-оксо-5-піридо$1,4]оксазин-6-іл)-5-фтор-n2-(3,4,5-триметоксифеніл)-2,4-піримідиндіаміну

Also Published As

Publication number Publication date
CN102482305B (zh) 2016-07-13
CA2766801C (en) 2018-03-13
US20110003986A1 (en) 2011-01-06
CN102482305A (zh) 2012-05-30
US20130274499A1 (en) 2013-10-17
HRP20160319T1 (hr) 2016-04-22
AU2010266213A1 (en) 2012-02-02
SI2448950T1 (sl) 2016-05-31
JP5739882B2 (ja) 2015-06-24
HUE027212T2 (en) 2016-10-28
RS54679B1 (sr) 2016-08-31
WO2011002999A1 (en) 2011-01-06
EP2448950A1 (en) 2012-05-09
AU2010266213B2 (en) 2015-06-18
CY1117489T1 (el) 2017-04-26
EP2448950B1 (en) 2016-01-13
DK2448950T3 (en) 2016-04-04
US8691798B2 (en) 2014-04-08
SMT201600084B (it) 2016-04-29
EA021657B1 (ru) 2015-08-31
US8481724B2 (en) 2013-07-09
CA2766801A1 (en) 2011-01-06
US8299242B2 (en) 2012-10-30
EA201270114A1 (ru) 2012-05-30
ME02388B (me) 2016-09-20
PL2448950T3 (pl) 2016-06-30
SG176799A1 (en) 2012-01-30
US20130018185A1 (en) 2013-01-17
UA108077C2 (xx) 2015-03-25
HK1169996A1 (zh) 2013-02-15
ES2565985T3 (es) 2016-04-08
JP2012532143A (ja) 2012-12-13

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Legal Events

Date Code Title Description
B06T Formal requirements before examination [chapter 6.20 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B12B Appeal against refusal [chapter 12.2 patent gazette]