BRPI0416590A - excipientes em veìculos de distribuição de fármacos - Google Patents

excipientes em veìculos de distribuição de fármacos

Info

Publication number
BRPI0416590A
BRPI0416590A BRPI0416590-0A BRPI0416590A BRPI0416590A BR PI0416590 A BRPI0416590 A BR PI0416590A BR PI0416590 A BRPI0416590 A BR PI0416590A BR PI0416590 A BRPI0416590 A BR PI0416590A
Authority
BR
Brazil
Prior art keywords
polymers
excipients
drug delivery
delivery vehicles
gel compositions
Prior art date
Application number
BRPI0416590-0A
Other languages
English (en)
Original Assignee
Alza Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alza Corp filed Critical Alza Corp
Publication of BRPI0416590A publication Critical patent/BRPI0416590A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/27Growth hormone [GH], i.e. somatotropin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

"EXCIPIENTES EM VEìCULOS DE DISTRIBUIçãO DE FáRMACOS". A presente invenção fornece composições de gel injetáveis para depósito e kits que fornecem um excipiente para modular uma taxa de liberação e estabilizar os agente benéficos. São fornecidos também métodos para administrar e preparar tais sistemas. As composições do gel compreendem polímeros biodegradáveis, bioerodíveis, e solventes imiscíveis em água, em quantidades eficazes para plastificar os polímeros e formar géis com os polímeros. Os excipientes apropriados incluem modificadores de pH, agentes redutores e antioxidantes.
BRPI0416590-0A 2003-11-14 2004-11-12 excipientes em veìculos de distribuição de fármacos BRPI0416590A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US51993603P 2003-11-14 2003-11-14
US10/985,122 US20050106214A1 (en) 2003-11-14 2004-11-10 Excipients in drug delivery vehicles
PCT/US2004/037781 WO2005049069A1 (en) 2003-11-14 2004-11-12 Excipients in drug delivery vehicles

Publications (1)

Publication Number Publication Date
BRPI0416590A true BRPI0416590A (pt) 2007-01-30

Family

ID=34576891

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0416590-0A BRPI0416590A (pt) 2003-11-14 2004-11-12 excipientes em veìculos de distribuição de fármacos

Country Status (12)

Country Link
US (2) US20050106214A1 (pt)
EP (1) EP1691826A4 (pt)
JP (1) JP4916887B2 (pt)
KR (1) KR20060125749A (pt)
AU (2) AU2004291093A1 (pt)
BR (1) BRPI0416590A (pt)
CA (1) CA2545923A1 (pt)
IL (1) IL175602A0 (pt)
MX (1) MXPA06005463A (pt)
NO (1) NO20062780L (pt)
TW (1) TW200529842A (pt)
WO (1) WO2005049069A1 (pt)

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Also Published As

Publication number Publication date
KR20060125749A (ko) 2006-12-06
TW200529842A (en) 2005-09-16
MXPA06005463A (es) 2006-08-11
EP1691826A4 (en) 2012-08-22
US20120177697A1 (en) 2012-07-12
IL175602A0 (en) 2006-09-05
JP4916887B2 (ja) 2012-04-18
WO2005049069A1 (en) 2005-06-02
AU2011201826A1 (en) 2011-05-19
NO20062780L (no) 2006-08-14
CA2545923A1 (en) 2005-06-02
EP1691826A1 (en) 2006-08-23
AU2004291093A1 (en) 2005-06-02
US20050106214A1 (en) 2005-05-19
JP2007511524A (ja) 2007-05-10
AU2011201826B2 (en) 2013-06-13

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.