BRPI0608454A2 - 8-n-benzimidazóis substituìdos com aminocarbonila, método para sua produção e seu uso como medicamentos - Google Patents
8-n-benzimidazóis substituìdos com aminocarbonila, método para sua produção e seu uso como medicamentos Download PDFInfo
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- BRPI0608454A2 BRPI0608454A2 BRPI0608454-0A BRPI0608454A BRPI0608454A2 BR PI0608454 A2 BRPI0608454 A2 BR PI0608454A2 BR PI0608454 A BRPI0608454 A BR PI0608454A BR PI0608454 A2 BRPI0608454 A2 BR PI0608454A2
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- Prior art keywords
- alkyl
- aryl
- alkylene
- heterocyclyl
- cycloalkyl
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Hematology (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005012873A DE102005012873B4 (de) | 2005-03-19 | 2005-03-19 | Aminocarbonyl substituierte 8-N-Benzimidazole, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| PCT/EP2006/002056 WO2006099941A1 (de) | 2005-03-19 | 2006-03-07 | Aminocarbonyl substituierte 8-n-benzimidazole, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0608454A2 true BRPI0608454A2 (pt) | 2010-01-05 |
Family
ID=36592884
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0608454-0A BRPI0608454A2 (pt) | 2005-03-19 | 2006-03-07 | 8-n-benzimidazóis substituìdos com aminocarbonila, método para sua produção e seu uso como medicamentos |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8138207B2 (cg-RX-API-DMAC10.html) |
| EP (1) | EP1863789B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP2008533065A (cg-RX-API-DMAC10.html) |
| AU (1) | AU2006226638A1 (cg-RX-API-DMAC10.html) |
| BR (1) | BRPI0608454A2 (cg-RX-API-DMAC10.html) |
| CA (1) | CA2602233A1 (cg-RX-API-DMAC10.html) |
| DE (1) | DE102005012873B4 (cg-RX-API-DMAC10.html) |
| IL (1) | IL185804A0 (cg-RX-API-DMAC10.html) |
| MX (1) | MX2007010837A (cg-RX-API-DMAC10.html) |
| WO (1) | WO2006099941A1 (cg-RX-API-DMAC10.html) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2010500300A (ja) | 2006-08-08 | 2010-01-07 | サノフィ−アベンティス | アリールアミノアリール−アルキル−置換イミダゾリジン−２，４−ジオン、それらの製造法、それらの化合物を含有する薬剤、およびそれらの使用 |
| DE102007005045B4 (de) | 2007-01-26 | 2008-12-18 | Sanofi-Aventis | Phenothiazin Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| WO2010003624A2 (en) | 2008-07-09 | 2010-01-14 | Sanofi-Aventis | Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof |
| WO2010068601A1 (en) | 2008-12-08 | 2010-06-17 | Sanofi-Aventis | A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof |
| SG178880A1 (en) | 2009-08-26 | 2012-04-27 | Sanofi Sa | Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use |
| WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
| EP2582709B1 (de) | 2010-06-18 | 2018-01-24 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
| US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
| TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
| TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
| TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
| US8846666B2 (en) | 2011-03-08 | 2014-09-30 | Sanofi | Oxathiazine derivatives which are substituted with benzyl or heteromethylene groups, method for producing them, their use as medicine and drug containing said derivatives and the use thereof |
| WO2012120054A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| EP2683698B1 (de) | 2011-03-08 | 2017-10-04 | Sanofi | Mit adamantan- oder noradamantan substituierte benzyl-oxathiazinderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
| EP2766349B1 (de) | 2011-03-08 | 2016-06-01 | Sanofi | Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120056A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| EP2683703B1 (de) | 2011-03-08 | 2015-05-27 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| EP2683704B1 (de) | 2011-03-08 | 2014-12-17 | Sanofi | Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| US8809324B2 (en) | 2011-03-08 | 2014-08-19 | Sanofi | Substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof |
| WO2012120055A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| EP2760862B1 (en) | 2011-09-27 | 2015-10-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| CN105142621A (zh) | 2012-10-24 | 2015-12-09 | 国家健康科学研究所 | 用于预防或治疗糖尿病和促进β-细胞存活的TPL2激酶抑制剂 |
| EP3273981B1 (en) | 2015-03-24 | 2020-04-29 | INSERM - Institut National de la Santé et de la Recherche Médicale | Method and pharmaceutical composition for use in the treatment of diabetes |
| BR112021002207A2 (pt) | 2018-08-10 | 2021-05-04 | Diapin Therapeutics, Llc | tri-peptídeos e tratamento de distúrbios metabólicos, cardiovasculares e inflamatórios |
| LT3860998T (lt) | 2018-10-05 | 2024-06-25 | Annapurna Bio Inc. | Junginiai ir kompozicijos, skirti gydyti būkles, susijusias su apj receptoriaus aktyvumu |
| TW202329937A (zh) | 2021-12-03 | 2023-08-01 | 美商英塞特公司 | 雙環胺ｃｋ１２抑制劑 |
| US12084453B2 (en) | 2021-12-10 | 2024-09-10 | Incyte Corporation | Bicyclic amines as CDK12 inhibitors |
Family Cites Families (7)
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| PE27997A1 (es) * | 1994-04-29 | 1997-09-20 | Lilly Co Eli | Antagonistas de receptores de taquicininas |
| US6025372A (en) * | 1997-04-04 | 2000-02-15 | Merck & Co., Inc. | Somatostatin agonists |
| AUPP150098A0 (en) * | 1998-01-27 | 1998-02-19 | Fujisawa Pharmaceutical Co., Ltd. | Benzamide derivatives |
| US6340681B1 (en) * | 1999-07-16 | 2002-01-22 | Pfizer Inc | 2-benzimidazolylamine compounds as ORL-1-receptor agonists |
| JP2004515496A (ja) * | 2000-12-07 | 2004-05-27 | アストラゼネカ・アクチエボラーグ | ベンズイミダゾール治療剤 |
| EP1553089B1 (en) * | 2002-07-30 | 2009-09-30 | Banyu Pharmaceutical Co., Ltd. | Antagonist of melanin-concentrating hormone receptor comprising benzimidazole derivative as active ingredient |
| WO2007069053A1 (en) * | 2005-12-14 | 2007-06-21 | Pfizer Products Inc. | Benzimidazole antagonists of the h-3 receptor |
-
2005
- 2005-03-19 DE DE102005012873A patent/DE102005012873B4/de not_active Expired - Fee Related
-
2006
- 2006-03-07 JP JP2008501195A patent/JP2008533065A/ja not_active Abandoned
- 2006-03-07 BR BRPI0608454-0A patent/BRPI0608454A2/pt not_active Application Discontinuation
- 2006-03-07 AU AU2006226638A patent/AU2006226638A1/en not_active Abandoned
- 2006-03-07 EP EP06723255.3A patent/EP1863789B1/de not_active Expired - Lifetime
- 2006-03-07 CA CA002602233A patent/CA2602233A1/en not_active Abandoned
- 2006-03-07 WO PCT/EP2006/002056 patent/WO2006099941A1/de not_active Ceased
- 2006-03-07 MX MX2007010837A patent/MX2007010837A/es not_active Application Discontinuation
-
2007
- 2007-09-06 IL IL185804A patent/IL185804A0/en unknown
- 2007-09-14 US US11/855,227 patent/US8138207B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP1863789B1 (de) | 2014-08-20 |
| CA2602233A1 (en) | 2006-09-28 |
| EP1863789A1 (de) | 2007-12-12 |
| DE102005012873B4 (de) | 2007-05-03 |
| IL185804A0 (en) | 2008-01-06 |
| DE102005012873A1 (de) | 2006-09-28 |
| JP2008533065A (ja) | 2008-08-21 |
| WO2006099941A8 (de) | 2006-11-09 |
| US20080090869A1 (en) | 2008-04-17 |
| US8138207B2 (en) | 2012-03-20 |
| AU2006226638A1 (en) | 2006-09-28 |
| MX2007010837A (es) | 2007-11-09 |
| WO2006099941A1 (de) | 2006-09-28 |
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| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |