BRPI0614843A2 - derivados de piperazina e piperidina, composição farmacêutica, método para preparar composições farmacêuticas, uso de um composto, e, processo para a preparação de composto - Google Patents

derivados de piperazina e piperidina, composição farmacêutica, método para preparar composições farmacêuticas, uso de um composto, e, processo para a preparação de composto Download PDF

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Publication number
BRPI0614843A2
BRPI0614843A2 BRPI0614843-3A BRPI0614843A BRPI0614843A2 BR PI0614843 A2 BRPI0614843 A2 BR PI0614843A2 BR PI0614843 A BRPI0614843 A BR PI0614843A BR PI0614843 A2 BRPI0614843 A2 BR PI0614843A2
Authority
BR
Brazil
Prior art keywords
compound
formula
disorders
compounds
oxide
Prior art date
Application number
BRPI0614843-3A
Other languages
English (en)
Portuguese (pt)
Inventor
Theodorus S M Koopman
Hendrik J Koster
Amsterdam Peter H Van
Marinus Verhage
Andrew C Mccreary
Mayke B Hesselink
Gustaaf J M Scharrenburg
Roelof W Feenstra
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Priority claimed from PCT/EP2006/065477 external-priority patent/WO2007023141A1/en
Publication of BRPI0614843A2 publication Critical patent/BRPI0614843A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0614843-3A 2005-08-22 2006-08-21 derivados de piperazina e piperidina, composição farmacêutica, método para preparar composições farmacêuticas, uso de um composto, e, processo para a preparação de composto BRPI0614843A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05107671.9 2005-08-22
EP05107671 2005-08-22
PCT/EP2006/065477 WO2007023141A1 (en) 2005-08-22 2006-08-21 N-oxides as prodrugs of piperazine & piperidine derivatives

Publications (1)

Publication Number Publication Date
BRPI0614843A2 true BRPI0614843A2 (pt) 2012-12-04

Family

ID=35502590

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0614843-3A BRPI0614843A2 (pt) 2005-08-22 2006-08-21 derivados de piperazina e piperidina, composição farmacêutica, método para preparar composições farmacêuticas, uso de um composto, e, processo para a preparação de composto

Country Status (7)

Country Link
CN (1) CN101248053B (zh)
AR (1) AR058022A1 (zh)
BR (1) BRPI0614843A2 (zh)
HK (1) HK1120261A1 (zh)
TW (1) TW200738656A (zh)
UA (1) UA94718C2 (zh)
ZA (1) ZA200800741B (zh)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE503170A (zh) * 1975-09-02
NZ331860A (en) * 1996-03-29 2000-04-28 Duphar Int Res Piperazine and piperidine compounds with affinity for both dopamine D2 and seratonin 5-HT1A receptors
UA71590C2 (en) * 1998-11-13 2004-12-15 Duphar Int Res Piperazine and piperidine derivatives
DZ3370A1 (fr) * 2000-05-12 2001-11-15 Solvay Pharm Bv Composes de piperazine et piperidine
PL214274B1 (pl) * 2002-01-16 2013-07-31 Movetis N V N-Tlenek prukaloprydu, sposób jego wytwarzania i zastosowanie oraz zawierająca go kompozycja i sposób jej wytwarzania

Also Published As

Publication number Publication date
AR058022A1 (es) 2008-01-23
CN101248053A (zh) 2008-08-20
CN101248053B (zh) 2011-06-01
ZA200800741B (en) 2009-01-28
UA94718C2 (ru) 2011-06-10
TW200738656A (en) 2007-10-16
HK1120261A1 (en) 2009-03-27

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B06G Technical and formal requirements: other requirements [chapter 6.7 patent gazette]

Free format text: SOLICITA-SE A REGULARIZACAO DA PROCURACAO, UMA VEZ QUE BASEADO NO ARTIGO 216 1O DA LPI, O DOCUMENTO DE PROCURACAO DEVE SER APRESENTADO NO ORIGINAL, TRASLADO OU FOTOCOPIA AUTENTICADA.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

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B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2256 DE 01/04/2014.