HK1120261A1 - N-oxides as prodrugs of piperazine & piperidine derivatives - Google Patents

N-oxides as prodrugs of piperazine & piperidine derivatives

Info

Publication number
HK1120261A1
HK1120261A1 HK08112134.4A HK08112134A HK1120261A1 HK 1120261 A1 HK1120261 A1 HK 1120261A1 HK 08112134 A HK08112134 A HK 08112134A HK 1120261 A1 HK1120261 A1 HK 1120261A1
Authority
HK
Hong Kong
Prior art keywords
prodrugs
piperazine
oxides
piperidine derivatives
piperidine
Prior art date
Application number
HK08112134.4A
Other languages
English (en)
Inventor
Theodorus S M Koopman
Hendrik J Koster
Peter H Van Amsterdam
Roelof W Feenstra
Marinus Verhage
Andrew C Mccreary
Mayke B Hesselink
Gustaaf J M Van Scharrenburg
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2006/065477 external-priority patent/WO2007023141A1/en
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Publication of HK1120261A1 publication Critical patent/HK1120261A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK08112134.4A 2005-08-22 2008-11-06 N-oxides as prodrugs of piperazine & piperidine derivatives HK1120261A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05107671 2005-08-22
PCT/EP2006/065477 WO2007023141A1 (en) 2005-08-22 2006-08-21 N-oxides as prodrugs of piperazine & piperidine derivatives

Publications (1)

Publication Number Publication Date
HK1120261A1 true HK1120261A1 (en) 2009-03-27

Family

ID=35502590

Family Applications (1)

Application Number Title Priority Date Filing Date
HK08112134.4A HK1120261A1 (en) 2005-08-22 2008-11-06 N-oxides as prodrugs of piperazine & piperidine derivatives

Country Status (7)

Country Link
CN (1) CN101248053B (zh)
AR (1) AR058022A1 (zh)
BR (1) BRPI0614843A2 (zh)
HK (1) HK1120261A1 (zh)
TW (1) TW200738656A (zh)
UA (1) UA94718C2 (zh)
ZA (1) ZA200800741B (zh)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE503170A (zh) * 1975-09-02
NZ331860A (en) * 1996-03-29 2000-04-28 Duphar Int Res Piperazine and piperidine compounds with affinity for both dopamine D2 and seratonin 5-HT1A receptors
UA71590C2 (en) * 1998-11-13 2004-12-15 Duphar Int Res Piperazine and piperidine derivatives
DZ3370A1 (fr) * 2000-05-12 2001-11-15 Solvay Pharm Bv Composes de piperazine et piperidine
PL214274B1 (pl) * 2002-01-16 2013-07-31 Movetis N V N-Tlenek prukaloprydu, sposób jego wytwarzania i zastosowanie oraz zawierająca go kompozycja i sposób jej wytwarzania

Also Published As

Publication number Publication date
AR058022A1 (es) 2008-01-23
CN101248053A (zh) 2008-08-20
CN101248053B (zh) 2011-06-01
ZA200800741B (en) 2009-01-28
UA94718C2 (ru) 2011-06-10
TW200738656A (en) 2007-10-16
BRPI0614843A2 (pt) 2012-12-04

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20150821