BRPI0516507A - produto, processo e intermediários de preparação de derivados de azetidina - Google Patents
produto, processo e intermediários de preparação de derivados de azetidinaInfo
- Publication number
- BRPI0516507A BRPI0516507A BRPI0516507-5A BRPI0516507A BRPI0516507A BR PI0516507 A BRPI0516507 A BR PI0516507A BR PI0516507 A BRPI0516507 A BR PI0516507A BR PI0516507 A BRPI0516507 A BR PI0516507A
- Authority
- BR
- Brazil
- Prior art keywords
- intermediates
- preparation product
- derivative preparation
- azetidine derivative
- azetidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Child & Adolescent Psychology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Psychology (AREA)
- Immunology (AREA)
- Hospice & Palliative Care (AREA)
- Reproductive Health (AREA)
- Epidemiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PRODUTO, PROCESSO E INTERMEDIáRIOS DE PREPARAçãO DE DERIVADOS DE AZETIDINA. A presente invenção refere-se a um novo processo de preparação de derivados de azetidina tais como a N-{1-¢bis-(4-clorofenil)metil!azetidin-3-iI}-N-quinol-6-iI-metilsulfonamid a e de seu dicloridrato e da N-{1 -¢bis-(4-clorofenil)-metil!azetidin-3-iI}-N-(3, 5 difluorfenil) metilsulfonamida.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0410844A FR2876688B1 (fr) | 2004-10-14 | 2004-10-14 | Nouveau produit, procede et intermediaires de preparation de derives d'azetidine |
PCT/FR2005/002490 WO2006040465A2 (fr) | 2004-10-14 | 2005-10-10 | Nouveau produit, procede et intermediaires de preparation de derives d'azetidine |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0516507A true BRPI0516507A (pt) | 2008-09-16 |
Family
ID=34954419
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0516507-5A BRPI0516507A (pt) | 2004-10-14 | 2005-10-10 | produto, processo e intermediários de preparação de derivados de azetidina |
Country Status (21)
Country | Link |
---|---|
US (1) | US7687493B2 (pt) |
EP (1) | EP1805167A2 (pt) |
JP (1) | JP2008516932A (pt) |
KR (1) | KR20070063544A (pt) |
CN (1) | CN101039931A (pt) |
AR (1) | AR051390A1 (pt) |
AU (1) | AU2005293454A1 (pt) |
BR (1) | BRPI0516507A (pt) |
CA (1) | CA2583992A1 (pt) |
EA (1) | EA011408B1 (pt) |
EC (1) | ECSP077332A (pt) |
FR (1) | FR2876688B1 (pt) |
IL (1) | IL181904A0 (pt) |
MA (1) | MA29513B1 (pt) |
MX (1) | MX2007003923A (pt) |
NO (1) | NO20072192L (pt) |
SG (1) | SG155193A1 (pt) |
TN (1) | TNSN07097A1 (pt) |
TW (1) | TW200630358A (pt) |
WO (1) | WO2006040465A2 (pt) |
ZA (1) | ZA200702528B (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN113045539B (zh) * | 2021-03-30 | 2021-12-07 | 苏州大学 | 2-(4,4-二氯-1-(8-喹啉基)-2-氮杂环丁基)羧酸酯衍生物的制备方法 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8709887D0 (en) * | 1987-04-27 | 1987-06-03 | Univ Alberta | Alkyl azodicarboxylates |
US5530134A (en) * | 1994-09-06 | 1996-06-25 | Synphar Laboratories Inc. | Synthesis of anabaseine, salts and derivatives thereof |
FR2805817B1 (fr) * | 2000-03-03 | 2002-04-26 | Aventis Pharma Sa | Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation |
US6355631B1 (en) * | 2000-03-03 | 2002-03-12 | Aventis Pharma S.A. | Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and their preparation |
ES2334858T3 (es) * | 2000-08-10 | 2010-03-16 | Mitsubishi Tanabe Pharma Corporation | Derivados de prolina y uso de los mismos como farmacos. |
CN101407471A (zh) * | 2003-08-29 | 2009-04-15 | 小野药品工业株式会社 | 能够结合s1p受体的化合物及其药物用途 |
-
2004
- 2004-10-14 FR FR0410844A patent/FR2876688B1/fr not_active Expired - Fee Related
-
2005
- 2005-10-10 EP EP05809232A patent/EP1805167A2/fr not_active Withdrawn
- 2005-10-10 JP JP2007536214A patent/JP2008516932A/ja active Pending
- 2005-10-10 KR KR1020077008461A patent/KR20070063544A/ko not_active Application Discontinuation
- 2005-10-10 SG SG200905236-6A patent/SG155193A1/en unknown
- 2005-10-10 WO PCT/FR2005/002490 patent/WO2006040465A2/fr active Application Filing
- 2005-10-10 MX MX2007003923A patent/MX2007003923A/es active IP Right Grant
- 2005-10-10 BR BRPI0516507-5A patent/BRPI0516507A/pt not_active IP Right Cessation
- 2005-10-10 AU AU2005293454A patent/AU2005293454A1/en not_active Withdrawn
- 2005-10-10 ZA ZA200702528A patent/ZA200702528B/xx unknown
- 2005-10-10 CN CNA2005800350837A patent/CN101039931A/zh active Pending
- 2005-10-10 EA EA200700840A patent/EA011408B1/ru not_active IP Right Cessation
- 2005-10-10 CA CA002583992A patent/CA2583992A1/fr not_active Abandoned
- 2005-10-13 AR ARP050104296A patent/AR051390A1/es unknown
- 2005-10-13 TW TW094135607A patent/TW200630358A/zh unknown
-
2007
- 2007-03-13 IL IL181904A patent/IL181904A0/en unknown
- 2007-03-16 TN TNP2007000097A patent/TNSN07097A1/fr unknown
- 2007-03-21 EC EC2007007332A patent/ECSP077332A/es unknown
- 2007-03-22 US US11/689,588 patent/US7687493B2/en not_active Expired - Fee Related
- 2007-04-27 NO NO20072192A patent/NO20072192L/no not_active Application Discontinuation
- 2007-05-11 MA MA29896A patent/MA29513B1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
EP1805167A2 (fr) | 2007-07-11 |
FR2876688A1 (fr) | 2006-04-21 |
WO2006040465A2 (fr) | 2006-04-20 |
EA200700840A1 (ru) | 2007-08-31 |
AU2005293454A1 (en) | 2006-04-20 |
CA2583992A1 (fr) | 2006-04-20 |
ZA200702528B (en) | 2008-07-30 |
TNSN07097A1 (fr) | 2008-06-02 |
ECSP077332A (es) | 2007-04-26 |
WO2006040465A3 (fr) | 2006-08-10 |
CN101039931A (zh) | 2007-09-19 |
MX2007003923A (es) | 2007-06-07 |
JP2008516932A (ja) | 2008-05-22 |
SG155193A1 (en) | 2009-09-30 |
MA29513B1 (fr) | 2008-06-02 |
US20070270463A1 (en) | 2007-11-22 |
NO20072192L (no) | 2007-04-27 |
IL181904A0 (en) | 2007-07-04 |
TW200630358A (en) | 2006-09-01 |
AR051390A1 (es) | 2007-01-10 |
EA011408B1 (ru) | 2009-02-27 |
KR20070063544A (ko) | 2007-06-19 |
US7687493B2 (en) | 2010-03-30 |
FR2876688B1 (fr) | 2007-03-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2160 DE 29/05/2012. |