BRPI0510639A - composto ou um sal ou uma pró-droga farmaceuticamente aceitável do mesmo, composição farmacêutica, métodos de tratar ou prevenir distúrbios, de terapia de reposição hormonal, de abaixar nìveis de colesterol, triglicerìdeos ou ldl, de tratar cognição prejudicada ou prover neuroproteção, de prevenir concepção, de modular ou agonizar especificamente um ou mais receptores de estrogênio e, uso de um composto - Google Patents

composto ou um sal ou uma pró-droga farmaceuticamente aceitável do mesmo, composição farmacêutica, métodos de tratar ou prevenir distúrbios, de terapia de reposição hormonal, de abaixar nìveis de colesterol, triglicerìdeos ou ldl, de tratar cognição prejudicada ou prover neuroproteção, de prevenir concepção, de modular ou agonizar especificamente um ou mais receptores de estrogênio e, uso de um composto

Info

Publication number
BRPI0510639A
BRPI0510639A BRPI0510639-7A BRPI0510639A BRPI0510639A BR PI0510639 A BRPI0510639 A BR PI0510639A BR PI0510639 A BRPI0510639 A BR PI0510639A BR PI0510639 A BRPI0510639 A BR PI0510639A
Authority
BR
Brazil
Prior art keywords
treating
preventing
methods
compound
estrogen receptors
Prior art date
Application number
BRPI0510639-7A
Other languages
English (en)
Inventor
Roger Olsson
Lene Hyldtoft
Fabrice Piu
Magnus Gustafsson
Original Assignee
Acadia Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Acadia Pharm Inc filed Critical Acadia Pharm Inc
Publication of BRPI0510639A publication Critical patent/BRPI0510639A/pt

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Abstract

COMPOSTO OU UM SAL OU UMA PRó-DROGA FARMACEUTICAMENTE ACEITáVEL DO MESMO, COMPOSIçãO FARMACêUTICA, MéTODOS DE TRATAR OU PREVENIR DISTúRBIOS, DE TERAPIA DE REPOSIçãO HORMONAL, DE ABAIXAR NìVEIS DE COLESTEROL, TRIGLICERìDEOS OU LDL, DE TRATAR COGNIçãO PREJUDICADA OU PROVER NEUROPROTEçãO, DE PREVENIR CONCEPçãO, DE MODULAR OU AGONIZAR ESPECIFICAMENTE UM OU MAIS RECEPTORES DE ESTROGêNIO E, USO DE UM COMPOSTO São aqui descritas novos compostos difenílicos e métodos para usar vários compostos difenílicos para tratamento de doenças e distúrbios associados com receptores de estrogênio.
BRPI0510639-7A 2004-05-04 2005-05-03 composto ou um sal ou uma pró-droga farmaceuticamente aceitável do mesmo, composição farmacêutica, métodos de tratar ou prevenir distúrbios, de terapia de reposição hormonal, de abaixar nìveis de colesterol, triglicerìdeos ou ldl, de tratar cognição prejudicada ou prover neuroproteção, de prevenir concepção, de modular ou agonizar especificamente um ou mais receptores de estrogênio e, uso de um composto BRPI0510639A (pt)

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US56833204P 2004-05-04 2004-05-04
PCT/US2005/015221 WO2005108337A2 (en) 2004-05-04 2005-05-03 Compounds with activity at estrogen receptor

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EP (1) EP1747182A2 (pt)
JP (1) JP2007536238A (pt)
KR (1) KR20070028400A (pt)
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EP1747182A2 (en) 2007-01-31
AU2005240609A1 (en) 2005-11-17
KR20070028400A (ko) 2007-03-12
WO2005108337A3 (en) 2005-12-22
JP2007536238A (ja) 2007-12-13
US20050256210A1 (en) 2005-11-17
CN1997618A (zh) 2007-07-11
RU2006142683A (ru) 2008-06-10
ZA200609870B (en) 2009-12-30
MXPA06012705A (es) 2007-03-26
WO2005108337A2 (en) 2005-11-17

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