BRPI0619868A8 - Dispersão sólida compreendendo um ingrediente ativo tendo um ponto de fusão baixo e comprimido para administração oral compreendendo o mesmo - Google Patents
Dispersão sólida compreendendo um ingrediente ativo tendo um ponto de fusão baixo e comprimido para administração oral compreendendo o mesmoInfo
- Publication number
- BRPI0619868A8 BRPI0619868A8 BRPI0619868A BRPI0619868A BRPI0619868A8 BR PI0619868 A8 BRPI0619868 A8 BR PI0619868A8 BR PI0619868 A BRPI0619868 A BR PI0619868A BR PI0619868 A BRPI0619868 A BR PI0619868A BR PI0619868 A8 BRPI0619868 A8 BR PI0619868A8
- Authority
- BR
- Brazil
- Prior art keywords
- solid dispersion
- active ingredient
- melting point
- oral administration
- same
- Prior art date
Links
- 239000007962 solid dispersion Substances 0.000 title abstract 4
- 239000004480 active ingredient Substances 0.000 title abstract 3
- 230000008018 melting Effects 0.000 title abstract 3
- 238000002844 melting Methods 0.000 title abstract 3
- 230000002745 absorbent Effects 0.000 abstract 1
- 239000002250 absorbent Substances 0.000 abstract 1
- 230000002035 prolonged effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/143—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR10-2005-0124386 | 2005-12-16 | ||
| KR20050124386 | 2005-12-16 | ||
| PCT/KR2006/005526 WO2007069874A1 (en) | 2005-12-16 | 2006-12-18 | Solid dispersion comprising an active ingredient having a low melting point and tablet for oral administration comprising same |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0619868A2 BRPI0619868A2 (pt) | 2011-10-25 |
| BRPI0619868A8 true BRPI0619868A8 (pt) | 2016-06-07 |
Family
ID=38163142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0619868A BRPI0619868A8 (pt) | 2005-12-16 | 2006-12-18 | Dispersão sólida compreendendo um ingrediente ativo tendo um ponto de fusão baixo e comprimido para administração oral compreendendo o mesmo |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20080292702A1 (enExample) |
| EP (1) | EP1968542B1 (enExample) |
| JP (1) | JP2009519326A (enExample) |
| CN (1) | CN101330904B (enExample) |
| AU (1) | AU2006325658B2 (enExample) |
| BR (1) | BRPI0619868A8 (enExample) |
| CA (1) | CA2633266C (enExample) |
| ES (1) | ES2429097T3 (enExample) |
| IL (1) | IL191804A0 (enExample) |
| NO (1) | NO339674B1 (enExample) |
| NZ (1) | NZ569813A (enExample) |
| RU (1) | RU2403013C2 (enExample) |
| WO (1) | WO2007069874A1 (enExample) |
| ZA (1) | ZA200806138B (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA06002731A (es) | 2003-09-11 | 2006-06-05 | Xenoport Inc | Tratamiento y/o prevencion de incontinencia urinaria utilizando profarmacos de analogos de gaba. |
| KR101005391B1 (ko) * | 2008-07-22 | 2010-12-30 | 한국콜마 주식회사 | 덱시부프로펜 함유 서방출성 시럽제 및 그의 제조방법 |
| KR101067224B1 (ko) * | 2008-07-22 | 2011-09-22 | 한국콜마 주식회사 | 이부프로펜 함유 서방출성 시럽제 및 그의 제조방법 |
| CN101961306B (zh) * | 2009-07-24 | 2011-11-09 | 北京化工大学 | 一种低熔点药物固体分散体的制备方法 |
| CN102144982B (zh) * | 2011-03-30 | 2012-12-12 | 江苏神龙药业有限公司 | 一种米诺膦酸片及其制备方法 |
| CN102406940B (zh) * | 2011-11-01 | 2013-07-03 | 温州大学 | 一种纳米级片状羧甲基淀粉钠在固体分散体中的应用 |
| WO2013154511A1 (en) * | 2012-04-13 | 2013-10-17 | Mahmut Bilgic | Film tablet formulations comprising dexibuprofen |
| UY36046A (es) | 2014-03-26 | 2015-10-30 | Millennium Pharm Inc | Formulaciones farmacéuticas, procesos para la preparación y métodos de uso |
| JP6647902B2 (ja) * | 2015-10-30 | 2020-02-14 | 株式会社ファンケル | 徐放性顆粒剤 |
| CN106265522A (zh) * | 2016-08-30 | 2017-01-04 | 铜陵翔宇商贸有限公司 | 布洛芬‑pvp共沉淀物及其制备方法 |
| JP7147262B2 (ja) * | 2017-05-23 | 2022-10-05 | 大正製薬株式会社 | 固形製剤 |
| JP7109255B2 (ja) * | 2017-05-23 | 2022-07-29 | ライオン株式会社 | 粉砕物の製造方法及び錠剤の製造方法 |
| EP3658123A4 (en) * | 2017-07-24 | 2021-04-28 | Acryspharm LLC | PHARMACEUTICAL COMPOSITIONS WITH A HIGH DRUG LOAD |
| RU2685294C1 (ru) * | 2018-05-10 | 2019-04-17 | Общество с ограниченной ответственностью "ДИНОН" (ООО "ДИНОН") | Поглотитель, способ его приготовления (варианты) и способ удаления диоксида углерода из газовых смесей |
| CN112263567B (zh) * | 2020-10-19 | 2022-05-03 | 南京易亨制药有限公司 | 一种布洛芬缓释胶囊及制备方法 |
| CN117363320B (zh) * | 2023-12-07 | 2024-02-13 | 黑龙江省鑫博鑫交通科技有限公司 | 一种公路用融雪剂及其制备方法 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56120616A (en) * | 1980-02-27 | 1981-09-22 | Kaken Pharmaceut Co Ltd | Ibuprofen-containing granule, its preparation, and internal medicine comprising it |
| GB8601204D0 (en) * | 1986-01-18 | 1986-02-19 | Boots Co Plc | Therapeutic agents |
| CH669523A5 (enExample) * | 1986-06-25 | 1989-03-31 | Mepha Ag | |
| US4806359A (en) * | 1987-04-22 | 1989-02-21 | Mcneilab, Inc. | Iburprofen sustained release matrix and process |
| DE19509807A1 (de) * | 1995-03-21 | 1996-09-26 | Basf Ag | Verfahren zur Herstellung von Wirkstoffzubereitungen in Form einer festen Lösung des Wirkstoffs in einer Polymermatrix sowie mit diesem Verfahren hergestellte Wirkstoffzubereitungen |
| IE80467B1 (en) * | 1995-07-03 | 1998-07-29 | Elan Corp Plc | Controlled release formulations for poorly soluble drugs |
| US6391338B1 (en) * | 1995-09-07 | 2002-05-21 | Biovail Technologies Ltd. | System for rendering substantially non-dissoluble bio-affecting agents bio-available |
| DE19536394A1 (de) * | 1995-09-29 | 1997-04-03 | Basf Ag | Feste Arzneiformen, erhältlich durch Extrusion einer Isomalt enthaltenden Polymer-Wirkstoff-Schmelze |
| DE69739165D1 (de) * | 1996-07-08 | 2009-01-29 | Penwest Pharmaceuticals Co | Matrix mit verzögerter freisetzung für hochdosierte unlösliche arzneistoffe |
| US6787157B1 (en) * | 1998-03-10 | 2004-09-07 | Abbott Laboratories | Multiphase active ingredient-containing formulations |
| US6183779B1 (en) * | 1999-03-22 | 2001-02-06 | Pharmascience Inc. | Stabilized pharmaceutical composition of a nonsteroidal anti-inflammatory agent and a prostaglandin |
| RU2246294C2 (ru) * | 1999-12-09 | 2005-02-20 | Дзе Бутс Компани ПЛС | Терапевтические средства |
| GB0113839D0 (en) * | 2001-06-07 | 2001-08-01 | Boots Co Plc | Therapeutic agents |
-
2006
- 2006-12-18 AU AU2006325658A patent/AU2006325658B2/en not_active Ceased
- 2006-12-18 CA CA2633266A patent/CA2633266C/en not_active Expired - Fee Related
- 2006-12-18 ZA ZA200806138A patent/ZA200806138B/xx unknown
- 2006-12-18 WO PCT/KR2006/005526 patent/WO2007069874A1/en not_active Ceased
- 2006-12-18 US US12/097,299 patent/US20080292702A1/en not_active Abandoned
- 2006-12-18 NZ NZ569813A patent/NZ569813A/en not_active IP Right Cessation
- 2006-12-18 ES ES06824193T patent/ES2429097T3/es active Active
- 2006-12-18 RU RU2008129041/15A patent/RU2403013C2/ru not_active IP Right Cessation
- 2006-12-18 EP EP06824193.4A patent/EP1968542B1/en not_active Not-in-force
- 2006-12-18 JP JP2008545503A patent/JP2009519326A/ja active Pending
- 2006-12-18 CN CN2006800474904A patent/CN101330904B/zh not_active Expired - Fee Related
- 2006-12-18 BR BRPI0619868A patent/BRPI0619868A8/pt not_active IP Right Cessation
-
2008
- 2008-05-29 IL IL191804A patent/IL191804A0/en unknown
- 2008-07-15 NO NO20083151A patent/NO339674B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2006325658A1 (en) | 2007-06-21 |
| EP1968542A4 (en) | 2010-06-02 |
| CA2633266C (en) | 2011-08-02 |
| IL191804A0 (en) | 2008-12-29 |
| JP2009519326A (ja) | 2009-05-14 |
| HK1126671A1 (en) | 2009-09-11 |
| NO339674B1 (no) | 2017-01-23 |
| AU2006325658B2 (en) | 2010-04-08 |
| RU2403013C2 (ru) | 2010-11-10 |
| BRPI0619868A2 (pt) | 2011-10-25 |
| ZA200806138B (en) | 2009-11-25 |
| CA2633266A1 (en) | 2007-06-21 |
| ES2429097T3 (es) | 2013-11-13 |
| NZ569813A (en) | 2011-07-29 |
| CN101330904B (zh) | 2012-04-18 |
| RU2008129041A (ru) | 2010-01-27 |
| EP1968542A1 (en) | 2008-09-17 |
| EP1968542B1 (en) | 2013-08-14 |
| NO20083151L (no) | 2008-09-05 |
| WO2007069874A1 (en) | 2007-06-21 |
| US20080292702A1 (en) | 2008-11-27 |
| CN101330904A (zh) | 2008-12-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25A | Requested transfer of rights approved |
Owner name: HANMI HOLDINGS CO., LTD. (KR) Free format text: TRANSFERIDO DE: HANMI PHARM. CO., LTD. |
|
| B25D | Requested change of name of applicant approved |
Owner name: HANMI SCIENCE CO., LTD. (KR) |
|
| B25G | Requested change of headquarter approved |
Owner name: HANMI SCIENCE CO., LTD. (KR) |
|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 12A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2494 DE 23-10-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |