BRPI1011043B8 - fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, seus usos e seu processo de preparação, e composição farmacêutica - Google Patents

fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, seus usos e seu processo de preparação, e composição farmacêutica

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Publication number
BRPI1011043B8
BRPI1011043B8 BRPI1011043A BRPI1011043A BRPI1011043B8 BR PI1011043 B8 BRPI1011043 B8 BR PI1011043B8 BR PI1011043 A BRPI1011043 A BR PI1011043A BR PI1011043 A BRPI1011043 A BR PI1011043A BR PI1011043 B8 BRPI1011043 B8 BR PI1011043B8
Authority
BR
Brazil
Prior art keywords
phenylureas
pharmaceutical composition
preparation process
receptor ligands
vanilloid receptor
Prior art date
Application number
BRPI1011043A
Other languages
English (en)
Inventor
Lesch Bernhard
John Saunders Derek
Bahrenberg Gregor
Stockhausen Hannelore
De Vry Jean
Lee Jeewoo
Schiene Klaus
Kim Myeon-Seop
Damann Nils
Frank Robert
Frormann Sven
Christoph Thomas
Kim Yong-Soo
Original Assignee
Gruenenthal Gmbh
Medifron Dbt Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40908456&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI1011043(B8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal Gmbh, Medifron Dbt Inc filed Critical Gruenenthal Gmbh
Publication of BRPI1011043A2 publication Critical patent/BRPI1011043A2/pt
Publication of BRPI1011043A8 publication Critical patent/BRPI1011043A8/pt
Publication of BRPI1011043B1 publication Critical patent/BRPI1011043B1/pt
Publication of BRPI1011043B8 publication Critical patent/BRPI1011043B8/pt

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Abstract

compostos de fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, sua composição farmacêutica, seu uso e seu processo de preparação. a presente invenção refere-se as fenilureias e fenilamidas substituídas, aos processos para a preparação das mesmas, as composições farmacêuticas contendo estes compostos e também ao emprego destes compostos para preparar composições farmacêuticas.
BRPI1011043A 2009-05-07 2010-05-06 fenilureias e fenilamidas substituídas como ligantes de receptor de vaniloide, seus usos e seu processo de preparação, e composição farmacêutica BRPI1011043B8 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US17628409P 2009-05-07 2009-05-07
EP09006237 2009-05-07
US61/176,284 2009-05-07
EP09006237.3 2009-05-07
PCT/EP2010/002786 WO2010127856A1 (en) 2009-05-07 2010-05-06 Substituted phenyllureas and phenylamides as vanilloid receptor ligands

Publications (4)

Publication Number Publication Date
BRPI1011043A2 BRPI1011043A2 (pt) 2016-09-13
BRPI1011043A8 BRPI1011043A8 (pt) 2017-09-12
BRPI1011043B1 BRPI1011043B1 (pt) 2020-10-13
BRPI1011043B8 true BRPI1011043B8 (pt) 2021-05-25

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US20100331381A1 (en) 2010-12-30
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BRPI1011043A8 (pt) 2017-09-12
NZ595759A (en) 2014-03-28
CO6440569A2 (es) 2012-05-15
CN102428071A (zh) 2012-04-25
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WO2010127856A1 (en) 2010-11-11
US20140142143A1 (en) 2014-05-22
PE20120374A1 (es) 2012-05-13
TW201043603A (en) 2010-12-16
AR076752A1 (es) 2011-07-06
CN106243037A (zh) 2016-12-21
KR101746016B1 (ko) 2017-06-14
BRPI1011043A2 (pt) 2016-09-13
ECSP11011433A (es) 2011-12-30
TWI491595B (zh) 2015-07-11
RU2553392C2 (ru) 2015-06-10
EP2427435B1 (en) 2017-06-14
ES2640257T3 (es) 2017-11-02
MX2011011797A (es) 2011-11-29
US8592471B2 (en) 2013-11-26
BRPI1011043B1 (pt) 2020-10-13
EP2427435A1 (en) 2012-03-14
CA2759951A1 (en) 2010-11-11
US20150011592A9 (en) 2015-01-08
ZA201107706B (en) 2014-03-26
CA2759951C (en) 2017-05-02
US9120756B2 (en) 2015-09-01
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